IL105909A - Fungicidal compositions comprising indole derivatives, certain such novel compounds and their preparation - Google Patents
Fungicidal compositions comprising indole derivatives, certain such novel compounds and their preparationInfo
- Publication number
- IL105909A IL105909A IL105909A IL10590993A IL105909A IL 105909 A IL105909 A IL 105909A IL 105909 A IL105909 A IL 105909A IL 10590993 A IL10590993 A IL 10590993A IL 105909 A IL105909 A IL 105909A
- Authority
- IL
- Israel
- Prior art keywords
- group
- represent
- hydrogen atom
- atom
- phenyl
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 3
- 230000000855 fungicidal effect Effects 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 title abstract 2
- 229940054051 antipsychotic indole derivative Drugs 0.000 title 1
- 150000002475 indoles Chemical class 0.000 title 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 6
- -1 4-ethoxyphenyl Chemical group 0.000 abstract 3
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 3
- 125000003545 alkoxy group Chemical group 0.000 abstract 2
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 125000001041 indolyl group Chemical group 0.000 abstract 2
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 2
- 125000004182 2-chlorophenyl group Chemical group [H]C1=C([H])C(Cl)=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000004198 2-fluorophenyl group Chemical group [H]C1=C([H])C(F)=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000004172 4-methoxyphenyl group Chemical group [H]C1=C([H])C(OC([H])([H])[H])=C([H])C([H])=C1* 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 229910052801 chlorine Inorganic materials 0.000 abstract 1
- 125000001309 chloro group Chemical group Cl* 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 125000000040 m-tolyl group Chemical group [H]C1=C([H])C(*)=C([H])C(=C1[H])C([H])([H])[H] 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 125000003854 p-chlorophenyl group Chemical group [H]C1=C([H])C(*)=C([H])C([H])=C1Cl 0.000 abstract 1
- 125000001037 p-tolyl group Chemical group [H]C1=C([H])C(=C([H])C([H])=C1*)C([H])([H])[H] 0.000 abstract 1
- 125000000951 phenoxy group Chemical group [H]C1=C([H])C([H])=C(O*)C([H])=C1[H] 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/36—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings
- A01N43/38—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom five-membered rings condensed with carbocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP92109525 | 1992-06-05 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL105909A0 IL105909A0 (en) | 1993-10-20 |
| IL105909A true IL105909A (en) | 1997-04-15 |
Family
ID=8209683
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL105909A IL105909A (en) | 1992-06-05 | 1993-06-04 | Fungicidal compositions comprising indole derivatives, certain such novel compounds and their preparation |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US5399559A (Direct) |
| EP (1) | EP0643695B1 (Direct) |
| JP (1) | JP3296490B2 (Direct) |
| CN (1) | CN1082318A (Direct) |
| AT (1) | ATE141260T1 (Direct) |
| AU (1) | AU666558B2 (Direct) |
| DE (1) | DE69304057T2 (Direct) |
| DK (1) | DK0643695T3 (Direct) |
| ES (1) | ES2091615T3 (Direct) |
| GE (1) | GEP19981431B (Direct) |
| GR (1) | GR3020807T3 (Direct) |
| HU (1) | HU216814B (Direct) |
| IL (1) | IL105909A (Direct) |
| MD (1) | MD1743B2 (Direct) |
| TW (1) | TW229140B (Direct) |
| WO (1) | WO1993025524A1 (Direct) |
| ZA (1) | ZA933846B (Direct) |
Families Citing this family (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1997006141A1 (en) * | 1995-08-04 | 1997-02-20 | Otsuka Kagaku Kabushiki Kaisha | Indole-2-carboxylic ester derivatives and agricultural and horticultural bacteriocides containing the same as the active ingredient |
