IL89480A - אוקסינדול 1,7-אנילאט-3- קארבוקסאמידים ותכשירי רוקחות המכילים אותם - Google Patents

אוקסינדול 1,7-אנילאט-3- קארבוקסאמידים ותכשירי רוקחות המכילים אותם

Info

Publication number
IL89480A
IL89480A IL8948089A IL8948089A IL89480A IL 89480 A IL89480 A IL 89480A IL 8948089 A IL8948089 A IL 8948089A IL 8948089 A IL8948089 A IL 8948089A IL 89480 A IL89480 A IL 89480A
Authority
IL
Israel
Prior art keywords
compound
thiazolyl
carboxamide
phenyl
formula
Prior art date
Application number
IL8948089A
Other languages
English (en)
Other versions
IL89480A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL89480A0 publication Critical patent/IL89480A0/xx
Publication of IL89480A publication Critical patent/IL89480A/he

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/06—Peri-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL8948089A 1988-03-11 1989-03-03 אוקסינדול 1,7-אנילאט-3- קארבוקסאמידים ותכשירי רוקחות המכילים אותם IL89480A (he)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US1988/000781 WO1989008654A1 (en) 1988-03-11 1988-03-11 Pyrroloquinoline and pyrrolophenothiazine carboxamides and related compounds

Publications (2)

Publication Number Publication Date
IL89480A0 IL89480A0 (en) 1989-09-10
IL89480A true IL89480A (he) 1994-04-12

Family

ID=22208596

Family Applications (1)

Application Number Title Priority Date Filing Date
IL8948089A IL89480A (he) 1988-03-11 1989-03-03 אוקסינדול 1,7-אנילאט-3- קארבוקסאמידים ותכשירי רוקחות המכילים אותם

Country Status (15)

Country Link
EP (1) EP0332364A3 (he)
JP (1) JPH0676408B2 (he)
KR (1) KR910002565B1 (he)
AU (1) AU605410B2 (he)
CA (1) CA1335592C (he)
DK (1) DK169723B1 (he)
FI (1) FI96315C (he)
HU (1) HU201757B (he)
IL (1) IL89480A (he)
MY (1) MY104955A (he)
NO (1) NO170418C (he)
NZ (1) NZ228299A (he)
PT (1) PT89954B (he)
WO (1) WO1989008654A1 (he)
ZA (1) ZA891800B (he)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3907388A1 (de) * 1989-03-08 1990-09-13 Kali Chemie Pharma Gmbh Verfahren zur herstellung von indolcarbonsaeurederivaten
JPH06279444A (ja) * 1993-03-31 1994-10-04 Tokyo Tanabe Co Ltd インドリジン誘導体
US6084098A (en) 1999-02-26 2000-07-04 Neurogen Corporation Benzylpiperazinyl and piperidinyl ethanone derivatives: dopamine receptor subtype specific ligands
PL342597A1 (en) * 1998-02-26 2001-06-18 Neurogen Corp Benzylopiperazinylic and benxylopiperidinylic derivatives of ethanone, method of obtaining them and their application as antagonists of dopamine d4 receptor
US6284759B1 (en) 1998-09-30 2001-09-04 Neurogen Corporation 2-piperazinoalkylaminobenzo-azole derivatives: dopamine receptor subtype specific ligands
DE602005020472D1 (de) * 2004-09-09 2010-05-20 Merck Sharp & Dohme Tricyclische anilid-spirohydantoin-cgrp-rezeptorantagonisten
WO2006031676A2 (en) * 2004-09-13 2006-03-23 Merck & Co., Inc. Tricyclic anilide spirohydantoin cgrp receptor antagonists
US7741317B2 (en) * 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
CN108853102B (zh) * 2017-05-15 2021-04-09 北京大学 作用于Dectin-1的稠合吖啶衍生物及其用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1394373A (en) * 1972-05-17 1975-05-14 Pfizer Ltd Control of plant diseases
DE3471308D1 (en) * 1983-10-17 1988-06-23 Synthelabo Imidazoline derivatives, their preparation and therapeutical use
FR2567126B1 (fr) * 1984-07-06 1986-12-12 Synthelabo Derives de pyrrolo(1,2,3-de) benzoxazine et benzothiazine, leur preparation et leur application en therapeutique
JPS6317885A (ja) * 1986-07-11 1988-01-25 Kyorin Pharmaceut Co Ltd スピロピロリジン−２，５−ジオン誘導体の製造方法

Also Published As

Publication number Publication date
KR890014545A (ko) 1989-10-24
PT89954B (pt) 1994-05-31
MY104955A (en) 1994-07-30
DK169723B1 (da) 1995-01-23
IL89480A0 (en) 1989-09-10
NO894350D0 (no) 1989-11-01
CA1335592C (en) 1995-05-16
AU3120489A (en) 1989-09-14
DK116689A (da) 1989-09-12
EP0332364A2 (en) 1989-09-13
ZA891800B (en) 1990-10-31
NZ228299A (en) 1990-09-26
HU201757B (en) 1990-12-28
FI895333A0 (fi) 1989-11-09
JPH0676408B2 (ja) 1994-09-28
NO170418B (no) 1992-07-06
NO170418C (no) 1992-10-14
HU885829D0 (en) 1990-02-28
DK116689D0 (da) 1989-03-10
EP0332364A3 (en) 1991-04-03
PT89954A (pt) 1989-11-10
NO894350L (no) 1989-11-01
WO1989008654A1 (en) 1989-09-21
FI96315B (fi) 1996-02-29
FI96315C (fi) 1996-06-10
KR910002565B1 (ko) 1991-04-26
JPH01275580A (ja) 1989-11-06
AU605410B2 (en) 1991-01-10

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Legal Events

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