HRP20060040A2 - PURE D-(17α)-13-ETHYL-17-HYDROXY-18,19-DINORPREGN-4-ENE-20-YNE-3-ONE-3E- AND -3Z-OXIME ISOMERS, AS WELL AS PROCESS FOR THE SYNTHESIS OF THE MIXTURE OF ISOMERS AND THE PURE ISOMERS - Google Patents
PURE D-(17α)-13-ETHYL-17-HYDROXY-18,19-DINORPREGN-4-ENE-20-YNE-3-ONE-3E- AND -3Z-OXIME ISOMERS, AS WELL AS PROCESS FOR THE SYNTHESIS OF THE MIXTURE OF ISOMERS AND THE PURE ISOMERSInfo
- Publication number
- HRP20060040A2 HRP20060040A2 HR20060040A HRP20060040A HRP20060040A2 HR P20060040 A2 HRP20060040 A2 HR P20060040A2 HR 20060040 A HR20060040 A HR 20060040A HR P20060040 A HRP20060040 A HR P20060040A HR P20060040 A2 HRP20060040 A2 HR P20060040A2
- Authority
- HR
- Croatia
- Prior art keywords
- isomers
- pure
- dinorpregn
- hydroxy
- synthesis
- Prior art date
Links
- 230000015572 biosynthetic process Effects 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 3
- 238000003786 synthesis reaction Methods 0.000 title abstract 3
- 239000000203 mixture Substances 0.000 title abstract 2
- SYSQUGFVNFXIIT-UHFFFAOYSA-N n-[4-(1,3-benzoxazol-2-yl)phenyl]-4-nitrobenzenesulfonamide Chemical compound C1=CC([N+](=O)[O-])=CC=C1S(=O)(=O)NC1=CC=C(C=2OC3=CC=CC=C3N=2)C=C1 SYSQUGFVNFXIIT-UHFFFAOYSA-N 0.000 title 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 239000013543 active substance Substances 0.000 abstract 1
- 239000000262 estrogen Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000000757 progestagenic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/30—Oestrogens
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/34—Gestagens
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Diabetes (AREA)
- Gynecology & Obstetrics (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Saccharide Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU0301981A HUP0301981A2 (hu) | 2003-06-30 | 2003-06-30 | Tiszta d-(17alfa)-13-etil-17-hidroxi-18,19-dinor-pregn-4-én-20-in-3-on-3E- és 3Z-oxim izomerek, valamint eljárás az izomer keverékek és a tiszta izomerek előállítására |
| PCT/HU2004/000030 WO2005000867A1 (en) | 2003-06-30 | 2004-04-29 | PURE D-(17α)-13-ETHYL-17-HYDROXY-18,19-DINORPREGN-4-ENE-20-YNE-3-ONE-3E- AND -3Z-OXIME ISOMERS, AS WELL AS PROCESS FOR THE SYNTHESIS OF THE MIXTURE OF ISOMERS AND THE PURE ISOMERS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HRP20060040A2 true HRP20060040A2 (en) | 2007-08-31 |
Family
ID=90001693
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HR20060040A HRP20060040A2 (en) | 2003-06-30 | 2006-01-27 | PURE D-(17α)-13-ETHYL-17-HYDROXY-18,19-DINORPREGN-4-ENE-20-YNE-3-ONE-3E- AND -3Z-OXIME ISOMERS, AS WELL AS PROCESS FOR THE SYNTHESIS OF THE MIXTURE OF ISOMERS AND THE PURE ISOMERS |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP1641812B1 (xx) |
| JP (1) | JP2007534617A (xx) |
| CN (1) | CN100497368C (xx) |
| AT (1) | ATE470669T1 (xx) |
| AU (1) | AU2004251117A1 (xx) |
| BR (1) | BRPI0411734A (xx) |
| CA (1) | CA2526305A1 (xx) |
| DE (1) | DE602004027629D1 (xx) |
| EA (1) | EA008174B1 (xx) |
| HR (1) | HRP20060040A2 (xx) |
| HU (1) | HUP0301981A2 (xx) |
| MX (1) | MXPA05012655A (xx) |
| NO (1) | NO20060456L (xx) |
| NZ (1) | NZ544481A (xx) |
| RS (1) | RS20050816A (xx) |
| UA (1) | UA85190C2 (xx) |
| WO (1) | WO2005000867A1 (xx) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6734277B2 (en) | 2002-05-09 | 2004-05-11 | General Electric Company | Method of enhancing pit replication in optical disks |
| US7816546B2 (en) | 2003-06-30 | 2010-10-19 | Richter Gedeon Vegyeszeti Gyar Rt. | Process for the synthesis of high purity d-(17α)-13-ethyl-17-hydroxy-18,19-dinorpregn-4-ene-20-yn-3-one-oxime |