| US6353007B1 (en) * | 2000-07-13 | 2002-03-05 | Boehringer Ingelheim Pharmaceuticals, Inc. | Substituted 1-(4-aminophenyl)indoles and their use as anti-inflammatory agents |
| EP1314733A1 (en) | 2001-11-22 | 2003-05-28 | Aventis Pharma Deutschland GmbH | Indole-2-carboxamides as factor Xa inhibitors |
| EP1479677A1 (en) * | 2003-05-19 | 2004-11-24 | Aventis Pharma Deutschland GmbH | New indole derivatives as factor xa inhibitors |
| SE0302035D0 (sv) * | 2003-07-09 | 2003-07-09 | Biolipox Ab | New compound |
| DE602005014233D1 (de) * | 2004-06-18 | 2009-06-10 | Biolipox Ab | Zur behandlung von entzündungen geeignete indole |
| BRPI0512252A (pt) | 2004-06-18 | 2008-02-19 | Biolipox Ab | composto ou um sal farmaceuticamente aceitável do mesmo, formulação farmacêutica, uso de um composto, método de tratamento de uma doença, produto combinado, e, processo para a preparação de um composto |
| KR20070029809A (ko) * | 2004-06-18 | 2007-03-14 | 바이올리폭스 에이비 | 염증치료에 유용한 인돌 |
| JP2008527030A (ja) * | 2005-01-19 | 2008-07-24 | バイオリポックス エービー | 炎症の治療に有用なインドール類 |
| WO2006077401A1 (en) * | 2005-01-19 | 2006-07-27 | Biolipox Ab | Pyrrolopyridines useful in the treatment of inflammation |
| EP1844013A1 (en) * | 2005-01-19 | 2007-10-17 | Biolipox AB | Indoles useful in the treatment of inflammation |
| CA2593155A1 (en) | 2005-01-19 | 2006-07-27 | Biolipox Ab | Indoles useful in the treatment of inflammation |
| JP2008527032A (ja) * | 2005-01-19 | 2008-07-24 | バイオリポックス エービー | 炎症の治療に有用なチエノピロール |
| US20090042949A1 (en) * | 2005-01-19 | 2009-02-12 | Benjamin Pelcman | Indoles Useful in the Treatment of Inflammation |
| AR056690A1 (es) | 2005-10-14 | 2007-10-17 | Athersys Inc | Derivados de indol como inhibidores de indol como inhibidores del receptor 3 de histamina para el tartamiento de trastornos del sueno y cognitivos obesidad y otros trastornos de snc |
| WO2007109178A2 (en) * | 2006-03-16 | 2007-09-27 | Pharmacyclics, Inc. | Indole derivatives as inhibitors of histone deacetylase |
| EA020332B1 (ru) * | 2007-08-10 | 2014-10-30 | Х. Лундбекк А/С | Аналоги гетероариламидов |
| DK2448938T5 (en) | 2009-06-29 | 2015-10-05 | Incyte Corp | Pyrimidinones AS PI3K inhibitors |
| US8759359B2 (en) | 2009-12-18 | 2014-06-24 | Incyte Corporation | Substituted heteroaryl fused derivatives as PI3K inhibitors |
| AR081823A1 (es) | 2010-04-14 | 2012-10-24 | Incyte Corp | DERIVADOS FUSIONADOS COMO INHIBIDORES DE PI3Kd |
| US9062055B2 (en) | 2010-06-21 | 2015-06-23 | Incyte Corporation | Fused pyrrole derivatives as PI3K inhibitors |
| AR084366A1 (es) | 2010-12-20 | 2013-05-08 | Incyte Corp | N-(1-(fenil sustituido)etil)-9h-purin-6-aminas como inhibidores de pi3k |
| WO2012125629A1 (en) | 2011-03-14 | 2012-09-20 | Incyte Corporation | Substituted diamino-pyrimidine and diamino-pyridine derivatives as pi3k inhibitors |
| US9126948B2 (en) | 2011-03-25 | 2015-09-08 | Incyte Holdings Corporation | Pyrimidine-4,6-diamine derivatives as PI3K inhibitors |
| HRP20170285T1 (hr) | 2011-09-02 | 2017-04-21 | Incyte Holdings Corporation | Heterociklilamini kao inhibitori pi3k |
| AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
| US10077277B2 (en) | 2014-06-11 | 2018-09-18 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors |
| MX373232B (es) | 2015-02-27 | 2020-05-08 | Incyte Holdings Corp | Sales del inhibidor fosfoinositida 3-cinasa (pi3k) y procesos para su preparación. |
| WO2016183060A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
| US9988401B2 (en) | 2015-05-11 | 2018-06-05 | Incyte Corporation | Crystalline forms of a PI3K inhibitor |
| MX2020012826A (es) | 2018-06-01 | 2021-03-09 | Incyte Corp | Regimen de dosificacion para el tratamiento de trastornos relacionados con fosfatidilinositol 3-cinasas (pi3k). |
