IL142502A0 - Intermediates for the preparation of biologically active benzothiazolone ethanamines - Google Patents
Intermediates for the preparation of biologically active benzothiazolone ethanaminesInfo
- Publication number
- IL142502A0 IL142502A0 IL14250296A IL14250296A IL142502A0 IL 142502 A0 IL142502 A0 IL 142502A0 IL 14250296 A IL14250296 A IL 14250296A IL 14250296 A IL14250296 A IL 14250296A IL 142502 A0 IL142502 A0 IL 142502A0
- Authority
- IL
- Israel
- Prior art keywords
- ethanamines
- intermediates
- preparation
- biologically active
- benzothiazolone
- Prior art date
Links
- OUSFTHZQIKIJGG-UHFFFAOYSA-N 1,3-benzothiazole 1-oxide ethanamine Chemical class CCN.C1=CC=C2S(=O)C=NC2=C1 OUSFTHZQIKIJGG-UHFFFAOYSA-N 0.000 title 1
- 239000000543 intermediate Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pulmonology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9526511.2A GB9526511D0 (en) | 1995-12-23 | 1995-12-23 | Pharmaceutically active compounds |
| PCT/SE1996/001650 WO1997023470A1 (en) | 1995-12-23 | 1996-12-13 | Biologically active benzothiazolone ethanamines |
| IL12499896A IL124998A0 (en) | 1995-12-23 | 1996-12-13 | Biologically active benzothiazolone ethanamines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL142502A0 true IL142502A0 (en) | 2002-03-10 |
Family
ID=10786064
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL14250296A IL142502A0 (en) | 1995-12-23 | 1996-12-13 | Intermediates for the preparation of biologically active benzothiazolone ethanamines |
| IL12499896A IL124998A0 (en) | 1995-12-23 | 1996-12-13 | Biologically active benzothiazolone ethanamines |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL12499896A IL124998A0 (en) | 1995-12-23 | 1996-12-13 | Biologically active benzothiazolone ethanamines |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US5929100A (cs) |
| EP (1) | EP0918760B1 (cs) |
| JP (1) | JP2000502681A (cs) |
| KR (1) | KR19990076688A (cs) |
| CN (1) | CN1072214C (cs) |
| AR (1) | AR005008A1 (cs) |
| AT (1) | ATE209638T1 (cs) |
| AU (1) | AU704506B2 (cs) |
| BR (1) | BR9612234A (cs) |
| CA (1) | CA2238877A1 (cs) |
| CZ (1) | CZ288704B6 (cs) |
| DE (1) | DE69617472D1 (cs) |
| EE (1) | EE03440B1 (cs) |
| GB (1) | GB9526511D0 (cs) |
| HU (1) | HUP9900100A3 (cs) |
| IL (2) | IL142502A0 (cs) |
| IS (1) | IS4759A (cs) |
| MX (1) | MX9804828A (cs) |
| NO (1) | NO982927D0 (cs) |
| NZ (1) | NZ325500A (cs) |
| PL (1) | PL327475A1 (cs) |
| RU (1) | RU2177476C2 (cs) |
| SK (1) | SK82098A3 (cs) |
| TR (1) | TR199801196T2 (cs) |
| TW (1) | TW401411B (cs) |
| WO (1) | WO1997023470A1 (cs) |
| ZA (1) | ZA9610354B (cs) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999009018A1 (en) * | 1997-08-14 | 1999-02-25 | Kirin Beer Kabushiki Kaisha | BENZOTHIAZOLONE DERIVATIVES HAVING SELECTIVE β2 RECEPTOR AGONIST ACTIVITY |
| GB0218629D0 (en) * | 2002-08-09 | 2002-09-18 | Novartis Ag | Organic compounds |
| AR040962A1 (es) * | 2002-08-09 | 2005-04-27 | Novartis Ag | Compuestos derivados de tiazol 1,3-2-ona, composicion farmaceutica y proceso de preparacion del compuesto |
| DE602004021959D1 (de) * | 2003-11-21 | 2009-08-20 | Theravance Inc | Verbindungen mit agonistischer wirkung am beta2-adrenergen rezeptor und am muscarinischen rezeptor |
| TW200738658A (en) | 2005-08-09 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
| TW200738659A (en) * | 2005-08-29 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
| TW200745067A (en) | 2006-03-14 | 2007-12-16 | Astrazeneca Ab | Novel compounds |
| TW200833670A (en) | 2006-12-20 | 2008-08-16 | Astrazeneca Ab | Novel compounds 569 |
| GB0702458D0 (en) | 2007-02-08 | 2007-03-21 | Astrazeneca Ab | Salts 668 |
| AU2009260899B2 (en) | 2008-06-18 | 2012-02-23 | Astrazeneca Ab | Benzoxazinone derivatives acting as beta2-adrenoreceptor agonist for the treatment of respiratory disorders |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4314944A (en) * | 1980-08-22 | 1982-02-09 | Smithkline Corporation | 4-Aminoalkyl-7-hydroxy-2(3H)-indolones |
| US4452808A (en) * | 1982-12-07 | 1984-06-05 | Smithkline Beckman Corporation | 4-Aminoalkyl-2(3H)-indolones |
