IL160194A0 - GLYCINE-SUBSTITUTED THIENO [2,3-d] PYRIMIDINE WITH COMBINED LH AND FSH AGONISTIC ACTIVITY - Google Patents

GLYCINE-SUBSTITUTED THIENO [2,3-d] PYRIMIDINE WITH COMBINED LH AND FSH AGONISTIC ACTIVITY

Info

Publication number
IL160194A0
IL160194A0 IL16019402A IL16019402A IL160194A0 IL 160194 A0 IL160194 A0 IL 160194A0 IL 16019402 A IL16019402 A IL 16019402A IL 16019402 A IL16019402 A IL 16019402A IL 160194 A0 IL160194 A0 IL 160194A0
Authority
IL
Israel
Prior art keywords
pyrimidine
glycine
combined
agonistic activity
substituted thieno
Prior art date
Application number
IL16019402A
Other languages
English (en)
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of IL160194A0 publication Critical patent/IL160194A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/06Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/06Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A61P5/08Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH for decreasing, blocking or antagonising the activity of the anterior pituitary hormones

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
IL16019402A 2001-09-04 2002-08-29 GLYCINE-SUBSTITUTED THIENO [2,3-d] PYRIMIDINE WITH COMBINED LH AND FSH AGONISTIC ACTIVITY IL160194A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01203328 2001-09-04
PCT/EP2002/009648 WO2003020727A1 (en) 2001-09-04 2002-08-29 GLYCINE-SUBSTITUTED THIENO [2,3-d]PYRIMIDINES WITH COMBINED LH AND FSH AGONISTIC ACTIVITY

Publications (1)

Publication Number Publication Date
IL160194A0 true IL160194A0 (en) 2004-07-25

Family

ID=8180877

Family Applications (2)

Application Number Title Priority Date Filing Date
IL16019402A IL160194A0 (en) 2001-09-04 2002-08-29 GLYCINE-SUBSTITUTED THIENO [2,3-d] PYRIMIDINE WITH COMBINED LH AND FSH AGONISTIC ACTIVITY
IL160194A IL160194A (en) 2001-09-04 2004-02-03 Theano [2,3 – d] glycine-converted pyrimidines with combined LH and FSH agonist activity

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL160194A IL160194A (en) 2001-09-04 2004-02-03 Theano [2,3 – d] glycine-converted pyrimidines with combined LH and FSH agonist activity

Country Status (27)

Country Link
US (1) US7375109B2 (is)
EP (1) EP1427734B1 (is)
JP (1) JP4263094B2 (is)
KR (1) KR100891630B1 (is)
CN (1) CN1261437C (is)
AR (1) AR036408A1 (is)
AT (1) ATE309251T1 (is)
AU (1) AU2002333750B2 (is)
BR (1) BR0212173A (is)
CA (1) CA2457212C (is)
CY (1) CY1106052T1 (is)
DE (1) DE60207280T2 (is)
DK (1) DK1427734T3 (is)
EC (1) ECSP044990A (is)
ES (1) ES2252540T3 (is)
HR (1) HRP20040194A2 (is)
HU (1) HUP0401443A3 (is)
IL (2) IL160194A0 (is)
IS (1) IS2419B (is)
MX (1) MXPA04002046A (is)
NO (1) NO328792B1 (is)
NZ (1) NZ531375A (is)
PE (1) PE20030467A1 (is)
PL (1) PL368388A1 (is)
RU (1) RU2294331C2 (is)
WO (1) WO2003020727A1 (is)
ZA (1) ZA200401459B (is)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6890923B2 (en) * 2002-12-16 2005-05-10 Astrazeneca Ab Compounds
KR100666484B1 (ko) * 2005-02-04 2007-01-09 삼성전자주식회사 반도체 메모리 장치의 입출력 회로 및 입출력 방법
CA2741030A1 (en) 2008-10-20 2010-04-29 Marvin C. Gershengorn Low molecular weight thyroid stimulating hormone receptor (tshr) agonists
CN101762915B (zh) * 2008-12-24 2013-04-17 北京京东方光电科技有限公司 Tft-lcd阵列基板及其驱动方法
CA2789818A1 (en) 2010-04-08 2011-10-13 The United States Of America, As Represented By The Secretary, Departmen T Of Health And Human Services Inverse agonists and neutral antagonists for the tsh receptor
PL2900675T3 (pl) * 2012-09-28 2019-08-30 Takeda Pharmaceutical Company Limited Sposób wytwarzania pochodnej tienopirymidyny

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE86484T1 (de) 1987-08-08 1993-03-15 Akzo Nv Kontrazeptives implantat.
TW564247B (en) 1999-04-08 2003-12-01 Akzo Nobel Nv Bicyclic heteraromatic compound

Also Published As

Publication number Publication date
BR0212173A (pt) 2004-07-20
JP4263094B2 (ja) 2009-05-13
KR20040029135A (ko) 2004-04-03
CN1261437C (zh) 2006-06-28
AU2002333750B2 (en) 2008-02-21
HUP0401443A3 (en) 2008-05-28
DE60207280T2 (de) 2006-05-18
DE60207280D1 (de) 2005-12-15
ECSP044990A (es) 2004-04-28
NO20040922L (no) 2004-03-03
ZA200401459B (en) 2004-11-22
CA2457212A1 (en) 2003-03-13
WO2003020727A1 (en) 2003-03-13
RU2004110036A (ru) 2005-10-10
KR100891630B1 (ko) 2009-04-03
IL160194A (en) 2009-06-15
CA2457212C (en) 2011-02-15
US7375109B2 (en) 2008-05-20
HRP20040194A2 (en) 2004-08-31
JP2005504784A (ja) 2005-02-17
DK1427734T3 (da) 2006-03-06
HUP0401443A2 (hu) 2004-11-29
EP1427734A1 (en) 2004-06-16
IS7152A (is) 2004-02-13
RU2294331C2 (ru) 2007-02-27
ATE309251T1 (de) 2005-11-15
CN1551883A (zh) 2004-12-01
PL368388A1 (en) 2005-03-21
EP1427734B1 (en) 2005-11-09
IS2419B (is) 2008-10-15
ES2252540T3 (es) 2006-05-16
US20040180907A1 (en) 2004-09-16
NZ531375A (en) 2005-06-24
PE20030467A1 (es) 2003-05-26
MXPA04002046A (es) 2004-07-16
AR036408A1 (es) 2004-09-08
CY1106052T1 (el) 2011-04-06
NO328792B1 (no) 2010-05-18

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