HUP0100558A3 - S-oxide and s,s,-dioxide tetrahydrothiopyran phenyloxazolidinones, their use for preparation of pharmaceutical compositions and process for determining the inhibitory activity of compounds to human monoamino oxidase - Google Patents
S-oxide and s,s,-dioxide tetrahydrothiopyran phenyloxazolidinones, their use for preparation of pharmaceutical compositions and process for determining the inhibitory activity of compounds to human monoamino oxidaseInfo
- Publication number
- HUP0100558A3 HUP0100558A3 HU0100558A HUP0100558A HUP0100558A3 HU P0100558 A3 HUP0100558 A3 HU P0100558A3 HU 0100558 A HU0100558 A HU 0100558A HU P0100558 A HUP0100558 A HU P0100558A HU P0100558 A3 HUP0100558 A3 HU P0100558A3
- Authority
- HU
- Hungary
- Prior art keywords
- phenyloxazolidinones
- compounds
- human
- oxide
- preparation
- Prior art date
Links
- DRQFDIUXANJKDA-UHFFFAOYSA-N 3-phenyl-1,3-oxazolidin-2-one;thiane Chemical class C1CCSCC1.O=C1OCCN1C1=CC=CC=C1 DRQFDIUXANJKDA-UHFFFAOYSA-N 0.000 title 1
- 102000004316 Oxidoreductases Human genes 0.000 title 1
- 108090000854 Oxidoreductases Proteins 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- RCCPEORTSYDPMB-UHFFFAOYSA-N hydroxy benzenecarboximidothioate Chemical compound OSC(=N)C1=CC=CC=C1 RCCPEORTSYDPMB-UHFFFAOYSA-N 0.000 title 1
- 230000002401 inhibitory effect Effects 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Catalysts (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6783097P | 1997-12-05 | 1997-12-05 | |
| US8949898P | 1998-06-16 | 1998-06-16 | |
| US10018598P | 1998-09-14 | 1998-09-14 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HUP0100558A2 HUP0100558A2 (hu) | 2002-05-29 |
| HUP0100558A3 true HUP0100558A3 (en) | 2002-08-28 |
Family
ID=27371238
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0100558A HUP0100558A3 (en) | 1997-12-05 | 1998-11-23 | S-oxide and s,s,-dioxide tetrahydrothiopyran phenyloxazolidinones, their use for preparation of pharmaceutical compositions and process for determining the inhibitory activity of compounds to human monoamino oxidase |
Country Status (22)
| Country | Link |
|---|---|
| US (2) | US6083967A (hu) |
| EP (2) | EP1036074B1 (hu) |
| JP (1) | JP2001525408A (hu) |
| KR (1) | KR20010032782A (hu) |
| CN (2) | CN1532535A (hu) |
| AT (1) | ATE231859T1 (hu) |
| AU (2) | AU752454B2 (hu) |
| BR (1) | BR9814897A (hu) |
| CA (1) | CA2309026A1 (hu) |
| DE (1) | DE69811117T2 (hu) |
| DK (1) | DK1036074T3 (hu) |
| ES (1) | ES2191985T3 (hu) |
| HK (1) | HK1032970A1 (hu) |
| HU (1) | HUP0100558A3 (hu) |
| ID (1) | ID21450A (hu) |
| NO (1) | NO316447B1 (hu) |
| NZ (1) | NZ504930A (hu) |
| PL (1) | PL340835A1 (hu) |
| SI (1) | SI1036074T1 (hu) |
| SK (1) | SK7692000A3 (hu) |
| TW (2) | TW553942B (hu) |
| WO (1) | WO1999029688A1 (hu) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6511468B1 (en) | 1997-10-17 | 2003-01-28 | Micro Therapeutics, Inc. | Device and method for controlling injection of liquid embolic composition |
| TR200003595T2 (tr) | 1998-06-05 | 2001-07-23 | Astrazeneca Ab | Kimyasal bileşikler |
| MY120189A (en) | 1999-11-04 | 2005-09-30 | Upjohn Co | Sultam and sultone derived oxazolidinones |
| DE19962924A1 (de) | 1999-12-24 | 2001-07-05 | Bayer Ag | Substituierte Oxazolidinone und ihre Verwendung |
