IL77198A - 13beta-milbemycin derivatives,their preparation and their use as pesticides - Google Patents

13beta-milbemycin derivatives,their preparation and their use as pesticides

Info

Publication number
IL77198A
IL77198A IL77198A IL7719885A IL77198A IL 77198 A IL77198 A IL 77198A IL 77198 A IL77198 A IL 77198A IL 7719885 A IL7719885 A IL 7719885A IL 77198 A IL77198 A IL 77198A
Authority
IL
Israel
Prior art keywords
13beta
pesticides
preparation
milbemycin derivatives
milbemycin
Prior art date
Application number
IL77198A
Other languages
English (en)
Original Assignee
Ciba Geigy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy filed Critical Ciba Geigy
Publication of IL77198A publication Critical patent/IL77198A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Wood Science & Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL77198A 1984-12-04 1985-12-02 13beta-milbemycin derivatives,their preparation and their use as pesticides IL77198A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH575084 1984-12-04

Publications (1)

Publication Number Publication Date
IL77198A true IL77198A (en) 1989-06-30

Family

ID=4298719

Family Applications (1)

Application Number Title Priority Date Filing Date
IL77198A IL77198A (en) 1984-12-04 1985-12-02 13beta-milbemycin derivatives,their preparation and their use as pesticides

Country Status (20)

Country Link
US (1) US4696945A (fr)
EP (1) EP0184173B1 (fr)
JP (1) JPH072748B2 (fr)
CN (1) CN85109491A (fr)
AU (1) AU584950B2 (fr)
CA (1) CA1261823A (fr)
DD (2) DD250457A5 (fr)
DE (1) DE3587746D1 (fr)
DK (1) DK559985A (fr)
ES (3) ES8704473A1 (fr)
FI (1) FI854773A (fr)
GB (1) GB2167751B (fr)
GR (1) GR852893B (fr)
HU (1) HUT39739A (fr)
IL (1) IL77198A (fr)
MA (1) MA20583A1 (fr)
NZ (1) NZ214425A (fr)
PT (1) PT81591B (fr)
ZA (1) ZA859247B (fr)
ZW (1) ZW21785A1 (fr)

