HRP20171678T1 - Postupci za smanjenje prejedanja ili kompulzivnog jedenja - Google Patents
Postupci za smanjenje prejedanja ili kompulzivnog jedenja Download PDFInfo
- Publication number
- HRP20171678T1 HRP20171678T1 HRP20171678TT HRP20171678T HRP20171678T1 HR P20171678 T1 HRP20171678 T1 HR P20171678T1 HR P20171678T T HRP20171678T T HR P20171678TT HR P20171678 T HRP20171678 T HR P20171678T HR P20171678 T1 HRP20171678 T1 HR P20171678T1
- Authority
- HR
- Croatia
- Prior art keywords
- use according
- pharmaceutical preparation
- patient
- eating
- treatment
- Prior art date
Links
- 208000010235 Food Addiction Diseases 0.000 title claims 8
- 208000014679 binge eating disease Diseases 0.000 title claims 8
- 206010004716 Binge eating Diseases 0.000 title claims 6
- 208000032841 Bulimia Diseases 0.000 title claims 6
- 239000000825 pharmaceutical preparation Substances 0.000 claims 14
- 206010020710 Hyperphagia Diseases 0.000 claims 4
- 235000020830 overeating Nutrition 0.000 claims 4
- 150000003839 salts Chemical class 0.000 claims 4
- SNPPWIUOZRMYNY-UHFFFAOYSA-N bupropion Chemical compound CC(C)(C)NC(C)C(=O)C1=CC=CC(Cl)=C1 SNPPWIUOZRMYNY-UHFFFAOYSA-N 0.000 claims 3
- 229960001058 bupropion Drugs 0.000 claims 3
- DQCKKXVULJGBQN-XFWGSAIBSA-N naltrexone Chemical compound N1([C@@H]2CC3=CC=C(C=4O[C@@H]5[C@](C3=4)([C@]2(CCC5=O)O)CC1)O)CC1CC1 DQCKKXVULJGBQN-XFWGSAIBSA-N 0.000 claims 3
- 229960003086 naltrexone Drugs 0.000 claims 3
- 208000024891 symptom Diseases 0.000 claims 3
- 230000007423 decrease Effects 0.000 claims 2
- 235000014632 disordered eating Nutrition 0.000 claims 2
- 238000013265 extended release Methods 0.000 claims 2
- 208000024714 major depressive disease Diseases 0.000 claims 2
- 208000020925 Bipolar disease Diseases 0.000 claims 1
- 239000008194 pharmaceutical composition Substances 0.000 claims 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0002—Galenical forms characterised by the drug release technique; Application systems commanded by energy
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Emergency Medicine (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Hematology (AREA)
- Psychiatry (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Child & Adolescent Psychology (AREA)
- Addiction (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicinal Preparation (AREA)
- Medicines Containing Plant Substances (AREA)
Claims (15)
1. Farmaceutski pripravak koji sadrži bupropion ili njegovu farmaceutski prihvatljivu sol, i naltrekson ili njegovu farmaceutski prihvatljivu sol naznačen time da je za uporabu za liječenje prejedanja ili kompulzivnog jedenja.
2. Farmaceutski pripravak za uporabu prema zahtjevu 1, naznačen time da dodatno sadrži: upućivanje pacijenta za dnevno davanje terapijski učinkovite količine.
3. Farmaceutski pripravak za uporabu prema bilo kojem od zahtjeva 1-2, naznačen time da je indeks tjelesne mase pacijenta veći od ili jednak 25 kg/m2.
4. Farmaceutski pripravak za uporabu prema bilo kojem od zahtjeva 1-3, naznačen time da pacijent ne pati od velikog depresivnog poremećaja.
5. Farmaceutski pripravak za uporabu prema bilo kojem od zahtjeva 1-4, naznačen time da dodatno sadrži utvrđivanje da li pacijent pati od velikog depresivnog poremećaja.
6. Farmaceutski pripravak za uporabu prema zahtjevu 5, naznačen time da pacijent ne pati od bipolarnog poremećaja.
7. Farmaceutski pripravak za uporabu prema bilo kojem od zahtjeva 1-6, naznačen time da je terapijski učinkovita količina naltreksona ili njegove farmaceutski prihvatljive soli 4 mg do 50 mg dnevno i terapijski učinkovita količina bupropiona ili njegove farmaceutski prihvatljive soli je 30 mg do 500 mg dnevno.
8. Farmaceutski pripravak za uporabu prema bilo kojem od zahtjeva 1-7, naznačen time da pacijent je žena.
9. Farmaceutski pripravak za uporabu prema bilo kojem od zahtjeva 1-8, naznačen time da se simptom ili mjera poremećaja prejedanja ili poremećaja kompulzivnog jedenja smanjuje za barem 5%.
10. Farmaceutski pripravak za uporabu prema zahtjevu 9, naznačen time da se smanjuje simptom ili mjera snage događaja prejedanja ili kompulzivnog jedenja.
