HUP0202762A3 - Solid lipid compositions, process for their preparation and use thereof - Google Patents

Solid lipid compositions, process for their preparation and use thereof

Info

Publication number
HUP0202762A3
HUP0202762A3 HU0202762A HUP0202762A HUP0202762A3 HU P0202762 A3 HUP0202762 A3 HU P0202762A3 HU 0202762 A HU0202762 A HU 0202762A HU P0202762 A HUP0202762 A HU P0202762A HU P0202762 A3 HUP0202762 A3 HU P0202762A3
Authority
HU
Hungary
Prior art keywords
preparation
solid lipid
lipid compositions
compositions
solid
Prior art date
Application number
HU0202762A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8238989&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUP0202762(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of HUP0202762A2 publication Critical patent/HUP0202762A2/hu
Publication of HUP0202762A3 publication Critical patent/HUP0202762A3/hu
Publication of HU229037B1 publication Critical patent/HU229037B1/hu

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365Lactones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007Effervescent
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Physiology (AREA)
  • Zoology (AREA)
  • Obesity (AREA)
  • Organic Chemistry (AREA)
  • Nutrition Science (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
HU0202762A 1999-09-13 2000-09-11 Solid lipid formulations comprising an inhibitor of lipases and a fatty acid ester of polyols HU229037B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP99118179 1999-09-13
PCT/EP2000/008857 WO2001019378A2 (en) 1999-09-13 2000-09-11 Solid lipid formulations comprising an inhibitor of lipases and a fatty acid ester of polyols

Publications (3)

Publication Number Publication Date
HUP0202762A2 HUP0202762A2 (hu) 2003-01-28
HUP0202762A3 true HUP0202762A3 (en) 2005-04-28
HU229037B1 HU229037B1 (en) 2013-07-29

Family

ID=8238989

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0202762A HU229037B1 (en) 1999-09-13 2000-09-11 Solid lipid formulations comprising an inhibitor of lipases and a fatty acid ester of polyols

Country Status (36)

