IL102521A - History of Decahydro - H8 - Isoquino] g-2,1 [] 1,6 [Naphthiridine and Decahydro - 11 - Sulfonyl - Benzo] a [Pyrrole] e-2,3 [Quinolizine, their preparation and pharmaceutical preparations - Google Patents

History of Decahydro - H8 - Isoquino] g-2,1 [] 1,6 [Naphthiridine and Decahydro - 11 - Sulfonyl - Benzo] a [Pyrrole] e-2,3 [Quinolizine, their preparation and pharmaceutical preparations

Info

Publication number
IL102521A
IL102521A IL10252192A IL10252192A IL102521A IL 102521 A IL102521 A IL 102521A IL 10252192 A IL10252192 A IL 10252192A IL 10252192 A IL10252192 A IL 10252192A IL 102521 A IL102521 A IL 102521A
Authority
IL
Israel
Prior art keywords
pyrrolo
llaa
decahydro
naphthyridine
decahydrobenzo
Prior art date
Application number
IL10252192A
Other languages
English (en)
Hebrew (he)
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of IL102521A publication Critical patent/IL102521A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL10252192A 1991-07-17 1992-07-16 History of Decahydro - H8 - Isoquino] g-2,1 [] 1,6 [Naphthiridine and Decahydro - 11 - Sulfonyl - Benzo] a [Pyrrole] e-2,3 [Quinolizine, their preparation and pharmaceutical preparations IL102521A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73169191A 1991-07-17 1991-07-17

Publications (1)

Publication Number Publication Date
IL102521A true IL102521A (en) 1996-05-14

Family

ID=24940584

Family Applications (1)

Application Number Title Priority Date Filing Date
IL10252192A IL102521A (en) 1991-07-17 1992-07-16 History of Decahydro - H8 - Isoquino] g-2,1 [] 1,6 [Naphthiridine and Decahydro - 11 - Sulfonyl - Benzo] a [Pyrrole] e-2,3 [Quinolizine, their preparation and pharmaceutical preparations

Country Status (14)

Country Link
EP (1) EP0524004A1 (it)
JP (1) JPH0665242A (it)
KR (1) KR930002346A (it)
AU (1) AU655998B2 (it)
CA (1) CA2074038A1 (it)
FI (1) FI923267A (it)
HU (2) HUT61550A (it)
IE (1) IE922314A1 (it)
IL (1) IL102521A (it)
IT (1) IT1256880B (it)
NO (1) NO922812L (it)
NZ (1) NZ243586A (it)
TW (1) TW209219B (it)
ZA (1) ZA925324B (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005000846A1 (en) 2003-06-20 2005-01-06 F.Hoffmann-La Roche Ag Hexahydropyridoisoqinolines as dpp-iv inhibitors
CN103387583B (zh) * 2012-05-09 2018-04-13 中国科学院上海药物研究所 二芳基并[a,g]喹嗪类化合物、其制备方法、药物组合物及其应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4791108A (en) * 1987-04-13 1988-12-13 Syntex (U.S.A.) Inc. Sulfonyl-decahydro-8H-isoquino[2,1-G][1,6]-naphthyridines and related compounds useful as α2 -blockers

Also Published As

Publication number Publication date
IE922314A1 (en) 1993-01-27
NO922812L (no) 1993-01-18
NO922812D0 (no) 1992-07-16
HU210711A9 (en) 1995-06-28
HUT61550A (en) 1993-01-28
AU2031392A (en) 1993-01-21
NZ243586A (en) 1995-03-28
JPH0665242A (ja) 1994-03-08
FI923267A (fi) 1993-01-18
KR930002346A (ko) 1993-02-23
AU655998B2 (en) 1995-01-19
FI923267A0 (fi) 1992-07-16
ZA925324B (en) 1994-07-17
IT1256880B (it) 1995-12-27
CA2074038A1 (en) 1993-01-18
TW209219B (it) 1993-07-11
HU9202333D0 (en) 1992-10-28
ITTO920606A1 (it) 1994-01-16
EP0524004A1 (en) 1993-01-20
ITTO920606A0 (it) 1992-07-16

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Legal Events

Date Code Title Description
FF Patent granted
KB Patent renewed
RH Patent void