IL130397A - Preparation of Ä1S-Ä1alpha,2beta,3beta,4alpha (S*)ÜÜ-4-Ä7-ÄÄ-3-chloro-2-thienyl)methylÜpropylÜaminoÜ-3H-imidazo Ä4,5-BÜpyridin-3-ylÜ-N-ethyl-2,3 dihydroxycyclopentane carboxamide - Google Patents
Preparation of Ä1S-Ä1alpha,2beta,3beta,4alpha (S*)ÜÜ-4-Ä7-ÄÄ-3-chloro-2-thienyl)methylÜpropylÜaminoÜ-3H-imidazo Ä4,5-BÜpyridin-3-ylÜ-N-ethyl-2,3 dihydroxycyclopentane carboxamideInfo
- Publication number
- IL130397A IL130397A IL13039797A IL13039797A IL130397A IL 130397 A IL130397 A IL 130397A IL 13039797 A IL13039797 A IL 13039797A IL 13039797 A IL13039797 A IL 13039797A IL 130397 A IL130397 A IL 130397A
- Authority
- IL
- Israel
- Prior art keywords
- ä1alpha
- ylü
- methylüpropylüaminoü
- büpyridin
- 2beta
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/69—Two or more oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IL15292197A IL152921A (en) | 1996-12-11 | 1997-11-24 | Preparation of 4-hydroxy-3-nitro-2(1h)-pyridone from 2-hydroxy-3-cyano-4-methoxypyridine |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US3276496P | 1996-12-11 | 1996-12-11 | |
PCT/US1997/021439 WO1998025921A1 (en) | 1996-12-11 | 1997-11-24 | PREPARATION OF [1S-[1a,2b,3b,4a(S*)]]-4-[7-[[1-(3-CHLORO-2-THIENYL) METHYL]PROPYL]AMINO]-3H-IMIDAZO[4,5-b]PYRIDIN-3-yl]-N-ETHYL-2,3-DIHYDROXYCYCLOPENTANECARBOXAMIDE |
Publications (2)
Publication Number | Publication Date |
---|---|
IL130397A0 IL130397A0 (en) | 2000-06-01 |
IL130397A true IL130397A (en) | 2005-11-20 |
Family
ID=21866680
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL13039797A IL130397A (en) | 1996-12-11 | 1997-11-24 | Preparation of Ä1S-Ä1alpha,2beta,3beta,4alpha (S*)ÜÜ-4-Ä7-ÄÄ-3-chloro-2-thienyl)methylÜpropylÜaminoÜ-3H-imidazo Ä4,5-BÜpyridin-3-ylÜ-N-ethyl-2,3 dihydroxycyclopentane carboxamide |
Country Status (27)
Country | Link |
---|---|
US (2) | US6143894A (zh) |
EP (2) | EP0946550B1 (zh) |
JP (1) | JP2001506626A (zh) |
KR (4) | KR20060002030A (zh) |
CN (3) | CN1191251C (zh) |
AP (1) | AP1063A (zh) |
AT (1) | ATE301120T1 (zh) |
AU (1) | AU738581B2 (zh) |
BG (1) | BG63805B1 (zh) |
BR (1) | BR9713705A (zh) |
CA (1) | CA2274630C (zh) |
DE (1) | DE69733897T2 (zh) |
DK (1) | DK0946550T3 (zh) |
EA (1) | EA001989B1 (zh) |
ES (1) | ES2242984T3 (zh) |
HK (2) | HK1023998A1 (zh) |
HU (1) | HUP0000342A3 (zh) |
IL (1) | IL130397A (zh) |
MX (1) | MXPA03006730A (zh) |
NO (2) | NO319722B1 (zh) |
OA (1) | OA11061A (zh) |
PT (1) | PT946550E (zh) |
SI (1) | SI0946550T1 (zh) |
SK (1) | SK71199A3 (zh) |
UA (1) | UA54479C2 (zh) |
WO (1) | WO1998025921A1 (zh) |
ZA (1) | ZA9711035B (zh) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2228163T3 (es) | 1998-12-31 | 2005-04-01 | Aventis Pharmaceuticals Inc. | Procedimiento para preparar derivados de desaza-adenosina n6-sustituidos. |
US7291603B2 (en) * | 2002-07-24 | 2007-11-06 | Ptc Therapeutics, Inc. | Nucleoside compounds and their use for treating cancer and diseases associated with somatic mutations |
FR2846656B1 (fr) * | 2002-11-05 | 2004-12-24 | Servier Lab | Nouveaux derives d'imidazopyridine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2095960T3 (es) * | 1990-09-25 | 1997-03-01 | Rhone Poulenc Rorer Int | Compuestos que tienen propiedades antihipertensivas y antiisquemicas. |
HUP0100179A3 (en) * | 1997-07-03 | 2002-12-28 | Bristol Myers Squibb Pharma Co | Imidazopyrimidine and imidazopyridine derivatives and pharmaceutical compositions thereof |
CZ20012283A3 (cs) * | 1998-12-21 | 2001-10-17 | Aventis Pharmaceuticals Products Inc. | Způsob přípravy derivátů deaza-adenosinů substituovaných v poloze N6 |
-
1997
- 1997-11-24 UA UA99073906A patent/UA54479C2/uk unknown
- 1997-11-24 DE DE69733897T patent/DE69733897T2/de not_active Expired - Fee Related
- 1997-11-24 PT PT97950663T patent/PT946550E/pt unknown
- 1997-11-24 CN CNB011370718A patent/CN1191251C/zh not_active Expired - Fee Related
- 1997-11-24 ES ES97950663T patent/ES2242984T3/es not_active Expired - Lifetime
- 1997-11-24 CA CA002274630A patent/CA2274630C/en not_active Expired - Fee Related
- 1997-11-24 MX MXPA03006730A patent/MXPA03006730A/es not_active Application Discontinuation
- 1997-11-24 HU HU0000342A patent/HUP0000342A3/hu unknown