Country Link
US (1) US6703369B1 (hu)
EP (1) EP1216048B1 (hu)
JP (1) JP4217017B2 (hu)
KR (1) KR100523879B1 (hu)
CN (1) CN1197554C (hu)
AR (1) AR025609A1 (hu)
AT (1) ATE285783T1 (hu)
AU (1) AU769016B2 (hu)
BR (1) BRPI0013940B1 (hu)
CA (1) CA2383036C (hu)
CO (1) CO5210857A1 (hu)
CZ (1) CZ301844B6 (hu)
DE (1) DE60017156T2 (hu)
EG (1) EG24225A (hu)
ES (1) ES2233444T3 (hu)
GC (1) GC0000259A (hu)
HK (1) HK1049798B (hu)
HR (1) HRP20020206B1 (hu)
HU (1) HU229037B1 (hu)
IL (2) IL148570A0 (hu)
JO (1) JO2300B1 (hu)
MA (1) MA26817A1 (hu)
ME (1) MEP90908A (hu)
MX (1) MXPA02002662A (hu)
MY (1) MY127430A (hu)
NO (1) NO328889B1 (hu)
NZ (1) NZ517396A (hu)
PE (1) PE20010661A1 (hu)
PL (1) PL199869B1 (hu)
PT (1) PT1216048E (hu)
RS (1) RS50373B (hu)
RU (1) RU2248218C2 (hu)
SI (1) SI1216048T1 (hu)
TR (1) TR200200605T2 (hu)
WO (1) WO2001019378A2 (hu)
ZA (1) ZA200201249B (hu)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR025609A1 (es) * 1999-09-13 2002-12-04 Hoffmann La Roche Formulaciones lipidas solidas
HRP20030029B1 (en) * 2000-07-28 2005-06-30 F. Hoffmann - La Roche Ag New pharmaceutical composition
US6730319B2 (en) 2001-06-06 2004-05-04 Hoffmann-La Roche Inc. Pharmaceutical compositions having depressed melting points
US20030027786A1 (en) * 2001-06-06 2003-02-06 Karsten Maeder Lipase inhibiting composition
DE10251963A1 (de) * 2002-11-08 2004-05-19 Lts Lohmann Therapie-Systeme Ag Transmucosale pharmazeutische Darreichungsform
US8372430B2 (en) * 2002-12-17 2013-02-12 The Procter & Gamble Company Compositions, methods, and kits useful for the alleviation of gastrointestinal effects
JP2006514672A (ja) * 2003-03-04 2006-05-11 ノストラム・ファーマスーティカルズ・インコーポレイテッド 疎水性物質を徐放剤として含有する制御性放出製剤
FI20045076L (fi) * 2004-03-15 2005-09-16 Bioferme Oy Funktionaalinen elintarvike
MX2007004973A (es) * 2004-10-25 2007-06-14 Japan Tobacco Inc Formulacion solida con solubilidad y estabilidad mejoradas y metodo para producir la formulacion.
KR100669497B1 (ko) * 2005-08-17 2007-01-16 보람제약주식회사 안정성과 용출률이 뛰어난 약리학적 조성물 및 그 제조방법
CN101340896A (zh) * 2005-12-22 2009-01-07 特瓦制药工业有限公司 含有低溶解性药物的压缩的固体剂型和其制备方法
US20070148245A1 (en) * 2005-12-22 2007-06-28 Ilan Zalit Compressed solid dosage forms with drugs of low solubility and process for making the same
EP1808163A1 (en) * 2005-12-22 2007-07-18 Teva Pharmaceutical Industries Ltd. Compressed solid dosage forms with drugs of low solubility and process for making the same
KR101252635B1 (ko) 2006-04-20 2013-04-10 (주)아모레퍼시픽 리파아제 저해제 및 친유성 오일흡수제를 포함하는 약학조성물 및 이로부터 제조된 경구 투여용 제제
KR100903504B1 (ko) * 2007-05-18 2009-06-17 강태용 비라칸사스 열매 추출물질을 포함하는 기능식품 및 체중 감소제
JP2010536798A (ja) * 2007-08-17 2010-12-02 テバ ファーマシューティカル インダストリーズ リミティド 難溶性薬物の生体利用率を制御するための方法及び組成物
ES2350798T3 (es) * 2007-09-12 2011-01-27 Mader S.R.L. Composiciones farmacéuticas para uso oral para tratar a pacientes afectados por la obesidad.
PL216542B1 (pl) 2008-03-20 2014-04-30 Zakłady Farmaceutyczne POLPHARMA Spółka Akcyjna Sposób wytwarzania stabilnej kompozycji orlistatu w postaci kapsułkowanego proszku
WO2010042499A1 (en) * 2008-10-06 2010-04-15 Banner Pharmacaps, Inc. Stable solutions of orlistat for pharmaceutical dosage forms
BRPI0901602B8 (pt) 2009-04-03 2021-05-25 Ems S/A formulação farmacêuticas
UA107369C2 (en) 2010-02-01 2014-12-25 Lab Bago S A Pharmaceutical composition with anti-obesity activity comprising a premixture of pure orlistat and preparation process
EP2486805A1 (en) * 2011-02-11 2012-08-15 Puratos N.V. An emulsion whippable at room-temperature
WO2012140937A1 (ja) * 2011-04-14 2012-10-18 株式会社J-オイルミルズ パーム系分別油脂、それを配合した油脂組成物及び食品
CN102552168B (zh) * 2012-01-31 2013-08-07 杭州华东医药集团生物工程研究所有限公司 一种含有奥利司他的药物组合物及其制备方法
GB2501535A (en) 2012-04-26 2013-10-30 Sony Corp Chrominance Processing in High Efficiency Video Codecs
EP2854763B1 (en) * 2012-05-31 2018-09-26 Repros Therapeutics Inc. Formulations for vaginal delivery of antiprogestins
US9980934B2 (en) 2013-10-28 2018-05-29 Nestec S.A. Monoacylglycerols for use in conjunction with a lipase inhibitor and/or diets low in fat and/or calories
CN115105476B (zh) * 2021-03-23 2023-11-14 山东新时代药业有限公司 一种奥利司他冻干口服制剂及其制备工艺

