IL108387A - Optically active beta-aminoalkoxyborane complex and its use in organic synthesis - Google Patents
Optically active beta-aminoalkoxyborane complex and its use in organic synthesisInfo
- Publication number
- IL108387A IL108387A IL10838794A IL10838794A IL108387A IL 108387 A IL108387 A IL 108387A IL 10838794 A IL10838794 A IL 10838794A IL 10838794 A IL10838794 A IL 10838794A IL 108387 A IL108387 A IL 108387A
- Authority
- IL
- Israel
- Prior art keywords
- optically active
- organic synthesis
- active beta
- aralkyl
- cycloalkyl
- Prior art date
Links
- 238000003786 synthesis reaction Methods 0.000 title 1
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 3
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 3
- 125000004209 (C1-C8) alkyl group Chemical group 0.000 abstract 2
- 125000000041 C6-C10 aryl group Chemical group 0.000 abstract 2
- PPBRXRYQALVLMV-UHFFFAOYSA-N Styrene Chemical compound C=CC1=CC=CC=C1 PPBRXRYQALVLMV-UHFFFAOYSA-N 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 1
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000005428 anthryl group Chemical group [H]C1=C([H])C([H])=C2C([H])=C3C(*)=C([H])C([H])=C([H])C3=C([H])C2=C1[H] 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000001624 naphthyl group Chemical group 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 125000005561 phenanthryl group Chemical group 0.000 abstract 1
- 229920000642 polymer Polymers 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B53/00—Asymmetric syntheses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C215/00—Compounds containing amino and hydroxy groups bound to the same carbon skeleton
- C07C215/02—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C215/22—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated
- C07C215/28—Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C29/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
- C07C29/132—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group
- C07C29/136—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group of >C=O containing groups, e.g. —COOH
- C07C29/143—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group of >C=O containing groups, e.g. —COOH of ketones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
- C07C67/31—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by introduction of functional groups containing oxygen only in singly bound form
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/12—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D215/14—Radicals substituted by oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
- C07F5/022—Boron compounds without C-boron linkages
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/02—Ortho- or ortho- and peri-condensed systems
- C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
- C07C2603/22—Ortho- or ortho- and peri-condensed systems containing three rings containing only six-membered rings
- C07C2603/24—Anthracenes; Hydrogenated anthracenes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/02—Ortho- or ortho- and peri-condensed systems
- C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
- C07C2603/22—Ortho- or ortho- and peri-condensed systems containing three rings containing only six-membered rings
- C07C2603/26—Phenanthrenes; Hydrogenated phenanthrenes
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP782793 | 1993-01-20 | ||
| JP6682593 | 1993-03-25 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL108387A0 IL108387A0 (en) | 1994-04-12 |