- 1997-11-24 DK DK97950663T patent/DK0946550T3/da active
- 1997-11-24 BR BR9713705-7A patent/BR9713705A/pt not_active Application Discontinuation
- 1997-11-24 EA EA199900527A patent/EA001989B1/ru not_active IP Right Cessation
- 1997-11-24 JP JP52670598A patent/JP2001506626A/ja not_active Ceased
- 1997-11-24 IL IL13039797A patent/IL130397A/xx not_active IP Right Cessation
- 1997-11-24 EP EP97950663A patent/EP0946550B1/en not_active Expired - Lifetime
- 1997-11-24 CN CN2005100037721A patent/CN1660842A/zh active Pending
- 1997-11-24 AP APAP/P/1999/001550A patent/AP1063A/en active
- 1997-11-24 EP EP05075298A patent/EP1609791A1/en not_active Withdrawn
- 1997-11-24 WO PCT/US1997/021439 patent/WO1998025921A1/en not_active Application Discontinuation
- 1997-11-24 KR KR1020057023522A patent/KR20060002030A/ko not_active Application Discontinuation
- 1997-11-24 SI SI9730709T patent/SI0946550T1/xx unknown
- 1997-11-24 KR KR1020057023521A patent/KR20060002029A/ko not_active Application Discontinuation
- 1997-11-24 CN CN97180580A patent/CN1090630C/zh not_active Expired - Fee Related
- 1997-11-24 AT AT97950663T patent/ATE301120T1/de not_active IP Right Cessation
- 1997-11-24 KR KR10-1999-7005191A patent/KR100510389B1/ko not_active IP Right Cessation
- 1997-11-24 KR KR1020057004675A patent/KR100571690B1/ko not_active IP Right Cessation
- 1997-11-24 SK SK711-99A patent/SK71199A3/sk unknown
- 1997-11-24 AU AU53607/98A patent/AU738581B2/en not_active Ceased
- 1997-12-09 ZA ZA9711035A patent/ZA9711035B/xx unknown
-
1999
- 1999-01-19 US US09/233,591 patent/US6143894A/en not_active Expired - Fee Related
- 1999-06-09 NO NO19992795A patent/NO319722B1/no unknown
- 1999-06-11 OA OA9900123A patent/OA11061A/en unknown
- 1999-06-11 BG BG103484A patent/BG63805B1/bg unknown
-
2000
- 2000-05-30 HK HK00103182A patent/HK1023998A1/xx not_active IP Right Cessation
- 2000-07-28 US US09/627,657 patent/US6235909B1/en not_active Expired - Fee Related
-
2003
- 2003-06-11 HK HK03104142A patent/HK1051862A1/xx not_active IP Right Cessation
-
2005
- 2005-05-12 NO NO20052327A patent/NO20052327D0/no unknown
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
GB2319250B (en) | Derivatives of 6,8-Difluoro-7-Hydroxycoumarin | |
PL338563A1 (en) | Substituted derivatives of 1,2,3,4-tetrahydronaphtalene | |
AU1450900A (en) | Methods of treatment of type 2 diabetes | |
PL327998A1 (en) | Novel derivatives of 19-nor-pregnene | |
PL324992A1 (en) | Novel derivatives of 2,3-dioxotetrahydoquinoxaline | |
PL329121A1 (en) | Substituted derivatives of 1,2,3,4-tetrahydronaphtalene | |
AU3284395A (en) | Synthesis of 1,1,1,3,3,-pentafluoropropane | |
AU4329396A (en) | Use of 3,4-diphenylchromans | |
AU1189399A (en) | Bathocuproine treatment of neurologic disease | |
PL340372A1 (en) | Novel 3,6x-hemiketals of 9a-azalydes class | |
ZA964129B (en) | N-acyl-2-aryl cyclopropylmethylamine derivatives as melatonerigics | |
PL312692A1 (en) | New derivatives of dialkoxy-pyridinol-benzimidazole | |
PL319270A1 (en) | Novel derivative of 2,3-dibenzodiazepin, method of obtaining them and pharmaceutic composition | |
HU9702480D0 (en) | New polymorphe modification of doxazosin-mesylate | |
GR3031738T3 (en) | Process for the preparation of 1,1-difluoroethane | |
AU2497595A (en) | New uses of difluoromethoxy-2,2,2-trifluoroethane | |
IL130397A (en) | Preparation of Ä1S-Ä1alpha,2beta,3beta,4alpha (S*)ÜÜ-4-Ä7-ÄÄ-3-chloro-2-thienyl)methylÜpropylÜaminoÜ-3H-imidazo Ä4,5-BÜpyridin-3-ylÜ-N-ethyl-2,3 dihydroxycyclopentane carboxamide | |
AU4361696A (en) | New uses of indolo-{2,3b}-quinoxalines | |
HU9702479D0 (en) | New polymorphe modification of doxazosin-mesylate | |
ZA945717B (en) | Preparation of electrode | |
ZA95694B (en) | Novel derivatives of tetramethylcyclopropane | |
AU7724194A (en) | Preparation of 1,1,2,3,3-pentafluoropropane | |
ZA965276B (en) | Carboxamide derivatives | |
IL119744A0 (en) | Use of 8,9-dehydroestrone | |
PL330141A1 (en) | Novel derivatives of 10,11-dihydro-10-oxo-5h-dibezyl(b,f)-azepin-5-carboxagmide |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FF | Patent granted | ||
MM9K | Patent not in force due to non-payment of renewal fees |