Families Citing this family (43)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4857509A (en) * 1985-01-22 1989-08-15 Ciba-Geigy Corporation 13β-alkylmilbemycin derivatives for controlling parasites of animals and plants
US4587247A (en) * 1985-02-25 1986-05-06 Merck & Co., Inc. Substituted and unsubstituted 13-(alkoxy)methoxy derivatives of the avermectin aglycones, compositions and use
ES8800986A1 (es) * 1985-07-27 1987-12-01 Pfizer Un procedimiento para la produccion de un nuevo derivado de avermectina
EP0235085A1 (fr) * 1986-02-20 1987-09-02 Ciba-Geigy Ag Dérivés de milbémycine substitués en position 13-bêta, leur préparation et utilisation comme agents ecto- et endoparasitaires pour le traitement d'animaux et de plantes
EP0238259B1 (fr) * 1986-03-12 1993-09-29 American Cyanamid Company Composés de macrolides
EP0240274A3 (fr) * 1986-04-03 1990-03-14 Merck & Co. Inc. Avermectine comme agents pour promotion de la croissance
EP0252879B1 (fr) * 1986-07-02 1992-05-06 Ciba-Geigy Ag Pesticides
US5840704A (en) * 1986-07-16 1998-11-24 Pfizer Inc. Antiparasitic agents and process for their preparation
JPS6393796A (ja) * 1986-10-09 1988-04-25 Shin Etsu Chem Co Ltd ペプチド合成の脱保護基用薬剤
US5212322A (en) * 1986-12-11 1993-05-18 Sankyo Company, Limited Macrolide compounds, their preparation and their use
AR243528A1 (es) * 1986-12-11 1993-08-31 Sankyo Co Procedimiento para preparar compuestos de macrolida y un procedimiento para producir con los mismos una composicion parasiticida.
US5525506A (en) * 1987-01-23 1996-06-11 Pfizer Inc. Process for production of avermectins and cultures therefor
US5234831A (en) * 1987-01-23 1993-08-10 Pfizer Inc Cultures for production of B avermectins
US5238848A (en) * 1987-01-23 1993-08-24 Pfizer Inc Cultures for production of avermectins
US5183749A (en) * 1987-02-04 1993-02-02 Sankyo Company, Ltd. Microbial process for the preparation of milbemycin derivatives
US4897416A (en) * 1987-02-18 1990-01-30 Ciba-Geigy Corporation Insecticides and parasiticides
US4871719A (en) * 1987-03-24 1989-10-03 Ciba-Geigy Corporation Composition for controlling parasites in productive livestock
GB8721647D0 (en) * 1987-09-15 1987-10-21 Pfizer Ltd Antiparasitic agents
US5240850A (en) * 1987-10-23 1993-08-31 Pfizer Inc. Cultures for production of avermectin aglycones
ATE87926T1 (de) * 1987-11-09 1993-04-15 Pfizer Ethylierte avermectine.
GB8726730D0 (en) 1987-11-14 1987-12-16 Pfizer Ltd Antiparasitic agents
US4918097A (en) * 1988-03-11 1990-04-17 Ciba-Geigy Corporation Insecticides and parasiticides
GB8811036D0 (en) * 1988-05-10 1988-06-15 Glaxo Group Ltd Chemical compounds
GB8811037D0 (en) * 1988-05-10 1988-06-15 Glaxo Group Ltd Chemical compounds
GB8813150D0 (en) * 1988-06-03 1988-07-06 American Cyanamid Co Chemical compounds
US5428034A (en) * 1988-09-02 1995-06-27 Sankyo Co., Ltd. Milbemycin derivatives, their preparation and their use
AU613521B2 (en) * 1988-09-02 1991-08-01 Sankyo Company Limited 13-substituted milbemycin derivatives, their preparation and use
NZ232422A (en) * 1989-02-16 1992-11-25 Merck & Co Inc 13-ketal milbemycin derivatives and parasiticides
TW202452B (fr) * 1989-12-01 1993-03-21 Ciba Geigy Ag
JPH085894B2 (ja) * 1990-03-01 1996-01-24 三共株式会社 ミルベマイシンエーテル誘導体
JP2622197B2 (ja) * 1990-03-01 1997-06-18 三共株式会社 13−エーテル置換ミルベマイシン誘導体
US5114930A (en) * 1990-05-14 1992-05-19 Merck & Co., Inc. Avermectin derivatives with a spacer inserted between the disaccharide and the aglycone useful as antiparasitic agents
US5188944A (en) * 1990-06-22 1993-02-23 Merck & Co., Inc. Process for the glycosylation of avermectin agylcones
US5208222A (en) * 1991-03-28 1993-05-04 Merck & Co., Inc. 4"-and 4'-alkylthio avermectin derivatives
EP0530901A1 (fr) * 1991-09-04 1993-03-10 Merck & Co. Inc. 13-bêta-O-méthoxyméthyl-22,23-dihydro avermectine B1A/B1B aglycone
JP2591552B2 (ja) * 1991-10-04 1997-03-19 三共株式会社 15−ヒドロキシミルベマイシン誘導体及びその製法
US6103504A (en) * 1992-03-25 2000-08-15 Pfizer Inc. Process for production of avermectins and cultures therefor
CA2105251C (fr) * 1992-09-01 2004-12-07 Mitsugi Shibano Methodes de preparation de derives de milbemycines etherifies en 13; nouveaux produits intermediaires utilises a cette fin
CA2213612C (fr) * 1995-02-24 2008-07-15 Novartis Ag Composition pour la lutte contre les parasites
WO1999017760A2 (fr) 1997-10-02 1999-04-15 Microcide Pharmaceuticals, Inc. Inhibiteurs de pompes d'efflux fongiques
US7919522B2 (en) 2007-05-03 2011-04-05 Merial Limited Compositions comprising C-13 alkoxyether macrolide compounds and phenylpyrazole compounds
CN101679451A (zh) * 2007-05-03 2010-03-24 梅瑞尔有限公司 包含c-13烷氧基醚大环内酯类化合物和苯基吡唑类化合物的组合物
JP5740676B2 (ja) * 2013-10-17 2015-06-24 メリアル リミテッド C−13アルコキシエーテルマクロライド化合物及びフェニルピラゾール化合物を含む組成物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH15982A (en) * 1977-10-03 1983-05-18 Merck & Co Inc Selective hydrogenation producta of c-076 compounds and derivatives thereof
US4199569A (en) * 1977-10-03 1980-04-22 Merck & Co., Inc. Selective hydrogenation products of C-076 compounds and derivatives thereof
JPS5461167A (en) * 1977-10-11 1979-05-17 Glaxo Group Ltd Novel substituted heterocyclic compounds* their manufacture and medical composition containing them
PH16612A (en) * 1977-12-19 1983-11-28 Merck & Co Inc 13-halo and 13-deoxy derivatives of c-076 compounds
US4200581A (en) * 1978-08-04 1980-04-29 Merck & Co., Inc. Alkyl derivatives of C-076 compounds
NZ201681A (en) * 1981-09-03 1985-11-08 Merck & Co Inc Avermectin derivatives and parasiticidal compositions
US4427663A (en) * 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4469682A (en) * 1983-01-28 1984-09-04 Merck & Co., Inc. Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use
US4587247A (en) * 1985-02-25 1986-05-06 Merck & Co., Inc. Substituted and unsubstituted 13-(alkoxy)methoxy derivatives of the avermectin aglycones, compositions and use