| IL108387A true IL108387A (en) | 2000-06-29 |
Family
ID=26342202
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL10838794A IL108387A (en) | 1993-01-20 | 1994-01-20 | Optically active beta-aminoalkoxyborane complex and its use in organic synthesis |
| IL11969696A IL119696A0 (en) | 1993-01-20 | 1996-11-26 | Optically active beta-aminoalcohols and process for their production |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL11969696A IL119696A0 (en) | 1993-01-20 | 1996-11-26 | Optically active beta-aminoalcohols and process for their production |
Country Status (18)
| Country | Link |
|---|---|
| US (6) | US5663348A (es) |
| EP (1) | EP0680484B1 (es) |
| JP (1) | JPH06329679A (es) |
| KR (1) | KR960700255A (es) |
| CN (2) | CN1047173C (es) |
| AT (1) | ATE169921T1 (es) |
| AU (1) | AU678427B2 (es) |
| CA (1) | CA2153695A1 (es) |
| CZ (1) | CZ185295A3 (es) |
| DE (1) | DE69412588T2 (es) |
| HU (1) | HU217182B (es) |
| IL (2) | IL108387A (es) |
| MX (1) | MX9400566A (es) |
| NO (2) | NO305602B1 (es) |
| NZ (1) | NZ259585A (es) |
| RU (1) | RU2126412C1 (es) |
| TW (1) | TW383309B (es) |
| WO (1) | WO1994017079A1 (es) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE146790T1 (de) * | 1992-05-14 | 1997-01-15 | Pfizer | Enantioselektive katalysatoren aus oxazaborolidin |
| JPH06329679A (ja) * | 1993-01-20 | 1994-11-29 | Nissan Chem Ind Ltd | 光学活性β−アミノアルコキシボラン錯体 |
| US5831132A (en) * | 1994-10-28 | 1998-11-03 | Sumika Fine Chemicals Company, Ltd. | Process for producing optically active carbinols |
| US6262283B1 (en) | 1996-12-06 | 2001-07-17 | Magainin Pharmaceuticals Inc. | Stereoselective synthesis of 24-hydroxylated compounds useful for the preparation of aminosterols, vitamin D analogs, and other compounds |
| CA2406847C (en) | 2000-04-12 | 2009-11-17 | Genaera Corporation | Regioselective and stereoselective oxidation of fused ring systems useful for the preparation of aminosterols |
| US6509472B2 (en) * | 2000-09-11 | 2003-01-21 | Schering Corporation | 4-Cyclohexyl-1,3,2-oxazaborolidine chiral accessories |
| US7173073B2 (en) * | 2002-01-14 | 2007-02-06 | Johnson & Johnson Vision Care, Inc. | Ophthalmic devices containing heterocyclic compounds and methods for their production |
| US7153889B2 (en) | 2002-11-12 | 2006-12-26 | Abbott Laboratories | Bicyclic-substituted amines as histamine-3 receptor ligands |
| US7098222B2 (en) | 2004-05-12 | 2006-08-29 | Abbott Laboratories | Bicyclic-substituted amines having cyclic-substituted monocyclic substituents |
| US7205316B2 (en) | 2004-05-12 | 2007-04-17 | Abbott Laboratories | Tri- and bi-cyclic heteroaryl histamine-3 receptor ligands |
| US7145005B2 (en) | 2004-05-12 | 2006-12-05 | Abbott Laboratories | 2-(6-{2-[(2R)-2-Methyl-1-pyrrolidin-1-yl]-ethyl}-2-naphthalen-2-yl)-2H-pyridazin-3-one salts and their preparation |
| TWI504394B (zh) | 2011-04-29 | 2015-10-21 | Ind Tech Res Inst | 安托芬之製備方法 |
| CA2837774A1 (en) | 2013-12-20 | 2015-06-20 | Heiner Ophardt | Piston pump with vacuum relief |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA772624A (en) * | 1967-11-28 | F. Crowther Albert | Substituted oxazolidines | |
| US2573606A (en) * | 1946-12-02 | 1951-10-30 | Parke Davis & Co | Lower alkyl and alkenyl n-(1-naphthyl methyl) n-hydroxyethyl amines |
| JPS57146786A (en) * | 1981-03-09 | 1982-09-10 | Kyowa Hakko Kogyo Co Ltd | Optically active borane compound and preparation of optically active compound using the same |
