IL161306A0 - Pharmaceutical formulation comprising (r)-bicalutamide - Google Patents

Pharmaceutical formulation comprising (r)-bicalutamide

Info

Publication number
IL161306A0
IL161306A0 IL16130602A IL16130602A IL161306A0 IL 161306 A0 IL161306 A0 IL 161306A0 IL 16130602 A IL16130602 A IL 16130602A IL 16130602 A IL16130602 A IL 16130602A IL 161306 A0 IL161306 A0 IL 161306A0
Authority
IL
Israel
Prior art keywords
bicalutamide
pharmaceutical formulation
formulation
pharmaceutical
Prior art date
Application number
IL16130602A
Other languages
English (en)
Original Assignee
Astrazeneca Uk Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Uk Ltd filed Critical Astrazeneca Uk Ltd
Publication of IL161306A0 publication Critical patent/IL161306A0/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/275Nitriles; Isonitriles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL16130602A 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r)-bicalutamide IL161306A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0103424A SE0103424D0 (sv) 2001-10-15 2001-10-15 Pharmaceutical formulation
PCT/GB2002/004621 WO2003032950A1 (en) 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r) -bicalutamide

Publications (1)

Publication Number Publication Date
IL161306A0 true IL161306A0 (en) 2004-09-27

Family

ID=20285650

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16130602A IL161306A0 (en) 2001-10-15 2002-10-11 Pharmaceutical formulation comprising (r)-bicalutamide

Country Status (19)

Country Link
US (1) US20060058381A1 (ja)
EP (1) EP1439823A1 (ja)
JP (1) JP3639587B2 (ja)
KR (1) KR20050035163A (ja)
CN (1) CN1571658A (ja)
AR (1) AR036877A1 (ja)
BR (1) BR0213248A (ja)
CA (1) CA2462219A1 (ja)
CO (1) CO5580755A2 (ja)
HU (1) HUP0401369A3 (ja)
IL (1) IL161306A0 (ja)
IS (1) IS7219A (ja)
MX (1) MXPA04003520A (ja)
NO (1) NO20041485L (ja)
PL (1) PL368226A1 (ja)
RU (1) RU2004115023A (ja)
SE (1) SE0103424D0 (ja)
WO (1) WO2003032950A1 (ja)
ZA (1) ZA200402729B (ja)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1503662A (zh) * 2001-02-27 2004-06-09 药物制剂
ES2332920T3 (es) 2004-01-20 2010-02-15 Novartis Ag Proceso y formulacion de compresion directa.
US20080161404A1 (en) * 2005-02-23 2008-07-03 Astrazeneca Ab Bicalutamide for Delivering Increasing Steady State Plasma Levels
US20080045600A1 (en) * 2006-08-17 2008-02-21 Gawande Rahul S Bicalutamide compositions
US20100048913A1 (en) 2008-03-14 2010-02-25 Angela Brodie Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens;Synthesis In Vitro Biological Activities, Pharmacokinetics and Antitumor Activity
JP2012516900A (ja) 2009-02-05 2012-07-26 トーカイ ファーマシューティカルズ,インク. ステロイド性cyp17阻害剤/抗アンドロゲン剤の新しいプロドラッグ
CN101987086B (zh) * 2009-08-03 2012-07-18 北京化工大学 一种超细比卡鲁胺口服片剂及其制备方法
BR112014001440A2 (pt) * 2011-07-18 2017-02-21 Tokai Pharmaceuticals Inc novas composições e métodos para o tratamento de câncer de próstata
CN105358535B (zh) 2012-09-11 2019-01-04 麦迪威森前列腺医疗有限责任公司 恩杂鲁胺制剂
SG11201507093WA (en) 2013-03-14 2015-10-29 Univ Maryland Baltimore Office Of Technology Transfer Androgen receptor down-regulating agents and uses thereof
RU2016104643A (ru) 2013-08-12 2017-09-19 Токай Фармасьютикалз, Инк. Биомаркёры для лечения неопластических заболеваний с применением нацеленных на андроген методов лечения
MA41107A (fr) * 2014-12-05 2017-10-10 Aragon Pharmaceuticals Inc Compositions anti-cancéreuses
ES2883187T3 (es) 2014-12-05 2021-12-07 Aragon Pharmaceuticals Inc Composiciones anticancerosas

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3629237A (en) * 1968-09-12 1971-12-21 Shinetsu Chemical Co Compositions useful as enteric coatings and method for preparing acid phthalates of cellulose ethers for them
US4309405A (en) * 1979-08-09 1982-01-05 American Home Products Corporation Sustained release pharmaceutical compositions
DE3372965D1 (en) * 1982-07-23 1987-09-17 Ici Plc Amide derivatives
US4946686A (en) * 1987-09-24 1990-08-07 Merck & Co., Inc. Solubility modulated drug delivery system
ATE159426T1 (de) * 1991-04-16 1997-11-15 Nippon Shinyaku Co Ltd Verfahren zur herstellung einer festen dispersion
JPH09508125A (ja) * 1994-01-21 1997-08-19 セプラコー,インコーポレイテッド 光学的純正r−(−)−カソデックスを使用した男性ホルモン依存疾患治療のための方法と組成
CN1503662A (zh) * 2001-02-27 2004-06-09 药物制剂
MXPA03008999A (es) * 2001-04-02 2004-02-12 Astrazeneca Ab Composicion farmaceutica solida que comprende 4-ciano -trifluor-3 -(4-fluorfenilsulfonil) -2-hidroxi-2 -metilpropino -m-toluidida y pvp.

Also Published As

Publication number Publication date
IS7219A (is) 2004-04-14
SE0103424D0 (sv) 2001-10-15
US20060058381A1 (en) 2006-03-16
WO2003032950A1 (en) 2003-04-24
EP1439823A1 (en) 2004-07-28
CO5580755A2 (es) 2005-11-30
CA2462219A1 (en) 2003-04-24
ZA200402729B (en) 2005-01-13
AR036877A1 (es) 2004-10-13
JP2004521963A (ja) 2004-07-22
CN1571658A (zh) 2005-01-26
BR0213248A (pt) 2004-09-28
NO20041485L (no) 2004-04-13
KR20050035163A (ko) 2005-04-15
PL368226A1 (en) 2005-03-21
RU2004115023A (ru) 2005-04-10
JP3639587B2 (ja) 2005-04-20
HUP0401369A2 (hu) 2004-11-29
MXPA04003520A (es) 2004-07-23
HUP0401369A3 (en) 2006-05-29

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