11. Farmaceutski pripravak za uporabu prema zahtjevu 9, naznačen time da se smanjuje simptom ili mjera frekvencije događaja prejedanja ili kompulzivnog jedenja.
12. Farmaceutski pripravak za uporabu prema bilo kojem od zahtjeva 1-11, naznačen time da se prejedanje ili kompulzivno jedenje kod pacijenta mjeri korištenjem skale prejedanja prije početka tretmana, te barem jednom nakon početka tretmana.
13. Farmaceutski pripravak za uporabu prema zahtjevu 12, naznačen time da se vrijednost skale prejedanja prije početka tretmana smanjuje za barem 10 nakon tretmana ili se smanjuje na manje od 17 nakon tretmana.
14. Farmaceutski pripravak za uporabu prema bilo kojem od zahtjeva 1-13, naznačen time da pacijent je identificiran kao pacijent koji pati od ili ima rizik od poremećaja prejedanja ili poremećaja kompulzivnog jedenja pomoću primjene kontrolnog popisa skale prejedanja.
15. Farmaceutski pripravak za uporabu prema bilo kojem od zahtjeva 1 do 14 naznačen time da dodatno sadrži:
identificiranje pacijenta koji pati od ili ima rizik od prejedanja ili kompulzivnog jedenja pomoću primjene kontrolnog popisa skale prejedanja, te pacijent ima indeks tjelesne mase (BMI) veći od ili jednak 27 kg/m2; i
davanje pacijentu 16 mg naltreksona s produženim otpuštanjem i 180 mg bupropiona s produženim otpuštanjem dva puta dnevno kroz period tretmana od više od 4 tjedna.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US41935410P | 2010-12-03 | 2010-12-03 | |
PCT/US2011/063170 WO2012075453A1 (en) | 2010-12-03 | 2011-12-02 | Methods for reducing binge or compulsive eating |
EP11844637.6A EP2646011B1 (en) | 2010-12-03 | 2011-12-02 | Methods for reducing binge or compulsive eating |
Publications (1)
Publication Number | Publication Date |
---|---|
HRP20171678T1 true HRP20171678T1 (hr) | 2017-12-15 |
Family
ID=46172302
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HRP20171678TT HRP20171678T1 (hr) | 2010-12-03 | 2017-11-02 | Postupci za smanjenje prejedanja ili kompulzivnog jedenja |
Country Status (26)
Country | Link |
---|---|
US (2) | US20130252995A1 (hr) |
EP (1) | EP2646011B1 (hr) |
JP (1) | JP2014508717A (hr) |
KR (1) | KR20140035319A (hr) |
CN (1) | CN103298462A (hr) |
AR (2) | AR084093A1 (hr) |
AU (3) | AU2011336298B2 (hr) |
BR (1) | BR112013015957B1 (hr) |
CA (1) | CA2819003A1 (hr) |
CL (1) | CL2013001565A1 (hr) |
CY (1) | CY1119560T1 (hr) |
DK (1) | DK2646011T3 (hr) |
ES (1) | ES2647232T3 (hr) |
HR (1) | HRP20171678T1 (hr) |
HU (1) | HUE034641T2 (hr) |
IL (1) | IL226483A0 (hr) |
LT (1) | LT2646011T (hr) |
MX (1) | MX350304B (hr) |
NO (1) | NO2646011T3 (hr) |
PL (1) | PL2646011T3 (hr) |
PT (1) | PT2646011T (hr) |
RS (1) | RS56548B1 (hr) |
RU (1) | RU2620913C2 (hr) |
SI (1) | SI2646011T1 (hr) |
TW (2) | TWI536986B (hr) |
WO (1) | WO2012075453A1 (hr) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2316456B1 (en) | 2003-04-29 | 2017-06-14 | Orexigen Therapeutics, Inc. | Compositions for affecting weight loss comprising an opioid antagonist and bupropion |
EP1951212A2 (en) | 2005-11-22 | 2008-08-06 | Orexigen Therapeutics, Inc. | Compositions and methods for increasing insulin sensitivity |
US8916195B2 (en) | 2006-06-05 | 2014-12-23 | Orexigen Therapeutics, Inc. | Sustained release formulation of naltrexone |
KR20090090316A (ko) | 2006-11-09 | 2009-08-25 | 오렉시젠 세러퓨틱스 인크. | 체중 감량 약물을 투여하기 위한 단위 용량 팩키지 및 투여 방법 |
CA2725930A1 (en) | 2008-05-30 | 2009-12-30 | Orexigen Therapeutics, Inc. | Methods for treating visceral fat conditions |
ES2762113T3 (es) | 2010-01-11 | 2020-05-22 | Nalpropion Pharmaceuticals Inc | Métodos de proporcionar terapia de pérdida de peso en pacientes con depresión mayor |
EP4104824A1 (en) | 2012-06-06 | 2022-12-21 | Nalpropion Pharmaceuticals LLC | Composition for use in a method of treating overweight and obesity in patients with high cardiovascular risk |
