IL163953A0 - Bicyclic heterocyclic compounds and pharmaceuticalcompositions containing the same - Google Patents

Bicyclic heterocyclic compounds and pharmaceuticalcompositions containing the same

Info

Publication number
IL163953A0
IL163953A0 IL16395303A IL16395303A IL163953A0 IL 163953 A0 IL163953 A0 IL 163953A0 IL 16395303 A IL16395303 A IL 16395303A IL 16395303 A IL16395303 A IL 16395303A IL 163953 A0 IL163953 A0 IL 163953A0
Authority
IL
Israel
Prior art keywords
same
heterocyclic compounds
bicyclic heterocyclic
pharmaceuticalcompositions
pharmaceuticalcompositions containing
Prior art date
Application number
IL16395303A
Other languages
English (en)
Original Assignee
Ortho Mcneil Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Mcneil Pharm Inc filed Critical Ortho Mcneil Pharm Inc
Publication of IL163953A0 publication Critical patent/IL163953A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL16395303A 2002-03-08 2003-03-07 Bicyclic heterocyclic compounds and pharmaceuticalcompositions containing the same IL163953A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US36273202P 2002-03-08 2002-03-08
PCT/US2003/007240 WO2003075858A2 (fr) 2002-03-08 2003-03-07 Heterocycles bicycliques pour le traitement des diabetes et d'autres maladies

Publications (1)

Publication Number Publication Date
IL163953A0 true IL163953A0 (en) 2005-12-18

Family

ID=27805219

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16395303A IL163953A0 (en) 2002-03-08 2003-03-07 Bicyclic heterocyclic compounds and pharmaceuticalcompositions containing the same

Country Status (9)

Country Link
US (1) US7196108B2 (fr)
EP (1) EP1487446A4 (fr)
JP (1) JP2005525371A (fr)
AU (1) AU2003223233A1 (fr)
BR (1) BR0308278A (fr)
CA (1) CA2478765A1 (fr)
IL (1) IL163953A0 (fr)
TW (1) TWI277415B (fr)
WO (1) WO2003075858A2 (fr)

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WO2002072543A2 (fr) * 2001-03-08 2002-09-19 Maxia Pharmaceuticals, Inc. Molecules activant un recepteur rxr
WO2003016267A1 (fr) * 2001-08-17 2003-02-27 Incyte San Diego Incorporated Derives d'oxime pour le traitement de la dyslipidemie et de l'hypercholesterolemie
US7196108B2 (en) 2002-03-08 2007-03-27 Incyte San Diego Inc. Bicyclic heterocycles for the treatment of diabetes and other diseases
US7102000B2 (en) * 2002-03-08 2006-09-05 Incyte San Diego Inc. Heterocyclic amide derivatives for the treatment of diabetes and other diseases
CA2490535A1 (fr) * 2002-06-25 2003-12-31 Helicon Therapeutics, Inc. Alteration de la memoire par modification de la fonction de staufen
BR0317483A (pt) 2002-12-20 2005-11-16 Glaxo Group Ltd Derivados de benzodiazepina para o tratamento de desordens neurológicas
CA2522759A1 (fr) * 2003-04-18 2004-11-04 Incyte San Diego Incorporated Composes isochromane substitues pour le traitement de troubles metaboliques, du cancer et d'autres maladies
US7122700B2 (en) 2004-07-30 2006-10-17 Xerox Corporation Arylamine processes
GT200500185A (es) * 2004-08-09 2006-04-10 Moduladores del receptor de progesterona que comprenden derivados de pirrol-oxindol y sus usos
RU2007139541A (ru) * 2005-04-22 2009-05-27 Вайет (Us) Производные хромана и хромена и их применение
JP2009512637A (ja) * 2005-09-30 2009-03-26 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ 異常脂血症、高コレステロール血症及び糖尿病の処置のためのｒｘｒアゴニストとしてのジヒドロ−［１ｈ］−キノリン−２−オン誘導体
KR20120034666A (ko) 2009-05-22 2012-04-12 엑셀리시스, 인코포레이티드 증식성 질환에 대한 벤족사제핀 기반 ｐ１３ｋ／ｍｔ０ｒ의 억제제
AU2010254200A1 (en) 2009-05-26 2011-12-08 Exelixis, Inc. Benzoxazepines as inhibitors of PI3K/m TOR and methods of their use and manufacture
DK2464645T3 (en) 2009-07-27 2017-10-23 Gilead Sciences Inc CONDENSED, HETEROCYCLIC COMPOUNDS AS IRON CHANNEL MODULATORS
CN103096977B (zh) 2010-07-02 2017-02-15 吉利德科学公司 作为离子通道调节剂的稠杂环化合物
US20130259807A1 (en) * 2010-09-01 2013-10-03 The Regents Of The University Of California Cell culture screen for agents that control adipogenesis and myofibroblast differentiation
US9056862B2 (en) 2011-05-10 2015-06-16 National University Corporation Kobe University Thioxothiazolidine derivative having Ras function inhibitory effect
WO2012154760A1 (fr) 2011-05-10 2012-11-15 Gilead Sciences, Inc. Composés hétérocycliques condensés utilisés comme modulateurs des canaux sodiques
NO3175985T3 (fr) 2011-07-01 2018-04-28
TWI549944B (zh) 2011-07-01 2016-09-21 吉李德科學股份有限公司 作為離子通道調節劑之稠合雜環化合物
AU2013347797A1 (en) 2012-11-25 2015-07-02 The Regents Of The University Of California Peptides that stimulate subcutaneous adipogenesis
US10844102B2 (en) 2014-05-28 2020-11-24 The Regents Of The University Of California Peptides, compositions, and methods for stimulating subcutaneous adipogenesis
AU2019255310B2 (en) 2018-04-18 2022-11-24 Constellation Pharmaceuticals, Inc. Modulators of methyl modifying enzymes, compositions and uses thereof
CA3100977A1 (fr) 2018-05-21 2019-11-28 Constellation Pharmaceuticals, Inc. Modulateurs d'enzymes de modification de methyle, compositions et utilisations de ceux-ci

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Also Published As

Publication number Publication date
US20040034004A1 (en) 2004-02-19
TWI277415B (en) 2007-04-01
CA2478765A1 (fr) 2003-09-18
AU2003223233A2 (en) 2003-09-22
WO2003075858A3 (fr) 2004-03-18
US7196108B2 (en) 2007-03-27
WO2003075858A2 (fr) 2003-09-18
EP1487446A2 (fr) 2004-12-22
EP1487446A4 (fr) 2006-04-19
BR0308278A (pt) 2005-02-09
AU2003223233A1 (en) 2003-09-22
TW200304814A (en) 2003-10-16
JP2005525371A (ja) 2005-08-25

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