| AU2005272647A1 (en) * | 2004-08-12 | 2006-02-23 | Sicor, Inc. | Process for the preparation of 3-oximino steroids |
| US20070098772A1 (en) * | 2005-09-23 | 2007-05-03 | Westcott Tyler D | Transdermal norelgestromin delivery system |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1123104A (en) * | 1965-10-22 | 1968-08-14 | Ortho Pharma Corp | 3-oxime-steroids and method of preparation |
| DE2409648A1 (de) * | 1973-03-01 | 1974-09-12 | Ortho Pharma Corp | Testosteron-3-oxim-derivate, verfahren zu ihrer herstellung und ihre verwendung als verhuetungsmittel post coitum |
| US4027019A (en) * | 1975-07-24 | 1977-05-31 | Ortho Pharmaceutical Corporation | 3-Oximes of D-17α-ethynyl-19-nortestosterone esters and method |
| JPS624400A (ja) * | 1985-06-29 | 1987-01-10 | 内藤 喜之 | マイクロ波用アンテナ |
| NZ226316A (en) * | 1987-09-24 | 1991-10-25 | Jencap Research Ltd | Pharmaceutical contraceptive preparations and packages containing from 20-35 unit dosages comprising an estrogen and a progestin; the unit dosages having alternating estrogen and progestin dominance |
| JP3534775B2 (ja) * | 1995-06-07 | 2004-06-07 | オーソ―マクニール ファーマシューティカル，インコーポレイテッド | １７−デアセチルノルゲスチマートを単独でまたはエストロゲンと組み合わせて投与するための経皮パッチおよび方法 |
-
2003
- 2003-06-30 HU HU0301981A patent/HUP0301981A2/hu unknown
-
2004
- 2004-04-29 BR BRPI0411734-4A patent/BRPI0411734A/pt not_active IP Right Cessation
- 2004-04-29 MX MXPA05012655A patent/MXPA05012655A/es unknown
- 2004-04-29 JP JP2006518377A patent/JP2007534617A/ja active Pending
- 2004-04-29 EA EA200600120A patent/EA008174B1/ru not_active IP Right Cessation
- 2004-04-29 CN CNB2004800152174A patent/CN100497368C/zh not_active Expired - Fee Related
- 2004-04-29 DE DE602004027629T patent/DE602004027629D1/de not_active Expired - Lifetime
- 2004-04-29 CA CA002526305A patent/CA2526305A1/en not_active Abandoned
- 2004-04-29 EP EP04730317A patent/EP1641812B1/en not_active Expired - Lifetime
- 2004-04-29 UA UAA200600814A patent/UA85190C2/ru unknown
- 2004-04-29 AT AT04730317T patent/ATE470669T1/de not_active IP Right Cessation
- 2004-04-29 NZ NZ544481A patent/NZ544481A/xx unknown
- 2004-04-29 WO PCT/HU2004/000030 patent/WO2005000867A1/en active Application Filing
- 2004-04-29 RS YUP-2005/0816A patent/RS20050816A/sr unknown
- 2004-04-29 AU AU2004251117A patent/AU2004251117A1/en not_active Abandoned
-
2006
- 2006-01-27 NO NO20060456A patent/NO20060456L/no not_active Application Discontinuation
- 2006-01-27 HR HR20060040A patent/HRP20060040A2/xx not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AU2004251117A1 (en) | 2005-01-06 |
| EP1641812A1 (en) | 2006-04-05 |
| DE602004027629D1 (de) | 2010-07-22 |
| EA008174B1 (ru) | 2007-04-27 |
| EP1641812B1 (en) | 2010-06-09 |
| UA85190C2 (xx) | 2009-01-12 |
| NO20060456L (no) | 2006-03-30 |
| JP2007534617A (ja) | 2007-11-29 |
| CN1798758A (zh) | 2006-07-05 |
| CN100497368C (zh) | 2009-06-10 |
| ATE470669T1 (de) | 2010-06-15 |
| NZ544481A (en) | 2009-05-31 |
| EA200600120A1 (ru) | 2006-06-30 |
| HUP0301981D0 (en) | 2003-09-29 |
| MXPA05012655A (es) | 2006-02-22 |
| RS20050816A (xx) | 2007-08-03 |
| HUP0301981A2 (hu) | 2005-04-28 |
| BRPI0411734A (pt) | 2006-08-08 |
| CA2526305A1 (en) | 2005-01-06 |
| WO2005000867A1 (en) | 2005-01-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| A1OB | Publication of a patent application | ||
| AIPI | Request for the grant of a patent on the basis of a substantive examination of a patent application | ||
| ODRP | Renewal fee for the maintenance of a patent |
Payment date: 20090414 Year of fee payment: 6 |
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| OBST | Application withdrawn |