IE40752B1 - -aryl-4-substituted piperidinoalkanol derivatives - Google Patents
-aryl-4-substituted piperidinoalkanol derivativesInfo
- Publication number
- IE40752B1 IE40752B1 IE19/75A IE1975A IE40752B1 IE 40752 B1 IE40752 B1 IE 40752B1 IE 19/75 A IE19/75 A IE 19/75A IE 1975 A IE1975 A IE 1975A IE 40752 B1 IE40752 B1 IE 40752B1
- Authority
- IE
- Ireland
- Prior art keywords
- carbon atoms
- phenyl
- group
- substituted
- straight
- Prior art date
Links
- 125000004432 carbon atom Chemical group C* 0.000 abstract 9
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 9
- 125000003545 alkoxy group Chemical group 0.000 abstract 3
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 125000001624 naphthyl group Chemical group 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 125000003282 alkyl amino group Chemical group 0.000 abstract 1
- 239000000043 antiallergic agent Substances 0.000 abstract 1
- 239000000739 antihistaminic agent Substances 0.000 abstract 1
- 229940124630 bronchodilator Drugs 0.000 abstract 1
- 239000000168 bronchodilator agent Substances 0.000 abstract 1
- 125000000113 cyclohexyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])C1([H])[H] 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 125000002911 monocyclic heterocycle group Chemical group 0.000 abstract 1
- 230000003287 optical effect Effects 0.000 abstract 1
- -1 pyrrolidino, piperidino, morpholino Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 125000001544 thienyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
- C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
- C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/440,855 US3941795A (en) | 1974-02-08 | 1974-02-08 | α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IE40752L IE40752L (en) | 1975-08-08 |
| IE40752B1 true IE40752B1 (en) | 1979-08-15 |
Family
ID=23750454
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IE19/75A IE40752B1 (en) | 1974-02-08 | 1975-01-03 | -aryl-4-substituted piperidinoalkanol derivatives |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US3941795A (en, 2012) |
| JP (1) | JPS50108266A (en, 2012) |
| BE (1) | BE825302R (en, 2012) |
| CA (1) | CA1082703A (en, 2012) |
| CH (1) | CH609972A5 (en, 2012) |
| DE (1) | DE2503362A1 (en, 2012) |
| DK (1) | DK41775A (en, 2012) |
| FR (1) | FR2260348A2 (en, 2012) |
| GB (1) | GB1437939A (en, 2012) |
| IE (1) | IE40752B1 (en, 2012) |
| IL (1) | IL46341A (en, 2012) |
| NL (1) | NL7501463A (en, 2012) |
| NO (1) | NO750394L (en, 2012) |
| PH (1) | PH11250A (en, 2012) |
| SE (1) | SE7501196L (en, 2012) |
| ZA (1) | ZA7548B (en, 2012) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4013647A (en) * | 1976-03-23 | 1977-03-22 | American Home Products Corporation | Morpholine containing tetrazole-5-carboxamide derivatives |
| US4285958A (en) * | 1979-04-10 | 1981-08-25 | Richardson-Merrell Inc. | 1-Piperidine-alkylene ketones, pharmaceutical compositions thereof and method of use thereof |
| US4254129A (en) * | 1979-04-10 | 1981-03-03 | Richardson-Merrell Inc. | Piperidine derivatives |
| US4254130A (en) * | 1979-04-10 | 1981-03-03 | Richardson-Merrell Inc. | Piperidine derivatives |
| US4285957A (en) * | 1979-04-10 | 1981-08-25 | Richardson-Merrell Inc. | 1-Piperidine-alkanol derivatives, pharmaceutical compositions thereof, and method of use thereof |
| US4810713A (en) * | 1985-12-20 | 1989-03-07 | A. H. Robins Company, Incorporated | Arylalkyl-heterocyclic amines, n-substituted by aryloxyalkyl groups used in a method for allergy treatment |
| DE3917241A1 (de) * | 1989-05-26 | 1990-11-29 | Schaper & Bruemmer Gmbh | 4-(hydroxydiphenylmethyl)-1-piperidyl-phenylalkan-derivate |
| IE903957A1 (en) * | 1989-11-06 | 1991-05-08 | Sanofi Sa | Aromatic amine compounds, their method of preparation and¹pharmaceutical compositions in which they are present |
