HRP20201832T1 - Sustavi aditiva za upotrebu u pegilaciji proteina - Google Patents

Sustavi aditiva za upotrebu u pegilaciji proteina Download PDF

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Publication number
HRP20201832T1
HRP20201832T1 HRP20201832TT HRP20201832T HRP20201832T1 HR P20201832 T1 HRP20201832 T1 HR P20201832T1 HR P20201832T T HRP20201832T T HR P20201832TT HR P20201832 T HRP20201832 T HR P20201832T HR P20201832 T1 HRP20201832 T1 HR P20201832T1
Authority
HR
Croatia
Prior art keywords
protein
peg
aminobenzoic acid
acid hydrazide
additive system
Prior art date
Application number
HRP20201832TT
Other languages
English (en)
Croatian (hr)
Inventor
Matthew R. Hickey
Antonio Ramirez
Original Assignee
Bristol-Myers Squibb Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol-Myers Squibb Company filed Critical Bristol-Myers Squibb Company
Publication of HRP20201832T1 publication Critical patent/HRP20201832T1/hr

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/59Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
    • A61K47/60Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C07K1/1072General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups
    • C07K1/1077General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups by covalent attachment of residues other than amino acids or peptide residues, e.g. sugars, polyols, fatty acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/475Growth factors; Growth regulators
    • C07K14/50Fibroblast growth factor [FGF]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/64Relaxins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Toxicology (AREA)
  • Epidemiology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Analytical Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
HRP20201832TT 2015-11-23 2016-11-22 Sustavi aditiva za upotrebu u pegilaciji proteina HRP20201832T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562258644P 2015-11-23 2015-11-23
PCT/US2016/063313 WO2017091568A1 (en) 2015-11-23 2016-11-22 Additive systems for use in protein pegylation
EP16816042.2A EP3380487B1 (en) 2015-11-23 2016-11-22 Additive systems for use in protein pegylation

Publications (1)

Publication Number Publication Date
HRP20201832T1 true HRP20201832T1 (hr) 2021-01-08

Family

ID=57589163

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20201832TT HRP20201832T1 (hr) 2015-11-23 2016-11-22 Sustavi aditiva za upotrebu u pegilaciji proteina

Country Status (17)

Country Link
US (3) US10617765B2 (https=)
EP (2) EP3789395B1 (https=)
JP (2) JP6921821B2 (https=)
KR (1) KR102688003B1 (https=)
CN (2) CN115819494A (https=)
CY (1) CY1123699T1 (https=)
DK (1) DK3380487T3 (https=)
ES (2) ES3055983T3 (https=)
HR (1) HRP20201832T1 (https=)
HU (1) HUE052634T2 (https=)
LT (1) LT3380487T (https=)
PL (1) PL3380487T3 (https=)
PT (1) PT3380487T (https=)
RS (1) RS61072B1 (https=)
SI (1) SI3380487T1 (https=)
SM (1) SMT202000649T1 (https=)
WO (1) WO2017091568A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT3380487T (pt) * 2015-11-23 2020-10-29 Bristol Myers Squibb Co Sistemas de aditivos para utilização na peguilação de proteínas
HRP20240016T1 (hr) * 2018-09-11 2024-03-29 Ambrx, Inc. Konjugati polipeptida interleukina-2 i njihove uporabe
CN111484551B (zh) * 2020-03-19 2022-02-11 北京翼方生物科技有限责任公司 一种聚乙二醇修饰的重组人碱性成纤维细胞生长因子

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19535571A1 (de) 1995-09-14 1997-03-20 Boehringer Mannheim Gmbh Pharmazeutische Kombinationspräparate und deren Verwendung zur Behandlung von Hämodialysepatienten
TW518219B (en) 1996-04-26 2003-01-21 Chugai Pharmaceutical Co Ltd Erythropoietin solution preparation
EP0885613A1 (de) 1997-06-21 1998-12-23 Roche Diagnostics GmbH Verwendung von modifizierten Hämoglobinen zur Behandlung von Anämien und Kombinationspräparate umfassend Erythropoietin und modifiziertes Hämoglobin
DE19734293A1 (de) 1997-08-08 1999-02-11 Boehringer Mannheim Gmbh Verwendung von pharmazeutischen Kombinationspräparaten enthaltend Erythropoietin und Eisenpräparate zur Behandlung von rheumatischen Erkrankungen
US7329516B2 (en) * 2004-03-17 2008-02-12 Anticancer, Inc. Methods for increasing protein polyethylene glycol (PEG) conjugation
US20060286657A1 (en) * 2005-06-01 2006-12-21 Samuel Zalipsky Novel bioconjugation reactions for acylating polyethylene glycol reagents
CN104710503B (zh) * 2005-11-08 2023-04-25 Ambrx 公司 用于修饰非天然氨基酸和非天然氨基酸多肽的促进剂
CA2682147C (en) * 2007-03-30 2017-08-08 Ambrx, Inc. Modified fgf-21 polypeptides and their uses
AU2014212308B2 (en) 2013-01-30 2018-08-09 Avelas Biosciences, Inc. Selective delivery molecules and methods of use
WO2014176284A1 (en) 2013-04-22 2014-10-30 Avelas Biosciences, Inc. Selective drug delivery compositions and methods of use
SMT202100388T1 (it) 2014-10-24 2021-09-14 Bristol Myers Squibb Co Polipeptidi fgf-21 modificati e loro usi
PT3380487T (pt) * 2015-11-23 2020-10-29 Bristol Myers Squibb Co Sistemas de aditivos para utilização na peguilação de proteínas

Also Published As

Publication number Publication date
ES2827776T3 (es) 2021-05-24
EP3789395A1 (en) 2021-03-10
JP7257457B2 (ja) 2023-04-13
RS61072B1 (sr) 2020-12-31
PT3380487T (pt) 2020-10-29
US11213589B2 (en) 2022-01-04
SI3380487T1 (sl) 2020-11-30
LT3380487T (lt) 2020-12-28
WO2017091568A1 (en) 2017-06-01
US20190351065A1 (en) 2019-11-21
CN108350025B (zh) 2023-02-21
US20220160883A1 (en) 2022-05-26
ES3055983T3 (en) 2026-02-17
WO2017091568A8 (en) 2018-01-04
EP3380487A1 (en) 2018-10-03
JP2019503994A (ja) 2019-02-14
PL3380487T3 (pl) 2020-12-28
HUE052634T2 (hu) 2021-05-28
EP3380487B1 (en) 2020-09-02
US20200276319A1 (en) 2020-09-03
CY1123699T1 (el) 2022-03-24
JP6921821B2 (ja) 2021-08-18
CN115819494A (zh) 2023-03-21
EP3789395B1 (en) 2025-08-27
US10617765B2 (en) 2020-04-14
JP2021176890A (ja) 2021-11-11
KR20180081610A (ko) 2018-07-16
SMT202000649T1 (it) 2021-01-05
CN108350025A (zh) 2018-07-31
KR102688003B1 (ko) 2024-07-23
DK3380487T3 (da) 2020-12-07

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