| GB8426200D0 (en) * | 1984-10-17 | 1984-11-21 | Glaxo Holdings Ltd | Chemical compounds |
| US4554287A (en) * | 1984-09-12 | 1985-11-19 | Smithkline Beckman Corporation | Antihypertensive 7-[2-(dialkylamino)ethyl]-4-hydroxy-1,3-benzimidazol-2-ones |
| US4554284A (en) * | 1984-09-12 | 1985-11-19 | Smithkline Beckman Corporation | 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones |
| EP0180994A3 (en) * | 1984-11-08 | 1987-09-23 | Syntex (U.S.A.) Inc. | Antihypertensive dialkyl aminoethylaniline derivatives |
| DE3728695A1 (de) * | 1987-08-25 | 1989-03-09 | Schering Ag | Neue benzimidazol-derivate |
| GB9211172D0 (en) * | 1992-05-27 | 1992-07-08 | Fisons Plc | Compounds |
| IE914003A1 (en) * | 1990-11-20 | 1992-05-20 | Astra Pharma Prod | Biologically Active Amines |
| GB9210632D0 (en) * | 1992-05-19 | 1992-07-01 | Fisons Plc | Compounds |
| US5648370A (en) * | 1990-11-20 | 1997-07-15 | Astra Pharmaceuticals Limited | 7-(2-aminoethyl) benzothiazolones |
-
1995
- 1995-12-23 GB GBGB9526511.2A patent/GB9526511D0/en active Pending
-
1996
- 1996-12-09 AR ARP960105568A patent/AR005008A1/es unknown
- 1996-12-09 ZA ZA9610354A patent/ZA9610354B/xx unknown
- 1996-12-11 TW TW085115316A patent/TW401411B/zh not_active IP Right Cessation
- 1996-12-13 HU HU9900100A patent/HUP9900100A3/hu unknown
- 1996-12-13 RU RU98114080/04A patent/RU2177476C2/ru active
- 1996-12-13 CZ CZ19981684A patent/CZ288704B6/cs not_active IP Right Cessation
- 1996-12-13 EE EE9800193A patent/EE03440B1/xx not_active IP Right Cessation
- 1996-12-13 WO PCT/SE1996/001650 patent/WO1997023470A1/en not_active Ceased
- 1996-12-13 US US08/793,706 patent/US5929100A/en not_active Expired - Fee Related
- 1996-12-13 SK SK820-98A patent/SK82098A3/sk unknown
- 1996-12-13 BR BR9612234A patent/BR9612234A/pt not_active Application Discontinuation
- 1996-12-13 IL IL14250296A patent/IL142502A0/xx unknown
- 1996-12-13 AU AU14025/97A patent/AU704506B2/en not_active Ceased
- 1996-12-13 EP EP96944153A patent/EP0918760B1/en not_active Expired - Lifetime
- 1996-12-13 TR TR1998/01196T patent/TR199801196T2/xx unknown
- 1996-12-13 KR KR1019980704800A patent/KR19990076688A/ko not_active Withdrawn
- 1996-12-13 IL IL12499896A patent/IL124998A0/xx unknown
- 1996-12-13 AT AT96944153T patent/ATE209638T1/de not_active IP Right Cessation
- 1996-12-13 NZ NZ325500A patent/NZ325500A/xx unknown
- 1996-12-13 CA CA002238877A patent/CA2238877A1/en not_active Abandoned
- 1996-12-13 JP JP09523560A patent/JP2000502681A/ja active Pending
- 1996-12-13 CN CN96199237A patent/CN1072214C/zh not_active Expired - Fee Related
- 1996-12-13 PL PL96327475A patent/PL327475A1/xx unknown
- 1996-12-13 DE DE69617472T patent/DE69617472D1/de not_active Expired - Lifetime
-
1998
- 1998-05-27 IS IS4759A patent/IS4759A/is unknown
- 1998-06-16 MX MX9804828A patent/MX9804828A/es unknown
- 1998-06-23 NO NO982927A patent/NO982927D0/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EE9800193A (et) | 1998-12-15 |
| EP0918760B1 (en) | 2001-11-28 |
| EP0918760A1 (en) | 1999-06-02 |
| JP2000502681A (ja) | 2000-03-07 |
| CA2238877A1 (en) | 1997-07-03 |
| US5929100A (en) | 1999-07-27 |
| NZ325500A (en) | 1999-01-28 |
| ZA9610354B (en) | 1997-06-23 |
| TR199801196T2 (xx) | 1998-10-21 |
| EE03440B1 (et) | 2001-06-15 |
| ATE209638T1 (de) | 2001-12-15 |
| KR19990076688A (ko) | 1999-10-15 |
| HUP9900100A3 (en) | 2001-10-29 |
| CZ168498A3 (cs) | 1998-09-16 |
| TW401411B (en) | 2000-08-11 |
| MX9804828A (es) | 1998-09-30 |
| SK82098A3 (en) | 1998-11-04 |
| NO982927L (no) | 1998-06-23 |
| CN1211242A (zh) | 1999-03-17 |
| NO982927D0 (no) | 1998-06-23 |
| AU1402597A (en) | 1997-07-17 |
| AR005008A1 (es) | 1999-04-07 |
| HUP9900100A2 (hu) | 1999-05-28 |
| WO1997023470A1 (en) | 1997-07-03 |
| IL124998A0 (en) | 1999-01-26 |
| AU704506B2 (en) | 1999-04-22 |
| DE69617472D1 (de) | 2002-01-10 |
| IS4759A (is) | 1998-05-27 |
| CN1072214C (zh) | 2001-10-03 |
| GB9526511D0 (en) | 1996-02-28 |
| BR9612234A (pt) | 1999-07-13 |
| CZ288704B6 (cs) | 2001-08-15 |
| RU2177476C2 (ru) | 2001-12-27 |
| PL327475A1 (en) | 1998-12-07 |
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