| US5063235A (en) * | 1990-04-30 | 1991-11-05 | A. H. Robins Company, Inc. | 4-[(diaryl)hydromethyl]-1-piperidinealkanols and esters and carbamates thereof useful in the treatment of allergic disorders |
| US5428037A (en) * | 1993-04-09 | 1995-06-27 | Syntex Pharmaceuticals, Ltd. | Heterocyclic derivatives in the treatment of Ischaemia and related diseases |
| US20020007068A1 (en) | 1999-07-16 | 2002-01-17 | D'ambra Thomas E. | Piperidine derivatives and process for their production |
| DK1369409T3 (da) * | 1993-06-24 | 2006-08-14 | Amr Technology Inc | Fremgangsmåde til fremstilling af forbindelser, der er anvendelige som mellemprodukter |
| US6147216A (en) * | 1993-06-25 | 2000-11-14 | Merrell Pharmaceuticals Inc. | Intermediates useful for the preparation of antihistaminic piperidine derivatives |
| EP2261208A1 (en) | 1993-06-25 | 2010-12-15 | Aventisub II Inc. | Intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives |
| FI973518A0 (fi) | 1995-02-28 | 1997-08-27 | Hoechst Marion Roussel Inc | Farmaseuttinen koostumus piperidinoalkanoliyhdisteille |
| US6153754A (en) * | 1995-12-21 | 2000-11-28 | Albany Molecular Research, Inc. | Process for production of piperidine derivatives |
| US6201124B1 (en) * | 1995-12-21 | 2001-03-13 | Albany Molecular Research, Inc. | Process for production of piperidine derivatives |
| US6613907B2 (en) | 2000-11-08 | 2003-09-02 | Amr Technology, Inc. | Process for the production of piperidine derivatives with microorganisms |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3839431A (en) * | 1970-07-13 | 1974-10-01 | Squibb & Sons Inc | Cyclopropylmethylphenylacetic acids and derivatives |
| BE794596A (fr) * | 1972-01-28 | 1973-05-16 | Richardson Merrell Inc | Piperidinoalcanone-oximes substituees et leur procede de preparation |
| ZA728544B (en) | 1972-01-28 | 1974-02-27 | Richardson Merrell Inc | Alpha-aryl-4-substituted piperidinoalkanol derivatives |
| US3806526A (en) * | 1972-01-28 | 1974-04-23 | Richardson Merrell Inc | 1-aroylalkyl-4-diphenylmethyl piperidines |
-
1974
- 1974-02-08 US US05/440,855 patent/US3941795A/en not_active Expired - Lifetime
- 1974-12-25 IL IL46341A patent/IL46341A/xx unknown
-
1975
- 1975-01-02 ZA ZA00750048A patent/ZA7548B/xx unknown
- 1975-01-03 IE IE19/75A patent/IE40752B1/xx unknown
- 1975-01-17 JP JP50007179A patent/JPS50108266A/ja active Pending
- 1975-01-27 GB GB339375A patent/GB1437939A/en not_active Expired
- 1975-01-28 DE DE19752503362 patent/DE2503362A1/de not_active Withdrawn
- 1975-01-31 CA CA219,191A patent/CA1082703A/en not_active Expired
- 1975-02-04 SE SE7501196A patent/SE7501196L/xx unknown
- 1975-02-04 CH CH129775A patent/CH609972A5/xx not_active IP Right Cessation
- 1975-02-06 FR FR7503733A patent/FR2260348A2/fr not_active Withdrawn
- 1975-02-06 DK DK41775*#A patent/DK41775A/da not_active Application Discontinuation
- 1975-02-07 NL NL7501463A patent/NL7501463A/xx not_active Application Discontinuation
- 1975-02-07 BE BE153164A patent/BE825302R/xx not_active IP Right Cessation
- 1975-02-07 NO NO750394A patent/NO750394L/no unknown
- 1975-02-10 PH PH16790A patent/PH11250A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PH11250A (en) | 1977-10-28 |
| CA1082703A (en) | 1980-07-29 |
| JPS50108266A (en, 2012) | 1975-08-26 |
| FR2260348A2 (en, 2012) | 1975-09-05 |
| NL7501463A (nl) | 1975-08-12 |
| IE40752L (en) | 1975-08-08 |
| AU7668874A (en) | 1976-06-24 |
| IL46341A0 (en) | 1975-03-13 |
| DE2503362A1 (de) | 1975-08-21 |
| IL46341A (en) | 1978-09-29 |
| BE825302R (fr) | 1975-05-29 |
| ZA7548B (en) | 1976-01-28 |
| DK41775A (en, 2012) | 1975-10-06 |
| GB1437939A (en) | 1976-06-03 |
| US3941795A (en) | 1976-03-02 |
| SE7501196L (en, 2012) | 1975-08-11 |
| CH609972A5 (en, 2012) | 1979-03-30 |
| NO750394L (en, 2012) | 1975-09-01 |
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