| DE10129725A1 (de) | 2001-06-20 | 2003-01-02 | Bayer Ag | Kombinationstherapie substituierter Oxazolidinone |
| US7141588B2 (en) | 2002-02-25 | 2006-11-28 | Pfizer, Inc. | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
| AR038536A1 (es) | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
| EP1539745B1 (en) | 2002-08-12 | 2006-03-29 | Pharmacia & Upjohn Company LLC | N-aryl-2-oxazolidinones and their derivatives |
| BR0316483A (pt) | 2002-11-21 | 2005-10-11 | Upjohn Co | Derivados de n-(4-(piperazin-1-il)-fenil-2-oxazolidinona-5-carboxami da e compostos relacionados como agentes antibacterianos |
| DE10300111A1 (de) * | 2003-01-07 | 2004-07-15 | Bayer Healthcare Ag | Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid |
| US7304050B2 (en) | 2003-09-16 | 2007-12-04 | Pfizer Inc. | Antibacterial agents |
| DE10355461A1 (de) | 2003-11-27 | 2005-06-23 | Bayer Healthcare Ag | Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung |
| DE102004062475A1 (de) * | 2004-12-24 | 2006-07-06 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung |
| EP1685841A1 (en) | 2005-01-31 | 2006-08-02 | Bayer Health Care Aktiengesellschaft | Prevention and treatment of thromboembolic disorders |
| DE102005045518A1 (de) | 2005-09-23 | 2007-03-29 | Bayer Healthcare Ag | 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung |
| SG166126A1 (en) | 2005-10-04 | 2010-11-29 | Bayer Schering Pharma Ag | Novel polymorphous form and the amorphous form of 5-chloro-n-({(5s)-2-oxo- 3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidine-5-yl}-methyl)-2-thiophene carboxamide |
| DE102005047558A1 (de) * | 2005-10-04 | 2008-02-07 | Bayer Healthcare Ag | Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen |
| DE102005047561A1 (de) | 2005-10-04 | 2007-04-05 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung |
| CN102262066A (zh) * | 2011-06-16 | 2011-11-30 | 董理 | 一种检测单胺氧化酶含量的方法和试剂盒 |
| CN104610479B (zh) * | 2013-11-05 | 2017-03-29 | 中国石油化工股份有限公司 | 用于乙烯聚合的负载化茂金属催化剂及其制备方法和应用 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1302422C (en) * | 1986-09-03 | 1992-06-02 | Margherita Strolin-Benedetti | 5-aminoethyloxazolidin-2-one derivatives, process for the preparation thereofand their therapeutic use |
| US4885154A (en) * | 1988-03-01 | 1989-12-05 | Alza Corporation | Method for reducing sensitization or irritation in transdermal drug delivery and means therefor |
| US5254577A (en) * | 1988-07-29 | 1993-10-19 | The Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
| US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
| US5130316A (en) * | 1988-07-29 | 1992-07-14 | Du Pont Merck Pharmaceutical Company | Aminomethyloxooxazlidinyl arylbenzene derivatives useful as antibacterial agents |
| JP2669579B2 (ja) * | 1991-10-23 | 1997-10-29 | エーザイ株式会社 | オキサゾリドン誘導体 |
| CA2119556C (en) * | 1991-11-01 | 2004-07-06 | Michael Robert Barbachyn | Substituted aryl- and heteroaryl-phenyloxazolidinones |
| ATE161833T1 (de) * | 1992-12-08 | 1998-01-15 | Upjohn Co | Durch eine tropon gruppe substituierte phenyloxazolidinone-derivate als antibakterielles mittel |
| RU2175324C2 (ru) * | 1995-09-01 | 2001-10-27 | Фармация Энд Апджон Компани | Фенилоксазолидиноны, имеющие с-с-связь с 4-8-членными гетероциклическими кольцами |
| GB9702213D0 (en) * | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
