IL102702A - OPTICALLY ACTIVE g-HALO- 2-AMINOALKANECARBOXYLIC ACID DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THEIR USE FOR THE PREPARATION OF OPTICALLY ACTIVE PHOSPHORUS-CONTAINING a-AMINO ACIDS - Google Patents
OPTICALLY ACTIVE g-HALO- 2-AMINOALKANECARBOXYLIC ACID DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THEIR USE FOR THE PREPARATION OF OPTICALLY ACTIVE PHOSPHORUS-CONTAINING a-AMINO ACIDSInfo
- Publication number
- IL102702A IL102702A IL102702A IL10270292A IL102702A IL 102702 A IL102702 A IL 102702A IL 102702 A IL102702 A IL 102702A IL 10270292 A IL10270292 A IL 10270292A IL 102702 A IL102702 A IL 102702A
- Authority
- IL
- Israel
- Prior art keywords
- optically active
- preparation
- halo
- substituted
- amino acids
- Prior art date
Links
- 239000002253 acid Substances 0.000 title abstract 2
- 238000000034 method Methods 0.000 title 1
- 125000003118 aryl group Chemical group 0.000 abstract 4
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 2
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 2
- 125000002915 carbonyl group Chemical group [*:2]C([*:1])=O 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000004191 (C1-C6) alkoxy group Chemical group 0.000 abstract 1
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 abstract 1
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000001584 benzyloxycarbonyl group Chemical group C(=O)(OCC1=CC=CC=C1)* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000004122 cyclic group Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- UYWQUFXKFGHYNT-UHFFFAOYSA-N phenylmethyl ester of formic acid Natural products O=COCC1=CC=CC=C1 UYWQUFXKFGHYNT-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/30—Phosphinic acids [R2P(=O)(OH)]; Thiophosphinic acids ; [R2P(=X1)(X2H) (X1, X2 are each independently O, S or Se)]
- C07F9/301—Acyclic saturated acids which can have further substituents on alkyl
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6527—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
- C07F9/653—Five-membered rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4125753 | 1991-08-03 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL102702A0 IL102702A0 (en) | 1993-01-14 |
| IL102702A true IL102702A (en) | 1997-04-15 |
Family
ID=6437631
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL102702A IL102702A (en) | 1991-08-03 | 1992-07-31 | OPTICALLY ACTIVE g-HALO- 2-AMINOALKANECARBOXYLIC ACID DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THEIR USE FOR THE PREPARATION OF OPTICALLY ACTIVE PHOSPHORUS-CONTAINING a-AMINO ACIDS |
Country Status (9)
| Country | Link |
|---|---|
| US (2) | US5633385A (xx) |
| EP (1) | EP0530506B1 (xx) |
| JP (1) | JP3212702B2 (xx) |
| AT (1) | ATE137498T1 (xx) |
| CA (1) | CA2075151A1 (xx) |
| DE (1) | DE59206163D1 (xx) |
| HU (1) | HUT63622A (xx) |
| IL (1) | IL102702A (xx) |
| ZA (1) | ZA925776B (xx) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4407197A1 (de) * | 1994-03-04 | 1995-09-07 | Hoechst Schering Agrevo Gmbh | Verfahren zur Herstellung von /L/-Homoalanin-4-yl-(methyl)phosphinsäure und deren Salze durch Racematspaltung |
| DE19505932B4 (de) * | 1995-02-21 | 2005-06-23 | Degussa Ag | Verfahren zur Herstellung von Oxazolidinonen, neue Oxazolidinone sowie Verwendung von Oxazolidinonen |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR208400A1 (es) * | 1974-03-13 | 1976-12-27 | Yoshitomi Pharmaceutical | Un metodo para producir nuevos acidos 5-alcoxi-4-oxazolalcanoicos 2-substituidos y sus esteres |
| US4265654A (en) * | 1977-12-28 | 1981-05-05 | Meiji Seika Kaisha Ltd. | Herbicidal compositions |
| DE3817956A1 (de) * | 1988-05-27 | 1989-12-07 | Hoechst Ag | Verfahren zur herstellung phosphorhaltiger l-aminosaeuren sowie ihrer ester und n-derivate |
-
1992
- 1992-07-31 DE DE59206163T patent/DE59206163D1/de not_active Expired - Fee Related
- 1992-07-31 JP JP20574292A patent/JP3212702B2/ja not_active Expired - Fee Related
- 1992-07-31 EP EP92113099A patent/EP0530506B1/de not_active Expired - Lifetime
- 1992-07-31 ZA ZA925776A patent/ZA925776B/xx unknown
- 1992-07-31 CA CA002075151A patent/CA2075151A1/en not_active Abandoned
- 1992-07-31 HU HU9202506A patent/HUT63622A/hu unknown
- 1992-07-31 IL IL102702A patent/IL102702A/xx not_active IP Right Cessation
- 1992-07-31 AT AT92113099T patent/ATE137498T1/de not_active IP Right Cessation
-
1995
- 1995-06-05 US US08/465,433 patent/US5633385A/en not_active Expired - Fee Related
- 1995-06-06 US US08/466,877 patent/US5591861A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| ZA925776B (en) | 1993-04-28 |
| DE59206163D1 (de) | 1996-06-05 |
| US5633385A (en) | 1997-05-27 |
| EP0530506A1 (de) | 1993-03-10 |
| IL102702A0 (en) | 1993-01-14 |
| HUT63622A (en) | 1993-09-28 |
| JPH05239079A (ja) | 1993-09-17 |
| JP3212702B2 (ja) | 2001-09-25 |
| CA2075151A1 (en) | 1993-02-04 |
| EP0530506B1 (de) | 1996-05-01 |
| ATE137498T1 (de) | 1996-05-15 |
| US5591861A (en) | 1997-01-07 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| RH | Patent void | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| MM9K | Patent not in force due to non-payment of renewal fees |