IL124213A - Sulfation of estrogen mixtures - Google Patents

Sulfation of estrogen mixtures

Info

Publication number
IL124213A
IL124213A IL12421398A IL12421398A IL124213A IL 124213 A IL124213 A IL 124213A IL 12421398 A IL12421398 A IL 12421398A IL 12421398 A IL12421398 A IL 12421398A IL 124213 A IL124213 A IL 124213A
Authority
IL
Israel
Prior art keywords
mixture
equilin
delta
compounds
estradiol
Prior art date
Application number
IL12421398A
Other languages
English (en)
Hebrew (he)
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of IL124213A publication Critical patent/IL124213A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J31/00Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J21/00Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005Ketals
    • C07J21/008Ketals at position 17
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
IL12421398A 1997-05-02 1998-04-24 Sulfation of estrogen mixtures IL124213A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP97201333 1997-05-02

Publications (1)

Publication Number Publication Date
IL124213A true IL124213A (en) 2004-12-15

Family

ID=8228294

Family Applications (1)

Application Number Title Priority Date Filing Date
IL12421398A IL124213A (en) 1997-05-02 1998-04-24 Sulfation of estrogen mixtures

Country Status (21)

Country Link
EP (1) EP0875515B1 (ja)
JP (1) JP4361976B2 (ja)
KR (1) KR100500498B1 (ja)
CN (1) CN1142175C (ja)
AR (1) AR012632A1 (ja)
AT (1) ATE277070T1 (ja)
AU (1) AU733743B2 (ja)
CA (1) CA2236648C (ja)
CZ (1) CZ293620B6 (ja)
DE (1) DE69826356T2 (ja)
DK (1) DK0875515T3 (ja)
ES (1) ES2230653T3 (ja)
HU (1) HUP9801018A3 (ja)
IL (1) IL124213A (ja)
NO (1) NO315654B1 (ja)
NZ (1) NZ330336A (ja)
PL (1) PL185664B1 (ja)
PT (1) PT875515E (ja)
RU (1) RU2184741C2 (ja)
TR (1) TR199800769A1 (ja)
ZA (1) ZA983631B (ja)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7335650B2 (en) 2000-01-14 2008-02-26 Sterix Limited Composition
US20030158432A1 (en) * 2002-01-08 2003-08-21 Leonard Thomas W. Synthesis of a mixture of sulfated estrogens using a sulfur trioxide complex

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB697531A (en) * 1951-04-17 1953-09-23 S B Penick & Company Improvements in or relating to the preparation of estrane sulfate salts
US5210081A (en) * 1992-02-26 1993-05-11 American Home Products Corporation Alkali metal 8,9-dehydroestrone sulfate esters
DE4334823C2 (de) * 1993-10-09 1998-09-17 Schering Ag Verfahren zur Herstellung von Schwefelsäurehalbestern von Estrogenen
US5395831A (en) * 1994-04-08 1995-03-07 American Home Products Corporation Treating cardiac disorders with Δ9(11)-dehydro-8-isoestrone
ZA968873B (en) * 1995-11-06 1997-05-28 Akzo Nobel Nv Isomerisation of equillin

Also Published As

Publication number Publication date
AU6376398A (en) 1998-11-05
NO981966D0 (no) 1998-04-30
KR100500498B1 (ko) 2005-10-25
CZ134098A3 (cs) 1998-11-11
EP0875515A2 (en) 1998-11-04
AR012632A1 (es) 2000-11-08
DK0875515T3 (da) 2005-01-10
EP0875515B1 (en) 2004-09-22
ATE277070T1 (de) 2004-10-15
DE69826356T2 (de) 2006-02-16
PT875515E (pt) 2005-01-31
HUP9801018A2 (hu) 1999-01-28
NO981966L (no) 1998-11-03
CN1201038A (zh) 1998-12-09
DE69826356D1 (de) 2004-10-28
ZA983631B (en) 1998-10-30
TR199800769A1 (xx) 1998-11-23
PL185664B1 (pl) 2003-06-30
ES2230653T3 (es) 2005-05-01
CA2236648C (en) 2007-09-18
KR19980086676A (ko) 1998-12-05
JPH1149795A (ja) 1999-02-23
PL326104A1 (en) 1998-11-09
NZ330336A (en) 1999-10-28
NO315654B1 (no) 2003-10-06
AU733743B2 (en) 2001-05-24
CZ293620B6 (cs) 2004-06-16
JP4361976B2 (ja) 2009-11-11
RU2184741C2 (ru) 2002-07-10
CA2236648A1 (en) 1998-11-02
EP0875515A3 (en) 1998-11-25
HUP9801018A3 (en) 2000-01-28
CN1142175C (zh) 2004-03-17

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees