IL113254A - Substituted azolone derivatives their preparation and pharmaceutical compositions containing them - Google Patents
Substituted azolone derivatives their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL113254A IL113254A IL11325495A IL11325495A IL113254A IL 113254 A IL113254 A IL 113254A IL 11325495 A IL11325495 A IL 11325495A IL 11325495 A IL11325495 A IL 11325495A IL 113254 A IL113254 A IL 113254A
- Authority
- IL
- Israel
- Prior art keywords
- image
- pct
- 4alkyl
- 6alkyl
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/70—One oxygen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/12—Oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Detergent Compositions (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Cephalosporin Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP94200938 | 1994-04-06 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL113254A0 IL113254A0 (en) | 1995-07-31 |
| IL113254A true IL113254A (en) | 1999-03-12 |
Family
ID=8216773
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL11325495A IL113254A (en) | 1994-04-06 | 1995-04-05 | Substituted azolone derivatives their preparation and pharmaceutical compositions containing them |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US5710156A (fi) |
| EP (1) | EP0754180B1 (fi) |
| JP (1) | JPH09511513A (fi) |
| CN (1) | CN1145067A (fi) |
| AT (1) | ATE207910T1 (fi) |
| AU (1) | AU685935B2 (fi) |
| BR (1) | BR9507289A (fi) |
| CA (1) | CA2185552A1 (fi) |
| CZ (1) | CZ287596A3 (fi) |
| DE (1) | DE69523581T2 (fi) |
| EE (1) | EE9600142A (fi) |
| FI (1) | FI963995A0 (fi) |
| HU (1) | HUT76287A (fi) |
| IL (1) | IL113254A (fi) |
| NO (1) | NO964216D0 (fi) |
| NZ (1) | NZ283346A (fi) |
| PL (1) | PL316655A1 (fi) |
| SK (1) | SK127196A3 (fi) |
| WO (1) | WO1995027704A1 (fi) |
| ZA (1) | ZA952810B (fi) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6326384B1 (en) | 1999-08-26 | 2001-12-04 | Robert R. Whittle | Dry blend pharmaceutical unit dosage form |
| US6262086B1 (en) | 1999-08-26 | 2001-07-17 | Robert R. Whittle | Pharmaceutical unit dosage form |
| US6316020B1 (en) | 1999-08-26 | 2001-11-13 | Robert R. Whittle | Pharmaceutical formulations |
| US6312723B1 (en) | 1999-08-26 | 2001-11-06 | Robert R. Whittle | Pharmaceutical unit dosage form |
| US6268385B1 (en) | 1999-08-26 | 2001-07-31 | Robert R. Whittle | Dry blend pharmaceutical formulations |
| US6312712B1 (en) | 1999-08-26 | 2001-11-06 | Robert R. Whittle | Method of improving bioavailability |
| US6780880B1 (en) * | 1999-08-26 | 2004-08-24 | Robert R. Whittle | FT-Raman spectroscopic measurement |
| US6262085B1 (en) | 1999-08-26 | 2001-07-17 | Robert R. Whittle | Alkoxy substituted Benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same |
| US6369087B1 (en) | 1999-08-26 | 2002-04-09 | Robert R. Whittle | Alkoxy substituted benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4791111A (en) * | 1985-12-23 | 1988-12-13 | Janssen Pharmaceutica, N.V. | [[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having anti-microbial properties |
| CA1331757C (en) * | 1988-02-29 | 1994-08-30 | Janssen Pharmaceutica Naamloze Vennootschap | 5-lipoxygenase inhibiting 4-(4-phenyl-1-piperazinyl)phenols |
| US5250528A (en) * | 1989-08-02 | 1993-10-05 | Fujisawa Pharmaceutical Co., Ltd. | New aminopiperazine derivatives |
| CA2076257A1 (en) * | 1991-09-13 | 1993-03-14 | Jan Heeres | 4-¬4-¬4-(4-hydroxyphenyl)-1- piperazinyl|phenyl|-5-methyl-3h -1,2,4-triazol-3-one derivatives |
| US5202346A (en) * | 1992-02-25 | 1993-04-13 | American Home Products Corporation | Piperidinyl and piperazinyl derivatives |
| TW279864B (fi) * | 1993-02-19 | 1996-07-01 | Janssen Pharmaceutica Nv |
-
1995
- 1995-03-29 AT AT95914329T patent/ATE207910T1/de not_active IP Right Cessation
- 1995-03-29 JP JP7526047A patent/JPH09511513A/ja not_active Ceased
- 1995-03-29 HU HU9602725A patent/HUT76287A/hu unknown
- 1995-03-29 BR BR9507289A patent/BR9507289A/pt not_active Application Discontinuation
- 1995-03-29 EP EP95914329A patent/EP0754180B1/en not_active Expired - Lifetime
- 1995-03-29 CA CA002185552A patent/CA2185552A1/en not_active Abandoned
- 1995-03-29 US US08/716,397 patent/US5710156A/en not_active Expired - Fee Related
- 1995-03-29 EE EE9600142A patent/EE9600142A/xx unknown
- 1995-03-29 CZ CZ962875A patent/CZ287596A3/cs unknown
- 1995-03-29 WO PCT/EP1995/001184 patent/WO1995027704A1/en active IP Right Grant
- 1995-03-29 DE DE69523581T patent/DE69523581T2/de not_active Expired - Fee Related
- 1995-03-29 PL PL95316655A patent/PL316655A1/xx unknown
- 1995-03-29 SK SK1271-96A patent/SK127196A3/sk unknown
- 1995-03-29 NZ NZ283346A patent/NZ283346A/en unknown
- 1995-03-29 CN CN95192436A patent/CN1145067A/zh active Pending
- 1995-03-29 AU AU21371/95A patent/AU685935B2/en not_active Ceased
- 1995-04-05 ZA ZA952810A patent/ZA952810B/xx unknown
- 1995-04-05 IL IL11325495A patent/IL113254A/xx not_active IP Right Cessation
-
1996
- 1996-10-04 NO NO964216A patent/NO964216D0/no unknown
- 1996-10-04 FI FI963995A patent/FI963995A0/fi unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JPH09511513A (ja) | 1997-11-18 |
| HUT76287A (en) | 1997-07-28 |
| DE69523581D1 (de) | 2001-12-06 |
| WO1995027704A1 (en) | 1995-10-19 |
| MX9604610A (es) | 1997-11-29 |
| HU9602725D0 (en) | 1996-11-28 |
| FI963995A (fi) | 1996-10-04 |
| DE69523581T2 (de) | 2002-07-11 |
| ATE207910T1 (de) | 2001-11-15 |
| AU685935B2 (en) | 1998-01-29 |
| EP0754180A1 (en) | 1997-01-22 |
| FI963995A0 (fi) | 1996-10-04 |
| PL316655A1 (en) | 1997-02-03 |
| NO964216L (no) | 1996-10-04 |
| SK127196A3 (en) | 1997-05-07 |
| NZ283346A (en) | 1997-05-26 |
| CZ287596A3 (en) | 1997-01-15 |
| CA2185552A1 (en) | 1995-10-19 |
| IL113254A0 (en) | 1995-07-31 |
| BR9507289A (pt) | 1997-09-23 |
| NO964216D0 (no) | 1996-10-04 |
| ZA952810B (en) | 1996-10-07 |
| EP0754180B1 (en) | 2001-10-31 |
| CN1145067A (zh) | 1997-03-12 |
| AU2137195A (en) | 1995-10-30 |
| EE9600142A (et) | 1997-04-15 |
| US5710156A (en) | 1998-01-20 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| MM9K | Patent not in force due to non-payment of renewal fees |