IL72757A0 - Benzodiazepine derivatives,their preparation and pharmaceutical compositions containing them - Google Patents
Benzodiazepine derivatives,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL72757A0 IL72757A0 IL72757A IL7275784A IL72757A0 IL 72757 A0 IL72757 A0 IL 72757A0 IL 72757 A IL72757 A IL 72757A IL 7275784 A IL7275784 A IL 7275784A IL 72757 A0 IL72757 A0 IL 72757A0
- Authority
- IL
- Israel
- Prior art keywords
- preparation
- pharmaceutical compositions
- compositions containing
- benzodiazepine derivatives
- benzodiazepine
- Prior art date
Links
- 229940053197 benzodiazepine derivative antiepileptics Drugs 0.000 title 1
- 125000003310 benzodiazepinyl group Chemical class N1N=C(C=CC2=C1C=CC=C2)* 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C247/00—Compounds containing azido groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/74—Quinazolines; Hydrogenated quinazolines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to ring carbon atoms of the hetero ring
- C07D239/76—N-oxides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/24—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Anesthesiology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US52619483A | 1983-08-25 | 1983-08-25 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL72757A0 true IL72757A0 (en) | 1984-11-30 |
Family
ID=24096318
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL72757A IL72757A0 (en) | 1983-08-25 | 1984-08-23 | Benzodiazepine derivatives,their preparation and pharmaceutical compositions containing them |
Country Status (16)
| Country | Link |
|---|---|
| EP (1) | EP0135770A3 (da) |
| JP (1) | JPS6067480A (da) |
| KR (1) | KR850001756A (da) |
| AU (1) | AU3237984A (da) |
| DK (1) | DK406384A (da) |
| ES (2) | ES535392A0 (da) |
| FI (1) | FI843356A7 (da) |
| GR (1) | GR80197B (da) |
| HU (1) | HU193588B (da) |
| IL (1) | IL72757A0 (da) |
| MC (1) | MC1616A1 (da) |
| NO (1) | NO843376L (da) |
| NZ (1) | NZ209316A (da) |
| PH (1) | PH20029A (da) |
| PT (1) | PT79131B (da) |
| ZA (1) | ZA845757B (da) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2635776B1 (fr) * | 1988-09-01 | 1993-06-11 | Rhone Poulenc Agrochimie | Derives amides, procede pour leur fabrication et compositions fongicides les contenant |
| IL91418A (en) * | 1988-09-01 | 1997-11-20 | Rhone Poulenc Agrochimie | (hetero) cyclic amide derivatives, process for their preparation and fungicidal compositions containing them |
| US5317018A (en) * | 1992-06-09 | 1994-05-31 | Armin Walser | Benzodiazepines and compositions for treating anxiety and panic disorders, and idiopathic and psychomotor epilepsy |
| TW234123B (da) * | 1992-12-16 | 1994-11-11 | Takeda Pharm Industry Co Ltd | |
| US6063921A (en) * | 1997-11-20 | 2000-05-16 | Pharm-Eco Laboratories, Inc. | Synthesis of 11-aryl-5,6-dihydro-11H-dibenz[b,e]azepines |
| US8119629B2 (en) | 2007-10-03 | 2012-02-21 | Bristol-Meyers Squibb Company | Carboxamide GABAA α2 modulators |
| AU2017313753B2 (en) | 2016-08-16 | 2022-01-27 | The Trustees Of Columbia University In The City Of New York | GABA(A) receptor modulators and methods to control airway hyperresponsiveness and inflammation in asthma |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA755418B (en) * | 1974-09-11 | 1977-06-29 | Hoffmann La Roche | Diazepine derivatives |
| AT361486B (de) * | 1975-08-07 | 1981-03-10 | Hoffmann La Roche | Verfahren zur herstellung von neuen imidazo(1,5 -a) (1,4)diazepinverbindungen, ihren salzen und optisch aktiven formen |
| US4125726A (en) * | 1977-03-11 | 1978-11-14 | Hoffmann-La Roche Inc. | Imidazo[1,5-a][1,4]benzodiazepines |
| DK151808C (da) * | 1982-11-16 | 1988-06-20 | Ferrosan As | Analogifremgangsmaade til fremstilling af oxadiazolylimidazo-oe1,4aa-benzodiazepinderivater |
-
1984
- 1984-07-25 ZA ZA845757A patent/ZA845757B/xx unknown
- 1984-08-13 EP EP84109639A patent/EP0135770A3/de not_active Withdrawn
- 1984-08-23 NO NO843376A patent/NO843376L/no unknown
- 1984-08-23 NZ NZ209316A patent/NZ209316A/en unknown
- 1984-08-23 IL IL72757A patent/IL72757A0/xx unknown
- 1984-08-23 MC MC841721A patent/MC1616A1/fr unknown
- 1984-08-23 GR GR80197A patent/GR80197B/el unknown
- 1984-08-24 PT PT79131A patent/PT79131B/pt unknown
- 1984-08-24 ES ES535392A patent/ES535392A0/es active Granted
- 1984-08-24 DK DK406384A patent/DK406384A/da not_active Application Discontinuation
- 1984-08-24 AU AU32379/84A patent/AU3237984A/en not_active Abandoned
- 1984-08-24 JP JP59175328A patent/JPS6067480A/ja active Pending
- 1984-08-24 KR KR1019840005134A patent/KR850001756A/ko not_active Withdrawn
- 1984-08-24 HU HU843179A patent/HU193588B/hu unknown
- 1984-08-24 PH PH31144A patent/PH20029A/en unknown
- 1984-08-24 FI FI843356A patent/FI843356A7/fi not_active Application Discontinuation
-
1985
- 1985-05-31 ES ES543717A patent/ES8603433A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| PT79131A (en) | 1984-09-01 |
| FI843356A7 (fi) | 1985-02-26 |
| NZ209316A (en) | 1987-04-30 |
| FI843356A0 (fi) | 1984-08-24 |
| KR850001756A (ko) | 1985-04-01 |
| HU193588B (en) | 1987-10-28 |
| GR80197B (en) | 1985-01-03 |
| ES8602700A1 (es) | 1985-12-01 |
| ES543717A0 (es) | 1986-01-01 |
| NO843376L (no) | 1985-02-26 |
| ZA845757B (en) | 1985-04-24 |
| EP0135770A2 (de) | 1985-04-03 |
| EP0135770A3 (de) | 1988-01-13 |
| ES8603433A1 (es) | 1986-01-01 |
| PH20029A (en) | 1986-09-04 |
| DK406384A (da) | 1985-02-26 |
| MC1616A1 (fr) | 1985-07-18 |
| ES535392A0 (es) | 1985-12-01 |
| AU3237984A (en) | 1985-02-28 |
| JPS6067480A (ja) | 1985-04-17 |
| HUT34978A (en) | 1985-05-28 |
| DK406384D0 (da) | 1984-08-24 |
| PT79131B (en) | 1986-11-14 |
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