IL92827A - C63-amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy-teicoplanins, their preparation and pharmaceutical compositions containing them - Google Patents

C63-amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy-teicoplanins, their preparation and pharmaceutical compositions containing them

Info

Publication number
IL92827A
IL92827A IL9282789A IL9282789A IL92827A IL 92827 A IL92827 A IL 92827A IL 9282789 A IL9282789 A IL 9282789A IL 9282789 A IL9282789 A IL 9282789A IL 92827 A IL92827 A IL 92827A
Authority
IL
Israel
Prior art keywords
hydrogen
formula
alkyl
compound
amine
Prior art date
Application number
IL9282789A
Other languages
English (en)
Other versions
IL92827A0 (en
Inventor
Adriano Malabarba
Jurgen Kurt Kettenring
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of IL92827A0 publication Critical patent/IL92827A0/xx
Publication of IL92827A publication Critical patent/IL92827A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
    • C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
    • C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Genetics & Genomics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Electric Stoves And Ranges (AREA)
IL9282789A 1988-12-27 1989-12-20 C63-amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy-teicoplanins, their preparation and pharmaceutical compositions containing them IL92827A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP88121708 1988-12-27

Publications (2)

Publication Number Publication Date
IL92827A0 IL92827A0 (en) 1990-09-17
IL92827A true IL92827A (en) 1994-08-26

Family

ID=8199722

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9282789A IL92827A (en) 1988-12-27 1989-12-20 C63-amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy-teicoplanins, their preparation and pharmaceutical compositions containing them

Country Status (19)

Country Link
EP (1) EP0376041B1 (ru)
JP (1) JPH02221298A (ru)
CN (1) CN1043941A (ru)
AT (1) ATE134646T1 (ru)
AU (1) AU629883B2 (ru)
CA (1) CA2006379A1 (ru)
DE (1) DE68925806T2 (ru)
DK (1) DK171404B1 (ru)
ES (1) ES2083374T3 (ru)
FI (1) FI91076C (ru)
GR (1) GR3020070T3 (ru)
HU (1) HU209939B (ru)
IE (1) IE71942B1 (ru)
IL (1) IL92827A (ru)
NO (1) NO178664C (ru)
NZ (1) NZ231863A (ru)
PT (1) PT92672B (ru)
RU (1) RU2068418C1 (ru)
ZA (1) ZA899772B (ru)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU647122B2 (en) * 1990-05-28 1994-03-17 Gruppo Lepetit S.P.A. C63-amide derivatives of 34-de(acetylglucosaminyl)-34-deoxy- teicoplanin and their use as medicaments against bacteria resistant to glycopeptide antibiotics
US5606036A (en) * 1991-03-27 1997-02-25 Gruppo Lepetit Spa Antibiotic A 40926 ester derivatives
UA41283C2 (uk) * 1991-07-29 2001-09-17 Біосерч Італіа С.П.А. Похідні антибіотику а 40926 та способи їх одержання
US5750509A (en) * 1991-07-29 1998-05-12 Gruppo Lepetit S.P.A. Amide derivatives of antibiotic A 40926
CN1249081C (zh) * 1998-12-23 2006-04-05 施万制药 糖肽衍生物或含有它们的药物组合物
SG87877A1 (en) * 1998-12-23 2002-04-16 Advanced Medicine Inc Glycopeptide derivatives and pharmaceutical compositions containing the same
TWI312785B (en) 2001-08-24 2009-08-01 Theravance Inc Process for preparing vancomycin derivatives
TWI275594B (en) 2001-08-24 2007-03-11 Theravance Inc Process for preparing vancomycin phosphonate derivatives
US20060074014A1 (en) 2002-11-18 2006-04-06 Vicuron Pharmaceuticals Inc. Dalbavancin compositions for treatment of bacterial infections
US7119061B2 (en) 2002-11-18 2006-10-10 Vicuron Pharmaceuticals, Inc. Dalbavancin compositions for treatment of bacterial infections
DK1565201T3 (en) 2002-11-18 2019-02-25 Vicuron Pharmaceuticals Llc METHODS OF ADMINISTRATING DALBAVANCIN TO TREAT Bacterial Infections

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8522574D0 (en) * 1985-09-12 1985-10-16 Lepetit Spa Amides of teicoplanin compounds
GB8529272D0 (en) * 1985-11-28 1986-01-02 Lepetit Spa Teicoplanin derivatives
GB8704847D0 (en) * 1987-03-02 1987-04-08 Lepetit Spa Substituted alkylamides of teicoplanin compounds
GB8711066D0 (en) * 1987-05-11 1987-06-17 Lepetit Spa Teicoplanin derivatives
GB8827202D0 (en) * 1988-11-22 1988-12-29 Lepetit Spa Process for preparing 63-carboxyamides of teicoplanin antibiotics

Also Published As

Publication number Publication date
GR3020070T3 (en) 1996-08-31
NO178664C (no) 1996-05-08
AU4698489A (en) 1990-07-05
HU896772D0 (en) 1990-03-28
NO178664B (no) 1996-01-29
DK640489A (da) 1990-06-28
RU2068418C1 (ru) 1996-10-27
PT92672B (pt) 1996-09-30
DE68925806T2 (de) 1996-09-26
ES2083374T3 (es) 1996-04-16
IE894143L (en) 1990-06-27
DK171404B1 (da) 1996-10-14
DK640489D0 (da) 1989-12-18
IL92827A0 (en) 1990-09-17
EP0376041A3 (en) 1991-11-13
ATE134646T1 (de) 1996-03-15
IE71942B1 (en) 1997-03-12
FI91076B (fi) 1994-01-31
DE68925806D1 (de) 1996-04-04
PT92672A (pt) 1990-06-29
EP0376041B1 (en) 1996-02-28
HUT53376A (en) 1990-10-28
NO895123L (no) 1990-06-28
EP0376041A2 (en) 1990-07-04
FI896199A0 (fi) 1989-12-22
CN1043941A (zh) 1990-07-18
NO895123D0 (no) 1989-12-19
JPH02221298A (ja) 1990-09-04
HU209939B (en) 1994-12-28
CA2006379A1 (en) 1990-06-27
FI91076C (fi) 1994-05-10
NZ231863A (en) 1992-08-26
ZA899772B (en) 1991-01-30
AU629883B2 (en) 1992-10-15

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Legal Events

Date Code Title Description
RH Patent void