-
1998
- 1998-11-20 US US09/196,890 patent/US6083967A/en not_active Expired - Fee Related
- 1998-11-23 DE DE69811117T patent/DE69811117T2/de not_active Expired - Fee Related
- 1998-11-23 JP JP2000524282A patent/JP2001525408A/ja active Pending
- 1998-11-23 EP EP98962811A patent/EP1036074B1/en not_active Expired - Lifetime
- 1998-11-23 BR BR9814897-4A patent/BR9814897A/pt not_active Application Discontinuation
- 1998-11-23 KR KR1020007006081A patent/KR20010032782A/ko not_active Application Discontinuation
- 1998-11-23 HU HU0100558A patent/HUP0100558A3/hu unknown
- 1998-11-23 CA CA002309026A patent/CA2309026A1/en not_active Abandoned
- 1998-11-23 WO PCT/US1998/024526 patent/WO1999029688A1/en active Search and Examination
- 1998-11-23 NZ NZ504930A patent/NZ504930A/en unknown
- 1998-11-23 AU AU17968/99A patent/AU752454B2/en not_active Ceased
- 1998-11-23 AT AT98962811T patent/ATE231859T1/de not_active IP Right Cessation
- 1998-11-23 EP EP02015566A patent/EP1254906A1/en not_active Withdrawn
- 1998-11-23 SK SK769-2000A patent/SK7692000A3/sk unknown
- 1998-11-23 SI SI9830371T patent/SI1036074T1/xx unknown
- 1998-11-23 DK DK98962811T patent/DK1036074T3/da active
- 1998-11-23 CN CNA2004100328277A patent/CN1532535A/zh active Pending
- 1998-11-23 ES ES98962811T patent/ES2191985T3/es not_active Expired - Lifetime
- 1998-11-23 PL PL98340835A patent/PL340835A1/xx unknown
- 1998-11-23 CN CNB988110695A patent/CN1154645C/zh not_active Expired - Fee Related
- 1998-11-26 ID IDP981545A patent/ID21450A/id unknown
- 1998-12-04 TW TW087120185A patent/TW553942B/zh not_active IP Right Cessation
- 1998-12-04 TW TW092121194A patent/TWI239331B/zh not_active IP Right Cessation
-
1999
- 1999-11-05 US US09/434,911 patent/US6265178B1/en not_active Expired - Fee Related
-
2000
- 2000-06-02 NO NO20002834A patent/NO316447B1/no unknown
-
2001
- 2001-05-24 HK HK01103598A patent/HK1032970A1/xx not_active IP Right Cessation
-
2002
- 2002-09-16 AU AU2002301031A patent/AU2002301031B2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| TW200307673A (en) | 2003-12-16 |
| BR9814897A (pt) | 2000-10-03 |
| CN1154645C (zh) | 2004-06-23 |
| EP1036074A1 (en) | 2000-09-20 |
| NO20002834L (no) | 2000-07-21 |
| HUP0100558A2 (hu) | 2002-05-29 |
| EP1254906A1 (en) | 2002-11-06 |
| PL340835A1 (en) | 2001-02-26 |
| CN1532535A (zh) | 2004-09-29 |
| TWI239331B (en) | 2005-09-11 |
| ES2191985T3 (es) | 2003-09-16 |
| AU1796899A (en) | 1999-06-28 |
| SI1036074T1 (en) | 2003-08-31 |
| NO20002834D0 (no) | 2000-06-02 |
| NO316447B1 (no) | 2004-01-26 |
| EP1036074B1 (en) | 2003-01-29 |
| DE69811117D1 (de) | 2003-03-06 |
| CN1278817A (zh) | 2001-01-03 |
| SK7692000A3 (en) | 2001-03-12 |
| ID21450A (id) | 1999-06-10 |
| ATE231859T1 (de) | 2003-02-15 |
| WO1999029688A1 (en) | 1999-06-17 |
| JP2001525408A (ja) | 2001-12-11 |
| TW553942B (en) | 2003-09-21 |
| AU2002301031B2 (en) | 2005-08-25 |
| NZ504930A (en) | 2002-05-31 |
| HK1032970A1 (en) | 2001-08-10 |
| KR20010032782A (ko) | 2001-04-25 |
| DE69811117T2 (de) | 2003-07-17 |
| DK1036074T3 (da) | 2003-06-23 |
| US6083967A (en) | 2000-07-04 |
| US6265178B1 (en) | 2001-07-24 |
| AU752454B2 (en) | 2002-09-19 |
| CA2309026A1 (en) | 1999-06-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD9A | Lapse of provisional protection due to non-payment of fees |