IL64083A - Meta-substituted 4-phenylalanyl-enkephalin analogs,their preparation and pharmaceutical compositions comprising them - Google Patents
Meta-substituted 4-phenylalanyl-enkephalin analogs,their preparation and pharmaceutical compositions comprising themInfo
- Publication number
- IL64083A IL64083A IL64083A IL6408381A IL64083A IL 64083 A IL64083 A IL 64083A IL 64083 A IL64083 A IL 64083A IL 6408381 A IL6408381 A IL 6408381A IL 64083 A IL64083 A IL 64083A
- Authority
- IL
- Israel
- Prior art keywords
- phenylalanyl
- meta
- substituted
- preparation
- pharmaceutical compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1027—Tetrapeptides containing heteroatoms different from O, S, or N
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Analytical Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pain & Pain Management (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US06/198,900 US4322340A (en) | 1980-10-20 | 1980-10-20 | Pharmacologically active peptides |
Publications (2)
Publication Number | Publication Date |
---|---|
IL64083A0 IL64083A0 (en) | 1982-01-31 |
IL64083A true IL64083A (en) | 1985-03-31 |
Family
ID=22735344
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL64083A IL64083A (en) | 1980-10-20 | 1981-10-19 | Meta-substituted 4-phenylalanyl-enkephalin analogs,their preparation and pharmaceutical compositions comprising them |
Country Status (27)
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0076557B1 (en) * | 1981-06-22 | 1985-11-13 | Imperial Chemical Industries Plc | Peptides and pseudopeptides in which the n terminus bears two substituents |
US4448717A (en) * | 1982-11-12 | 1984-05-15 | Eli Lilly And Company | Pharmacologically active peptides |
US4473497A (en) * | 1983-03-07 | 1984-09-25 | Eli Lilly And Company | Pharmacologically active peptides |
DK134784A (da) * | 1983-03-07 | 1984-09-08 | Lilly Co Eli | Farmakologisk virksomme tripeptid-derivater og fremgangsmaade til fremstilling deraf |
US4510082A (en) * | 1983-03-07 | 1985-04-09 | Eli Lilly And Company | Pharmacologically active peptides |
US4495178A (en) * | 1983-10-06 | 1985-01-22 | G. D. Searle & Co. | Enkephalin analogs |
JPH0449298A (ja) * | 1990-06-19 | 1992-02-18 | Univ New York State | 新規なエンケファリン誘導体および鎮痛剤 |
US5209930A (en) * | 1990-12-10 | 1993-05-11 | Rohm And Haas Company | Preparation and use of n-iodopropargyl oxycarbonyl amino acid esters and derivatives as antimicrobial agents |
US5952465A (en) * | 1993-04-23 | 1999-09-14 | Virginia Commonwealth University | Polypeptides that include conformation-constraining groups which flank a protein-protein interaction site |
AU6770794A (en) * | 1993-04-23 | 1994-11-21 | Herbert J. Evans | Polypeptides that include conformation-constraining groups which flank a protein-protein interaction site |
US5965698A (en) * | 1993-04-23 | 1999-10-12 | Virginia Commonwealth University | Polypeptides that include conformation-constraining groups which flank a protein--protein interaction site |
US6258550B1 (en) | 1993-04-23 | 2001-07-10 | Virginia Commonwealth University | Polypeptides that include conformation-constraining groups which flank a protein-protein interaction site |
US5928896A (en) * | 1993-04-23 | 1999-07-27 | Virginia Commonwealth University | Polypeptides that include conformation-constraining groups which flank a protein--protein interaction site |
US6084066A (en) * | 1993-10-29 | 2000-07-04 | Virginia Commonwealth University | Polypetides that include conformation-constraining groups which flank a protein-protein interaction site |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1577115A (en) * | 1976-07-27 | 1980-10-22 | Reckitt & Colmann Prod Ltd | Container closure units |
FI770219A (US06815460-20041109-C00097.png) * | 1976-02-02 | 1977-08-03 | Sandoz Ag | |
CH619686A5 (en) * | 1976-02-02 | 1980-10-15 | Sandoz Ag | Process for the preparation of novel peptides or peptide derivatives |
US4264491A (en) * | 1977-10-03 | 1981-04-28 | Eli Lilly And Company | Analgesic compounds |
US4265808A (en) * | 1979-12-17 | 1981-05-05 | Eli Lilly And Company | Pharmacologically active peptides |
-
1980
- 1980-10-20 US US06/198,900 patent/US4322340A/en not_active Expired - Lifetime
-
1981
- 1981-10-13 PH PH26344A patent/PH17006A/en unknown
- 1981-10-13 NZ NZ198628A patent/NZ198628A/en unknown
- 1981-10-13 CA CA000387762A patent/CA1187871A/en not_active Expired
- 1981-10-13 GR GR66269A patent/GR75342B/el unknown
- 1981-10-13 ZA ZA817063A patent/ZA817063B/xx unknown
- 1981-10-14 FI FI813198A patent/FI813198L/fi not_active Application Discontinuation
- 1981-10-14 RO RO105558A patent/RO83301B/ro unknown
- 1981-10-16 BG BG8153871A patent/BG36928A3/xx unknown
- 1981-10-16 IE IE2442/81A patent/IE52186B1/en unknown
- 1981-10-16 ES ES506316A patent/ES506316A0/es active Granted
- 1981-10-16 HU HU812999A patent/HU185320B/hu unknown
- 1981-10-19 AU AU76574/81A patent/AU547221B2/en not_active Expired - Fee Related
- 1981-10-19 AR AR287129A patent/AR230046A1/es active
- 1981-10-19 PL PL1981233498A patent/PL131155B1/pl unknown
- 1981-10-19 DK DK461481A patent/DK461481A/da not_active Application Discontinuation
- 1981-10-19 IL IL64083A patent/IL64083A/xx unknown
- 1981-10-19 DE DE8181304859T patent/DE3162823D1/de not_active Expired
- 1981-10-19 YU YU02490/81A patent/YU249081A/xx unknown
- 1981-10-19 EP EP81304859A patent/EP0050502B1/en not_active Expired
- 1981-10-19 GB GB8131402A patent/GB2085893B/en not_active Expired
- 1981-10-19 SU SU813345906A patent/SU1082319A3/ru active
- 1981-10-19 DD DD81234209A patent/DD200798A5/de unknown
- 1981-10-19 AT AT81304859T patent/ATE6777T1/de not_active IP Right Cessation
- 1981-10-19 PT PT73839A patent/PT73839B/pt unknown
- 1981-10-20 KR KR1019810003971A patent/KR830007518A/ko unknown
- 1981-10-20 JP JP56169398A patent/JPS57108052A/ja active Pending
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