IL146871A0 - Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases - Google Patents
Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseasesInfo
- Publication number
- IL146871A0 IL146871A0 IL14687100A IL14687100A IL146871A0 IL 146871 A0 IL146871 A0 IL 146871A0 IL 14687100 A IL14687100 A IL 14687100A IL 14687100 A IL14687100 A IL 14687100A IL 146871 A0 IL146871 A0 IL 146871A0
- Authority
- IL
- Israel
- Prior art keywords
- metabotropic glutamate
- nervous system
- central nervous
- receptor antagonists
- glutamate receptor
- Prior art date
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- Pyridine Compounds (AREA)
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- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
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Application Number | Priority Date | Filing Date | Title |
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US13727299P | 1999-06-02 | 1999-06-02 | |
PCT/US2000/015222 WO2000073283A1 (en) | 1999-06-02 | 2000-06-02 | Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases |
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IL146871A0 true IL146871A0 (en) | 2002-08-14 |
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IL14687100A IL146871A0 (en) | 1999-06-02 | 2000-06-02 | Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases |
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EP (2) | EP1196397B1 (xx) |
JP (1) | JP2003500480A (xx) |
CN (2) | CN1361768A (xx) |
AT (1) | ATE302194T1 (xx) |
AU (2) | AU778063C (xx) |
CA (1) | CA2376024A1 (xx) |
CH (1) | CH1196397H1 (xx) |
DE (1) | DE60022050C5 (xx) |
DK (1) | DK1196397T3 (xx) |
ES (1) | ES2249272T3 (xx) |
HK (1) | HK1048635A1 (xx) |
IL (1) | IL146871A0 (xx) |
MX (1) | MXPA01012445A (xx) |
NZ (1) | NZ515894A (xx) |
WO (1) | WO2000073283A1 (xx) |
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JP5617799B2 (ja) * | 2010-12-07 | 2014-11-05 | 信越化学工業株式会社 | 化学増幅レジスト材料及びパターン形成方法 |
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JO3367B1 (ar) | 2013-09-06 | 2019-03-13 | Janssen Pharmaceutica Nv | مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2 |
HUE053734T2 (hu) | 2014-01-21 | 2021-07-28 | Janssen Pharmaceutica Nv | 2-es altípusú metabotróp glutamáterg receptor pozitív allosztérikus modulátorait tartalmazó kombinációk és alkalmazásuk |
EA201891617A3 (ru) | 2014-01-21 | 2019-04-30 | Янссен Фармацевтика Нв | Комбинации, содержащие положительные аллостерические модуляторы или ортостерические агонисты метаботропного глутаматергического рецептора 2 подтипа, и их применение |
KR102529578B1 (ko) | 2014-08-29 | 2023-05-09 | (주)아모레퍼시픽 | 신규 아다만탄 유도체 화합물 |
CN104860901B (zh) * | 2015-04-20 | 2017-04-19 | 北京工业大学 | 一种苯并噻唑‑2‑羧酸的制备方法 |
BR112018012469B1 (pt) * | 2015-12-17 | 2020-11-24 | Astex Therapeutics Limited | compostos quinolina-3-carboxamidas como inibidores da h-pgds, composição farmacêutica compreendendo os ditos compostos e uso terapêutico dos mesmos. |
KR20190115451A (ko) | 2017-02-03 | 2019-10-11 | 세르타 테라퓨틱스 피티와이 엘티디. | 항-섬유성 화합물 |
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US6204292B1 (en) * | 1997-07-18 | 2001-03-20 | Georgetown University | Bicyclic metabotropic glutamate receptor ligands |
CA2311131A1 (en) * | 1997-11-21 | 1999-06-03 | Nps Pharmaceuticals, Inc. | Metabotropic glutamate receptor antagonists for treating central nervous system diseases |
-
2000
- 2000-06-02 CN CN00810658A patent/CN1361768A/zh active Pending
- 2000-06-02 CA CA002376024A patent/CA2376024A1/en not_active Abandoned
- 2000-06-02 DE DE60022050T patent/DE60022050C5/de not_active Expired - Fee Related
- 2000-06-02 EP EP00936465A patent/EP1196397B1/en not_active Expired - Lifetime
- 2000-06-02 NZ NZ515894A patent/NZ515894A/xx unknown
- 2000-06-02 IL IL14687100A patent/IL146871A0/xx unknown
- 2000-06-02 AU AU51780/00A patent/AU778063C/en not_active Ceased
- 2000-06-02 CH CH00936465T patent/CH1196397H1/de unknown
- 2000-06-02 ES ES00936465T patent/ES2249272T3/es not_active Expired - Lifetime
- 2000-06-02 CN CNA2005101186507A patent/CN1789246A/zh active Pending
- 2000-06-02 WO PCT/US2000/015222 patent/WO2000073283A1/en active IP Right Grant
- 2000-06-02 DK DK00936465T patent/DK1196397T3/da active
- 2000-06-02 JP JP2000621349A patent/JP2003500480A/ja active Pending
- 2000-06-02 AT AT00936465T patent/ATE302194T1/de not_active IP Right Cessation
- 2000-06-02 EP EP05017791A patent/EP1595871A3/en not_active Withdrawn
- 2000-06-02 MX MXPA01012445A patent/MXPA01012445A/es active IP Right Grant
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2003
- 2003-01-30 HK HK03100778.5A patent/HK1048635A1/zh unknown
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Also Published As
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AU2005200633A1 (en) | 2005-03-17 |
EP1196397A1 (en) | 2002-04-17 |
AU778063C (en) | 2005-12-15 |
EP1595871A3 (en) | 2005-11-30 |
CA2376024A1 (en) | 2000-12-07 |
CH1196397H1 (de) | 2007-05-31 |
CN1361768A (zh) | 2002-07-31 |
EP1196397B1 (en) | 2005-08-17 |
DE60022050C5 (de) | 2007-10-11 |
DK1196397T3 (da) | 2006-01-02 |
NZ515894A (en) | 2003-09-26 |
MXPA01012445A (es) | 2003-09-10 |
EP1595871A2 (en) | 2005-11-16 |
DE60022050T2 (de) | 2006-06-14 |
HK1048635A1 (zh) | 2003-04-11 |
AU5178000A (en) | 2000-12-18 |
ES2249272T3 (es) | 2006-04-01 |
WO2000073283A1 (en) | 2000-12-07 |
CN1789246A (zh) | 2006-06-21 |
AU778063B2 (en) | 2004-11-11 |
JP2003500480A (ja) | 2003-01-07 |
ATE302194T1 (de) | 2005-09-15 |
DE60022050D1 (de) | 2005-09-22 |
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