| EP4561991A1 (en) * | 2022-07-25 | 2025-06-04 | Cayman Chemical Company, Inc. | Novel heterocycles as spla2-x inhibitors |
| CN118546085B (zh) * | 2024-07-25 | 2024-12-03 | 西北农林科技大学深圳研究院 | 植物病害防治组合物及其制备方法和应用 |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1966206A1 (de) * | 1968-04-26 | 1972-01-20 | Sumitomo Chemical Co | 1,4-Benzodiazepine und Arzneipraeparate |
| US3634402A (en) * | 1968-04-26 | 1972-01-11 | Sumitomo Chemical Co | Process for producing 1 4-benzodiazepine derivatives and their salts |
| DE1935671C3 (de) * | 1968-04-26 | 1975-01-09 | Sumitomo Chemical Co | 2-Aminomethylindole und ihre Salze |
| GB1305458A (Direct) * | 1969-02-26 | 1973-01-31 | ||
| US3582285A (en) * | 1970-03-19 | 1971-06-01 | Xerox Corp | Chemical package |
| US4431307A (en) * | 1981-11-19 | 1984-02-14 | Labsystems Oy | Set of cuvettes |
| US4599315A (en) * | 1983-09-13 | 1986-07-08 | University Of California Regents | Microdroplet test apparatus |
| DE3677277D1 (de) * | 1985-02-08 | 1991-03-07 | Synthelabo | (dihydro-4,5-1h-imidazolyl-2)-2-dihydro-2,3-indolderivate, ihre herstellung und anwendung als heilmittel. |
| US4925629A (en) * | 1988-07-28 | 1990-05-15 | Bioquant, Inc. | Diagnostic device |
| US5147529A (en) * | 1988-08-10 | 1992-09-15 | E. I. Du Pont De Nemours And Company | Method for automatically processing magnetic solid phase reagents |
| US5041266A (en) * | 1989-12-21 | 1991-08-20 | Hoffmann-La Roche Inc. | Tray for immunometric determinations |
| JP2964182B2 (ja) * | 1991-09-10 | 1999-10-18 | 花王株式会社 | 象牙質知覚過敏治療剤 |
| JP2986256B2 (ja) * | 1991-09-12 | 1999-12-06 | 扶桑薬品工業株式会社 | 血液透析用顆粒剤 |
-
1993
- 1993-05-24 TW TW082104079A patent/TW229140B/zh active
- 1993-06-02 ZA ZA933846A patent/ZA933846B/xx unknown
- 1993-06-03 EP EP93912878A patent/EP0643695B1/en not_active Expired - Lifetime
- 1993-06-03 ES ES93912878T patent/ES2091615T3/es not_active Expired - Lifetime
- 1993-06-03 DK DK93912878.1T patent/DK0643695T3/da active
- 1993-06-03 AU AU43226/93A patent/AU666558B2/en not_active Ceased
- 1993-06-03 MD MD96-0305A patent/MD1743B2/ro unknown
- 1993-06-03 GE GEAP19932593A patent/GEP19981431B/en unknown
- 1993-06-03 HU HU9403475A patent/HU216814B/hu not_active IP Right Cessation
- 1993-06-03 WO PCT/EP1993/001406 patent/WO1993025524A1/en not_active Ceased
- 1993-06-03 US US08/071,894 patent/US5399559A/en not_active Expired - Lifetime
- 1993-06-03 JP JP50108994A patent/JP3296490B2/ja not_active Expired - Fee Related
- 1993-06-03 AT AT93912878T patent/ATE141260T1/de not_active IP Right Cessation
- 1993-06-03 DE DE69304057T patent/DE69304057T2/de not_active Expired - Fee Related
- 1993-06-04 IL IL105909A patent/IL105909A/xx not_active IP Right Cessation
- 1993-06-04 CN CN93108296A patent/CN1082318A/zh active Pending
-
1996
- 1996-08-16 GR GR960401179T patent/GR3020807T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DK0643695T3 (da) | 1996-09-02 |
| ES2091615T3 (es) | 1996-11-01 |
| MD1743B2 (ro) | 2001-09-30 |
| GR3020807T3 (en) | 1996-11-30 |
| TW229140B (Direct) | 1994-09-01 |
| IL105909A0 (en) | 1993-10-20 |
| EP0643695B1 (en) | 1996-08-14 |
| AU4322693A (en) | 1994-01-04 |
| JPH07507323A (ja) | 1995-08-10 |
| US5399559A (en) | 1995-03-21 |
| GEP19981431B (en) | 1998-10-30 |
| HU216814B (hu) | 1999-08-30 |
| DE69304057T2 (de) | 1997-02-06 |
| ZA933846B (en) | 1993-12-28 |
| AU666558B2 (en) | 1996-02-15 |
| ATE141260T1 (de) | 1996-08-15 |
| WO1993025524A1 (en) | 1993-12-23 |
| CN1082318A (zh) | 1994-02-23 |
| JP3296490B2 (ja) | 2002-07-02 |
| HUT69737A (en) | 1995-09-28 |
| EP0643695A1 (en) | 1995-03-22 |
| DE69304057D1 (de) | 1996-09-19 |
| HU9403475D0 (en) | 1995-03-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| RH1 | Patent not in force |