IL113254A - Substituted azolone derivatives their preparation and pharmaceutical compositions containing them - Google Patents
Substituted azolone derivatives their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL113254A IL113254A IL11325495A IL11325495A IL113254A IL 113254 A IL113254 A IL 113254A IL 11325495 A IL11325495 A IL 11325495A IL 11325495 A IL11325495 A IL 11325495A IL 113254 A IL113254 A IL 113254A
- Authority
- IL
- Israel
- Prior art keywords
- image
- pct
- 4alkyl
- 6alkyl
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/70—One oxygen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D249/12—Oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Cephalosporin Compounds (AREA)
- Detergent Compositions (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP94200938 | 1994-04-06 |
Publications (2)
Publication Number | Publication Date |
---|---|
IL113254A0 IL113254A0 (en) | 1995-07-31 |
IL113254A true IL113254A (en) | 1999-03-12 |
Family
ID=8216773
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL11325495A IL113254A (en) | 1994-04-06 | 1995-04-05 | Substituted azolone derivatives their preparation and pharmaceutical compositions containing them |
Country Status (20)
Country | Link |
---|---|
US (1) | US5710156A (de) |
EP (1) | EP0754180B1 (de) |
JP (1) | JPH09511513A (de) |
CN (1) | CN1145067A (de) |
AT (1) | ATE207910T1 (de) |
AU (1) | AU685935B2 (de) |
BR (1) | BR9507289A (de) |
CA (1) | CA2185552A1 (de) |
CZ (1) | CZ287596A3 (de) |
DE (1) | DE69523581T2 (de) |
EE (1) | EE9600142A (de) |
FI (1) | FI963995A (de) |
HU (1) | HUT76287A (de) |
IL (1) | IL113254A (de) |
NO (1) | NO964216L (de) |
NZ (1) | NZ283346A (de) |
PL (1) | PL316655A1 (de) |
SK (1) | SK127196A3 (de) |
WO (1) | WO1995027704A1 (de) |
ZA (1) | ZA952810B (de) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6268385B1 (en) | 1999-08-26 | 2001-07-31 | Robert R. Whittle | Dry blend pharmaceutical formulations |
US6312723B1 (en) | 1999-08-26 | 2001-11-06 | Robert R. Whittle | Pharmaceutical unit dosage form |
US6262086B1 (en) | 1999-08-26 | 2001-07-17 | Robert R. Whittle | Pharmaceutical unit dosage form |
US6326384B1 (en) | 1999-08-26 | 2001-12-04 | Robert R. Whittle | Dry blend pharmaceutical unit dosage form |
US6262085B1 (en) | 1999-08-26 | 2001-07-17 | Robert R. Whittle | Alkoxy substituted Benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same |
US6316020B1 (en) | 1999-08-26 | 2001-11-13 | Robert R. Whittle | Pharmaceutical formulations |
US6780880B1 (en) * | 1999-08-26 | 2004-08-24 | Robert R. Whittle | FT-Raman spectroscopic measurement |
US6312712B1 (en) | 1999-08-26 | 2001-11-06 | Robert R. Whittle | Method of improving bioavailability |
US6369087B1 (en) | 1999-08-26 | 2002-04-09 | Robert R. Whittle | Alkoxy substituted benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4791111A (en) * | 1985-12-23 | 1988-12-13 | Janssen Pharmaceutica, N.V. | [[4-[4-(4-phenyl-1-piperazinyl)phenoxymethyl]-1,3-dioxolan-2-yl]methyl]-1H-imidazoles and 1H-1,2,4-triazoles having anti-microbial properties |
CA1331757C (en) * | 1988-02-29 | 1994-08-30 | Janssen Pharmaceutica Naamloze Vennootschap | 5-lipoxygenase inhibiting 4-(4-phenyl-1-piperazinyl)phenols |
US5250528A (en) * | 1989-08-02 | 1993-10-05 | Fujisawa Pharmaceutical Co., Ltd. | New aminopiperazine derivatives |
CA2076257A1 (en) * | 1991-09-13 | 1993-03-14 | Jan Heeres | 4-¬4-¬4-(4-hydroxyphenyl)-1- piperazinyl|phenyl|-5-methyl-3h -1,2,4-triazol-3-one derivatives |
US5202346A (en) * | 1992-02-25 | 1993-04-13 | American Home Products Corporation | Piperidinyl and piperazinyl derivatives |
TW279864B (de) * | 1993-02-19 | 1996-07-01 | Janssen Pharmaceutica Nv |
-
1995
- 1995-03-29 WO PCT/EP1995/001184 patent/WO1995027704A1/en active IP Right Grant
- 1995-03-29 BR BR9507289A patent/BR9507289A/pt not_active Application Discontinuation
- 1995-03-29 DE DE69523581T patent/DE69523581T2/de not_active Expired - Fee Related