Also Published As

Publication number Publication date
EP0184173B1 (fr) 1994-02-02
GR852893B (fr) 1986-04-01
FI854773A (fi) 1986-06-05
MA20583A1 (fr) 1986-07-01
FI854773A0 (fi) 1985-12-02
DD250457A5 (de) 1987-10-14
NZ214425A (en) 1988-05-30
DK559985D0 (da) 1985-12-03
JPH072748B2 (ja) 1995-01-18
GB2167751B (en) 1988-04-27
EP0184173A2 (fr) 1986-06-11
EP0184173A3 (en) 1989-03-15
GB2167751A (en) 1986-06-04
DK559985A (da) 1986-06-05
ES556926A0 (es) 1987-10-01
ZW21785A1 (en) 1986-07-02
CN85109491A (zh) 1986-07-23
ES8708233A1 (es) 1987-10-01
CA1261823A (fr) 1989-09-26
ES8708232A1 (es) 1987-10-01
JPS61178986A (ja) 1986-08-11
ES8704473A1 (es) 1987-04-01
ES549508A0 (es) 1987-04-01
AU5071985A (en) 1986-06-12
ZA859247B (en) 1986-07-30
HUT39739A (en) 1986-10-29
US4696945A (en) 1987-09-29
DE3587746D1 (de) 1994-03-17
DD262662A5 (de) 1988-12-07
PT81591B (de) 1987-10-16
AU584950B2 (en) 1989-06-08
PT81591A (de) 1986-01-01
ES556927A0 (es) 1987-10-01
GB8529637D0 (en) 1986-01-08

Similar Documents

Publication Publication Date Title
IL77198A (en) 13beta-milbemycin derivatives,their preparation and their use as pesticides
IL87866A0 (en) 2-anilinopyrimidine derivatives,their preparation and their use as pesticides
IL82507A0 (en) 1-aralkylpyrazoles,their preparation and their use as pesticides
ZA85849B (en) New 2-cyanobenzimidazole derivatives,their preparation and their use as fungicides
IL77140A0 (en) 5-azolylacetoxymilbemycin derivatives,their preparation and their use as pesticides
IL77310A (en) 13beta-acyloxymilbemycin derivatives,their preparation and their use as pesticides
IL77650A (en) 13beta-alkylmilbemycin derivatives,their preparation and their use as pesticides
IL76392A0 (en) 13-halo-and 13-hydroxymilbemycine derivatives,their preparation and their use as pesticides
IL80991A0 (en) 5-heterocyclyl-1-aryl-pyrazoles,their preparation and their use as pesticides
IL83630A0 (en) Substituted 1-aryl-3-tert-butyl-pyrazoles,their preparation and their use as pesticides
IL76330A0 (en) Carbamoylimidazole derivatives,their preparation and their use as fungicides
IL79532A0 (en) Substituted trioxabicyclooctanes,their preparation and their use as pesticides
DE3560679D1 (en) 4-hydroxy-2h-1-benzothiopyran-2-one derivatives, their preparation and uses
IL73965A (en) 15-hydroxy-15h-milbemycin derivatives,their preparation and their use as pesticides
IL82611A0 (en) 5-oxy-and 5-thio-pyrazole derivatives,their preparation and their use as pesticides
IL77106A0 (en) Homopropargylamines,their preparation and their use as fungicides
IL75428A0 (en) Milbemycin derivatives,their preparation and their use as pesticides
IL73610A (en) 15-chloro-14-demethyl-14-methylene-15h-milbemycin derivatives,their preparation and their use as pesticides
IL72332A0 (en) Formamidoxime derivatives,their preparation and their use as pesticides
ZA857272B (en) Vinyltetrazolylphenyl derivatives,their preparation and their use
IL76214A0 (en) Sulphonylisourea derivatives,their preparation and their use as herbicides
IL75711A0 (en) Imidazo-pyrrolo-pyridine derivatives,their preparation and their use as herbicides
IL76224A0 (en) Substituted carbonylphenylsulphonylguanidines,their preparation and their use as herbicides
IL76213A0 (en) Substituted arylsulphonylguanidines,their preparation and their use as herbicides
IL74164A0 (en) Phenoxypropionyloxyalkanephosphonates,their preparation and their use as herbicides