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1247547A (en) * 1983-06-22 1988-12-28 Paul Hadvary Leucine derivatives
FR2710264B1 (fr) * 1993-09-21 1995-12-08 Rocher Yves Biolog Vegetale Utilisation pour le traitement des peaux mixtes d'une quantité efficace de substances actives.
AU5185398A (en) * 1996-12-04 1998-06-29 James S Pincott Process and apparatus for making crumb rubber from scrap tyres
TR199901853T2 (xx) 1997-02-05 1999-12-21 F. Hoffmann-La Roche Ag. Gastrointestinal lipaz inhibit�r�n�n kullan�lmas�.
US6004996A (en) * 1997-02-05 1999-12-21 Hoffman-La Roche Inc. Tetrahydrolipstatin containing compositions
US6267952B1 (en) 1998-01-09 2001-07-31 Geltex Pharmaceuticals, Inc. Lipase inhibiting polymers
EP1105123B1 (en) * 1998-08-14 2004-04-07 F.Hoffmann-La Roche Ag Pharmaceutical compositions containing lipase inhibitors and chitosan
PT1105122E (pt) 1998-08-14 2005-08-31 Hoffmann La Roche Composicoes farmaceuticas que contem inibidores de lipase
AR025609A1 (es) * 1999-09-13 2002-12-04 Hoffmann La Roche Formulaciones lipidas solidas

Also Published As

Publication number Publication date
DE60017156T2 (de) 2006-01-05
ES2233444T3 (es) 2005-06-16
AU7517700A (en) 2001-04-17
MXPA02002662A (es) 2002-07-30
PT1216048E (pt) 2005-04-29
HUP0202762A2 (hu) 2003-01-28
ZA200201249B (en) 2003-07-30
NO20021205L (no) 2002-03-12
EG24225A (en) 2008-11-10
WO2001019378A2 (en) 2001-03-22
YU13602A (sh) 2006-01-16
RU2248218C2 (ru) 2005-03-20
CZ301844B6 (cs) 2010-07-07
AR025609A1 (es) 2002-12-04
ATE285783T1 (de) 2005-01-15
HK1049798A1 (en) 2003-05-30
CA2383036C (en) 2006-01-10
HRP20020206A2 (en) 2004-04-30
PL356154A1 (en) 2004-06-14
NZ517396A (en) 2003-10-31
KR100523879B1 (ko) 2005-10-26
ME00675B (me) 2011-12-20
NO20021205D0 (no) 2002-03-12
MY127430A (en) 2006-11-30
TR200200605T2 (tr) 2002-08-21
RS50373B (sr) 2009-11-10
HK1049798B (zh) 2005-08-05
HU229037B1 (en) 2013-07-29
KR20020060177A (ko) 2002-07-16
JP4217017B2 (ja) 2009-01-28
CZ20021277A3 (cs) 2003-04-16
CN1373659A (zh) 2002-10-09
GC0000259A (en) 2006-11-01
US6703369B1 (en) 2004-03-09
JO2300B1 (en) 2005-09-12
BR0013940A (pt) 2002-05-14
CA2383036A1 (en) 2001-03-22
IL148570A0 (en) 2002-09-12
PE20010661A1 (es) 2001-06-25
PL199869B1 (pl) 2008-11-28
RU2002107450A (ru) 2004-01-10
CO5210857A1 (es) 2002-10-30
CN1197554C (zh) 2005-04-20
IL148570A (en) 2007-03-08
MA26817A1 (fr) 2004-12-20
MEP90908A (en) 2011-12-20
DE60017156D1 (de) 2005-02-03
JP2003509373A (ja) 2003-03-11
AU769016B2 (en) 2004-01-15
WO2001019378A3 (en) 2001-05-10
EP1216048A2 (en) 2002-06-26
SI1216048T1 (en) 2005-06-30
EP1216048B1 (en) 2004-12-29
HRP20020206B1 (en) 2011-02-28
BRPI0013940B1 (pt) 2016-06-21
NO328889B1 (no) 2010-06-07

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Legal Events

Date Code Title Description
GB9A Succession in title

Owner name: CHEPLAPHARM ARZNEIMITTEL GMBH, DE

Free format text: FORMER OWNER(S): F. HOFFMANN-LA ROCHE AG, CH