- 1995-03-29 CZ CZ962875A patent/CZ287596A3/cs unknown
- 1995-03-29 US US08/716,397 patent/US5710156A/en not_active Expired - Fee Related
- 1995-03-29 SK SK1271-96A patent/SK127196A3/sk unknown
- 1995-03-29 JP JP7526047A patent/JPH09511513A/ja not_active Ceased
- 1995-03-29 CA CA002185552A patent/CA2185552A1/en not_active Abandoned
- 1995-03-29 EP EP95914329A patent/EP0754180B1/de not_active Expired - Lifetime
- 1995-03-29 HU HU9602725A patent/HUT76287A/hu unknown
- 1995-03-29 AU AU21371/95A patent/AU685935B2/en not_active Ceased
- 1995-03-29 NZ NZ283346A patent/NZ283346A/en unknown
- 1995-03-29 EE EE9600142A patent/EE9600142A/xx unknown
- 1995-03-29 PL PL95316655A patent/PL316655A1/xx unknown
- 1995-03-29 CN CN95192436A patent/CN1145067A/zh active Pending
- 1995-03-29 AT AT95914329T patent/ATE207910T1/de not_active IP Right Cessation
- 1995-04-05 ZA ZA952810A patent/ZA952810B/xx unknown
- 1995-04-05 IL IL11325495A patent/IL113254A/xx not_active IP Right Cessation
-
1996
- 1996-10-04 FI FI963995A patent/FI963995A/fi unknown
- 1996-10-04 NO NO964216A patent/NO964216L/no unknown
Also Published As
Publication number | Publication date |
---|---|
DE69523581T2 (de) | 2002-07-11 |
ZA952810B (en) | 1996-10-07 |
DE69523581D1 (de) | 2001-12-06 |
JPH09511513A (ja) | 1997-11-18 |
SK127196A3 (en) | 1997-05-07 |
BR9507289A (pt) | 1997-09-23 |
ATE207910T1 (de) | 2001-11-15 |
NO964216D0 (no) | 1996-10-04 |
EP0754180A1 (de) | 1997-01-22 |
FI963995A0 (fi) | 1996-10-04 |
EP0754180B1 (de) | 2001-10-31 |
NZ283346A (en) | 1997-05-26 |
HUT76287A (en) | 1997-07-28 |
HU9602725D0 (en) | 1996-11-28 |
IL113254A0 (en) | 1995-07-31 |
MX9604610A (es) | 1997-11-29 |
EE9600142A (et) | 1997-04-15 |
CN1145067A (zh) | 1997-03-12 |
CA2185552A1 (en) | 1995-10-19 |
AU685935B2 (en) | 1998-01-29 |
FI963995A (fi) | 1996-10-04 |
PL316655A1 (en) | 1997-02-03 |
WO1995027704A1 (en) | 1995-10-19 |
NO964216L (no) | 1996-10-04 |
AU2137195A (en) | 1995-10-30 |
US5710156A (en) | 1998-01-20 |
CZ287596A3 (en) | 1997-01-15 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IL114537A0 (en) | Sulfonamide derivatives of azolones their preparation and pharmaceutical compositions containing them | |
MX9700339A (es) | Derivados de azolona anti-helcobacter que contienen urea y tiourea. | |
MY117852A (en) | Alkylaminobenzothiazole and- benzoxazole derivatives | |
IL92358A0 (en) | Diaryl compounds,their preparation and pharmaceutical compositions containing them | |
IL113254A (en) | Substituted azolone derivatives their preparation and pharmaceutical compositions containing them | |
DE69720715D1 (en) | Hexahydro-pyrido (4,3-b)indolderivate als antipsychotische arzneimittel | |
IL124966A0 (en) | 1-indanyl- and 1-indanylidene-acetic derivatives | |
HUT43943A (en) | Herbicide compositions comprising urea derivatives as active substance and process for preparing such compounds | |
IL115184A0 (en) | Anthracycline derivatives their preparation and use | |
ES8103071A1 (es) | Procedimiento de preparacion de nuevos derivados aminicos del benzotiazol | |
DE2966809D1 (en) | 3,4-diaza-bicyclo(4.1.0)hepten-2-ones-5, process for their preparation and therapeutical compositions containing them | |
MY120046A (en) | Angiogenesis inhibiting thiadiazolyl pyridazine derivatives. | |
GR3025050T3 (en) | Etoposide derivatives, process for their preparation, their use as a drug and in the preparation of a drug for treating cancer. | |
TW261605B (de) | ||
ES8307778A1 (es) | Procedimiento para preparar difenilbutil-1-piperazinocarboxilatos. | |
MY118312A (en) | Angiogenesis inhibiting 5- substituted- 1,2,4- thiadiazolyl derivatives | |
ES8307798A1 (es) | Un procedimiento para la preparacion de derivados de piperazilmetil-4-dibenzofuranona, o, dibenzofuranol. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FF | Patent granted | ||
MM9K | Patent not in force due to non-payment of renewal fees |