US8969371B1 (en) | 2013-12-06 | 2015-03-03 | Orexigen Therapeutics, Inc. | Compositions and methods for weight loss in at risk patient populations |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
RU2197250C2 (ru) * | 2000-10-30 | 2003-01-27 | Соколовский Сергей Ростиславович | Способ лечения наркоманий |
EP2316456B1 (en) * | 2003-04-29 | 2017-06-14 | Orexigen Therapeutics, Inc. | Compositions for affecting weight loss comprising an opioid antagonist and bupropion |
US20070099947A1 (en) * | 2005-11-03 | 2007-05-03 | Alkermes, Inc. | Methods and compositions for the treatment of brain reward system disorders by combination therapy |
WO2007089318A2 (en) * | 2005-11-23 | 2007-08-09 | Orexigen Therapeutics, Inc. | Compositions and methods for reducing food cravings |
US8916195B2 (en) | 2006-06-05 | 2014-12-23 | Orexigen Therapeutics, Inc. | Sustained release formulation of naltrexone |
TW201811315A (zh) | 2006-11-09 | 2018-04-01 | 美商歐瑞根治療有限公司 | 層狀醫藥調配物 |
KR20090090316A (ko) | 2006-11-09 | 2009-08-25 | 오렉시젠 세러퓨틱스 인크. | 체중 감량 약물을 투여하기 위한 단위 용량 팩키지 및 투여 방법 |
GB2447949B (en) * | 2007-03-29 | 2010-03-31 | Renasci Consultancy Ltd | A method for identifying a compound for treating a disorder or condition associated with dysfunction of monoamine neurotransmission |
WO2009035473A2 (en) * | 2007-09-13 | 2009-03-19 | Sanfilippo Louis C | Method of treating binge eating disorder, obesity resulting from binge eating behavior and depressive disorders |
CA2709861A1 (en) * | 2007-12-20 | 2009-07-02 | Neurosearch A/S | Pharmaceutical compositions |
KR20220047894A (ko) * | 2010-11-08 | 2022-04-19 | 오메로스 코포레이션 | Pde7 억제제를 사용한 중독 및 충동-조절 장애의 치료 |
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2011
- 2011-12-02 CN CN2011800595435A patent/CN103298462A/zh active Pending
- 2011-12-02 DK DK11844637.6T patent/DK2646011T3/da active
- 2011-12-02 NO NO11844637A patent/NO2646011T3/no unknown
- 2011-12-02 BR BR112013015957-0A patent/BR112013015957B1/pt active IP Right Grant
- 2011-12-02 SI SI201131336T patent/SI2646011T1/en unknown
- 2011-12-02 EP EP11844637.6A patent/EP2646011B1/en active Active
- 2011-12-02 AU AU2011336298A patent/AU2011336298B2/en active Active
- 2011-12-02 RS RS20171107A patent/RS56548B1/sr unknown
- 2011-12-02 WO PCT/US2011/063170 patent/WO2012075453A1/en active Application Filing
- 2011-12-02 TW TW100144461A patent/TWI536986B/zh active
- 2011-12-02 JP JP2013542227A patent/JP2014508717A/ja active Pending
- 2011-12-02 PL PL11844637T patent/PL2646011T3/pl unknown
- 2011-12-02 LT LTEP11844637.6T patent/LT2646011T/lt unknown
- 2011-12-02 ES ES11844637.6T patent/ES2647232T3/es active Active
- 2011-12-02 CA CA2819003A patent/CA2819003A1/en not_active Abandoned
- 2011-12-02 HU HUE11844637A patent/HUE034641T2/en unknown
- 2011-12-02 RU RU2013127420A patent/RU2620913C2/ru active
- 2011-12-02 TW TW105105528A patent/TW201735912A/zh unknown
- 2011-12-02 PT PT118446376T patent/PT2646011T/pt unknown
- 2011-12-02 AR ARP110104511A patent/AR084093A1/es not_active Application Discontinuation
- 2011-12-02 US US13/991,372 patent/US20130252995A1/en not_active Abandoned
- 2011-12-02 MX MX2013006070A patent/MX350304B/es active IP Right Grant
- 2011-12-02 KR KR1020137017316A patent/KR20140035319A/ko not_active Application Discontinuation
-
2013
- 2013-05-21 IL IL226483A patent/IL226483A0/en unknown
- 2013-05-31 CL CL2013001565A patent/CL2013001565A1/es unknown
-
2017
- 2017-04-27 AU AU2017202793A patent/AU2017202793B2/en active Active
- 2017-11-02 HR HRP20171678TT patent/HRP20171678T1/hr unknown
- 2017-11-14 CY CY20171101188T patent/CY1119560T1/el unknown
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2018
- 2018-06-04 AU AU2018203921A patent/AU2018203921A1/en not_active Abandoned
-
2021
- 2021-06-02 US US17/336,546 patent/US20210283126A1/en active Pending
- 2021-12-23 AR ARP210103652A patent/AR124497A2/es unknown
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