| GB8313571D0 (en) * | 1983-05-17 | 1983-06-22 | Wellcome Found | Chemical compounds |
| US4719055A (en) * | 1983-05-17 | 1988-01-12 | Burroughs Wellcome Co. | Phenanthrene derivatives |
| JPS6118790A (ja) * | 1984-07-05 | 1986-01-27 | Sumitomo Chem Co Ltd | 光学活性ボラン錯体およびその製造法 |
| JPH0778052B2 (ja) * | 1986-11-28 | 1995-08-23 | 富士薬品工業株式会社 | Ｄｌ−パントラクトンの光学分割法 |
| US4897490A (en) * | 1987-02-25 | 1990-01-30 | Bristol-Meyers Company | Antihypercholesterolemic tetrazole compounds |
| US5254692A (en) * | 1990-04-06 | 1993-10-19 | Bayer Aktiengesellschaft | 2,6-dialkyl-4-(benzothiazol- or benzoxazol-7-yl)-1,4-dihydropyridines |
| US5157129A (en) * | 1990-04-18 | 1992-10-20 | Merck & Co., Inc. | Enantiospecific synthesis of s-(+)-5,6-dihydro-4-(r-amino)-4h-thieno(2,3-b)thiopyran-2-sulfonamide-7,7-dioxide |
| ATE146790T1 (de) * | 1992-05-14 | 1997-01-15 | Pfizer | Enantioselektive katalysatoren aus oxazaborolidin |
| JPH06329679A (ja) * | 1993-01-20 | 1994-11-29 | Nissan Chem Ind Ltd | 光学活性β−アミノアルコキシボラン錯体 |
| DK0724552T3 (da) * | 1993-11-30 | 1997-12-22 | Pfizer | Fremgangsmåde til fremstilling af chiralt tetralon |
| DE69518497T2 (de) * | 1994-12-07 | 2001-04-19 | Japan Science And Technology Corp., Kawaguchi | Verfahren zur Herstellung eines Alkohols |
-
1993
- 1993-12-27 JP JP5332498A patent/JPH06329679A/ja active Pending
-
1994
- 1994-01-14 TW TW083100279A patent/TW383309B/zh not_active IP Right Cessation
- 1994-01-17 RU RU95115845A patent/RU2126412C1/ru active
- 1994-01-17 EP EP94904332A patent/EP0680484B1/en not_active Expired - Lifetime
- 1994-01-17 WO PCT/JP1994/000056 patent/WO1994017079A1/en not_active Application Discontinuation
- 1994-01-17 DE DE69412588T patent/DE69412588T2/de not_active Expired - Fee Related
- 1994-01-17 US US08/481,505 patent/US5663348A/en not_active Expired - Fee Related
- 1994-01-17 HU HU9502184A patent/HU217182B/hu not_active IP Right Cessation
- 1994-01-17 CA CA002153695A patent/CA2153695A1/en not_active Abandoned
- 1994-01-17 CZ CZ951852A patent/CZ185295A3/cs unknown
- 1994-01-17 CN CN94190966A patent/CN1047173C/zh not_active Expired - Fee Related
- 1994-01-17 AU AU58431/94A patent/AU678427B2/en not_active Ceased
- 1994-01-17 KR KR1019950702983A patent/KR960700255A/ko not_active Application Discontinuation
- 1994-01-17 NZ NZ259585A patent/NZ259585A/en unknown
- 1994-01-17 AT AT94904332T patent/ATE169921T1/de not_active IP Right Cessation
- 1994-01-20 MX MX9400566A patent/MX9400566A/es not_active Application Discontinuation
- 1994-01-20 IL IL10838794A patent/IL108387A/xx not_active IP Right Cessation
-
1995
- 1995-07-19 NO NO952870A patent/NO305602B1/no unknown
-
1996
- 1996-11-26 IL IL11969696A patent/IL119696A0/xx unknown
-
1997
- 1997-01-07 US US08/779,621 patent/US5767277A/en not_active Expired - Fee Related
- 1997-04-29 US US08/848,174 patent/US5852221A/en not_active Expired - Fee Related
- 1997-04-29 US US08/848,173 patent/US5739347A/en not_active Expired - Fee Related
- 1997-04-29 US US08/848,169 patent/US5808098A/en not_active Expired - Fee Related
- 1997-04-29 US US08/848,172 patent/US5786485A/en not_active Expired - Fee Related
-
1998
- 1998-10-28 NO NO985016A patent/NO985016D0/no not_active Application Discontinuation
-
1999
- 1999-04-09 CN CN99105088A patent/CN1234392A/zh active Pending
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| MM9K | Patent not in force due to non-payment of renewal fees |