IL315172A - Method for producing cis-4-aminotetrahydrofuran-2-carboxylic acid esters - Google Patents
Method for producing cis-4-aminotetrahydrofuran-2-carboxylic acid estersInfo
- Publication number
- IL315172A IL315172A IL315172A IL31517224A IL315172A IL 315172 A IL315172 A IL 315172A IL 315172 A IL315172 A IL 315172A IL 31517224 A IL31517224 A IL 31517224A IL 315172 A IL315172 A IL 315172A
- Authority
- IL
- Israel
- Prior art keywords
- process according
- compounds
- aminotetrahydrofuran
- esters
- production
- Prior art date
Links
- 238000000034 method Methods 0.000 title claims 9
- 238000004519 manufacturing process Methods 0.000 title claims 2
- 150000001732 carboxylic acid derivatives Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 claims 6
- 239000002253 acid Substances 0.000 claims 4
- OKKJLVBELUTLKV-UHFFFAOYSA-N Methanol Chemical group OC OKKJLVBELUTLKV-UHFFFAOYSA-N 0.000 claims 3
- 239000003054 catalyst Substances 0.000 claims 3
- 239000011541 reaction mixture Substances 0.000 claims 3
- 150000003839 salts Chemical class 0.000 claims 3
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 claims 2
- 229910052703 rhodium Inorganic materials 0.000 claims 2
- 239000010948 rhodium Substances 0.000 claims 2
- MHOVAHRLVXNVSD-UHFFFAOYSA-N rhodium atom Chemical compound [Rh] MHOVAHRLVXNVSD-UHFFFAOYSA-N 0.000 claims 2
- 239000002904 solvent Substances 0.000 claims 2
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 1
- 229910052739 hydrogen Inorganic materials 0.000 claims 1
- 239000001257 hydrogen Substances 0.000 claims 1
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 1
- 239000000203 mixture Substances 0.000 claims 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D307/18—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/24—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Furan Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP22158629 | 2022-02-24 | ||
| PCT/EP2023/054258 WO2023161204A1 (de) | 2022-02-24 | 2023-02-21 | Verfahren zur herstellung von cis-4-aminotetrahydrofuran-2-carbonsäureestern |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL315172A true IL315172A (en) | 2024-10-01 |
Family
ID=80461327
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL315172A IL315172A (en) | 2022-02-24 | 2023-02-21 | Method for producing cis-4-aminotetrahydrofuran-2-carboxylic acid esters |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP4482828A1 (de) |
| JP (1) | JP2025506282A (de) |
| KR (1) | KR20240153353A (de) |
| CN (1) | CN118748994A (de) |
| IL (1) | IL315172A (de) |
| MX (1) | MX2024010418A (de) |
| TW (1) | TW202400568A (de) |
| WO (1) | WO2023161204A1 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2026008692A1 (en) | 2024-07-04 | 2026-01-08 | Bayer Aktiengesellschaft | Process for the preparation of methyl 4-[[3-(3,5-difluorophenyl)-5-vinyl-4h-isoxazole-5-carbonyl]amino]tetrahydrofuran-2-carboxylate |
| EP4696683A1 (de) | 2024-08-15 | 2026-02-18 | Bayer Aktiengesellschaft | Verfahren zur herstellung von cis-4-aminotetrahydrofuran-2-carbonsäureestern |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EA024512B1 (ru) | 2011-03-31 | 2016-09-30 | Байер Интеллектуэль Проперти Гмбх | Гербицидно и фунгицидно действующие 3-фенилизоксазолин-5-карбоксамиды и 3-фенилизоксазолин-5-тиоамиды |
| WO2016145082A1 (en) * | 2015-03-09 | 2016-09-15 | Northwestern University | Tetrahydrothiophene-based gaba aminotransferase inactivators |
| AU2018291688B2 (en) * | 2017-06-27 | 2022-02-03 | Janssen Pharmaceutica Nv | Heteroaryldihydropyrimidine derivatives and methods of treating hepatitis B infections |
| WO2021170464A1 (en) | 2020-02-28 | 2021-09-02 | Basf Se | Herbicidal malonamides |
| MX2023000970A (es) | 2020-07-23 | 2023-03-01 | Bayer Ag | Metodo de preparacion de aminofuranos. |
-
2023
- 2023-02-21 EP EP23705428.3A patent/EP4482828A1/de active Pending
- 2023-02-21 MX MX2024010418A patent/MX2024010418A/es unknown
- 2023-02-21 JP JP2024550264A patent/JP2025506282A/ja active Pending
- 2023-02-21 IL IL315172A patent/IL315172A/en unknown
- 2023-02-21 CN CN202380023391.6A patent/CN118748994A/zh active Pending
- 2023-02-21 KR KR1020247031124A patent/KR20240153353A/ko active Pending
- 2023-02-21 WO PCT/EP2023/054258 patent/WO2023161204A1/de not_active Ceased
- 2023-02-22 TW TW112106409A patent/TW202400568A/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN118748994A (zh) | 2024-10-08 |
| MX2024010418A (es) | 2024-09-05 |
| KR20240153353A (ko) | 2024-10-22 |
| EP4482828A1 (de) | 2025-01-01 |
| WO2023161204A1 (de) | 2023-08-31 |
| TW202400568A (zh) | 2024-01-01 |
| JP2025506282A (ja) | 2025-03-07 |
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