IL152023A0 - Compounds having adenosine a2 receptor antagonism and pharmaceutical compositions containing the same - Google Patents

Compounds having adenosine a2 receptor antagonism and pharmaceutical compositions containing the same

Info

Publication number
IL152023A0
IL152023A0 IL15202301A IL15202301A IL152023A0 IL 152023 A0 IL152023 A0 IL 152023A0 IL 15202301 A IL15202301 A IL 15202301A IL 15202301 A IL15202301 A IL 15202301A IL 152023 A0 IL152023 A0 IL 152023A0
Authority
IL
Israel
Prior art keywords
adenosine
compounds
same
pharmaceutical compositions
defecation
Prior art date
Application number
IL15202301A
Other languages
English (en)
Original Assignee
Eisai Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai Co Ltd filed Critical Eisai Co Ltd
Publication of IL152023A0 publication Critical patent/IL152023A0/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • A61K31/522Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/10Laxatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • HELECTRICITY
    • H04ELECTRIC COMMUNICATION TECHNIQUE
    • H04BTRANSMISSION
    • H04B10/00Transmission systems employing electromagnetic waves other than radio-waves, e.g. infrared, visible or ultraviolet light, or employing corpuscular radiation, e.g. quantum communication
    • H04B10/11Arrangements specific to free-space transmission, i.e. transmission through air or vacuum
    • H04B10/112Line-of-sight transmission over an extended range

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Signal Processing (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Electromagnetism (AREA)
  • Physics & Mathematics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Computer Networks & Wireless Communication (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL15202301A 2000-04-26 2001-04-26 Compounds having adenosine a2 receptor antagonism and pharmaceutical compositions containing the same IL152023A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2000126489 2000-04-26
JP2000220124 2000-07-21
PCT/JP2001/003643 WO2001080893A1 (fr) 2000-04-26 2001-04-26 Compositions medicinales favorisant les mouvements intestinaux

Publications (1)

Publication Number Publication Date
IL152023A0 true IL152023A0 (en) 2003-04-10

Family

ID=26590887

Family Applications (2)

Application Number Title Priority Date Filing Date
IL15202301A IL152023A0 (en) 2000-04-26 2001-04-26 Compounds having adenosine a2 receptor antagonism and pharmaceutical compositions containing the same
IL188052A IL188052A0 (en) 2000-04-26 2007-12-11 A defecation promoting agent having adenosine a2 receptor antagonism and pharmaceutical compositions containing the same

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL188052A IL188052A0 (en) 2000-04-26 2007-12-11 A defecation promoting agent having adenosine a2 receptor antagonism and pharmaceutical compositions containing the same

Country Status (16)

Country Link
US (3) US7189717B2 (ko)
EP (2) EP1510222A3 (ko)
JP (1) JP4128360B2 (ko)
KR (2) KR20070058022A (ko)
CN (1) CN1197621C (ko)
AT (1) ATE284712T1 (ko)
AU (2) AU2001252606B2 (ko)
CA (1) CA2407013A1 (ko)
DE (1) DE60107835T2 (ko)
HU (1) HUP0300927A2 (ko)
IL (2) IL152023A0 (ko)
MX (1) MXPA02010552A (ko)
NO (1) NO20025116L (ko)
NZ (1) NZ521633A (ko)
RU (2) RU2294762C2 (ko)
WO (1) WO2001080893A1 (ko)

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ES2580702B1 (es) * 2015-02-25 2017-06-08 Palobiofarma, S.L. Derivados de 2-aminopiridina como antagonistas del receptor A2b de adenosina y ligandos del receptor MT3 de melatonina
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Also Published As

Publication number Publication date
EP1510222A2 (en) 2005-03-02
US20070054876A1 (en) 2007-03-08
US7189717B2 (en) 2007-03-13
AU2001252606B2 (en) 2005-07-07
AU5260601A (en) 2001-11-07
EP1283056B1 (en) 2004-12-15
MXPA02010552A (es) 2003-03-10
EP1283056A1 (en) 2003-02-12
IL188052A0 (en) 2008-03-20
JP4128360B2 (ja) 2008-07-30
ATE284712T1 (de) 2005-01-15
US20030171383A1 (en) 2003-09-11
CN1197621C (zh) 2005-04-20
RU2005127415A (ru) 2007-03-10
CA2407013A1 (en) 2002-10-22
KR20070058022A (ko) 2007-06-07
DE60107835T2 (de) 2005-12-22
NO20025116L (no) 2002-12-23
US20060270674A1 (en) 2006-11-30
CN1426310A (zh) 2003-06-25
NZ521633A (en) 2005-01-28
NO20025116D0 (no) 2002-10-24
WO2001080893A1 (fr) 2001-11-01
KR20020089495A (ko) 2002-11-29
DE60107835D1 (de) 2005-01-20
KR100782091B1 (ko) 2007-12-04
EP1510222A3 (en) 2007-05-23
RU2002131637A (ru) 2004-03-27
RU2294762C2 (ru) 2007-03-10
EP1283056A4 (en) 2003-07-02
HUP0300927A2 (hu) 2003-07-28

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