HK1250138A1 - 毒蕈碱激動劑 - Google Patents

毒蕈碱激動劑

Info

Publication number
HK1250138A1
HK1250138A1 HK18109572.7A HK18109572A HK1250138A1 HK 1250138 A1 HK1250138 A1 HK 1250138A1 HK 18109572 A HK18109572 A HK 18109572A HK 1250138 A1 HK1250138 A1 HK 1250138A1
Authority
HK
Hong Kong
Prior art keywords
muscarinic agonists
muscarinic
agonists
Prior art date
Application number
HK18109572.7A
Other languages
English (en)
Inventor
蓋爾斯‧艾伯特‧布朗
朱莉‧坎斯菲爾德
馬克‧皮克沃斯
本杰明‧杰拉爾德‧特漢
Original Assignee
赫普泰雅治療有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 赫普泰雅治療有限公司 filed Critical 赫普泰雅治療有限公司
Publication of HK1250138A1 publication Critical patent/HK1250138A1/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK18109572.7A 2015-08-03 2018-07-24 毒蕈碱激動劑 HK1250138A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB1513743.3A GB201513743D0 (en) 2015-08-03 2015-08-03 Muscarinic agonists
PCT/GB2016/052385 WO2017021729A1 (en) 2015-08-03 2016-08-03 Muscarinic agonists

Publications (1)

Publication Number Publication Date
HK1250138A1 true HK1250138A1 (zh) 2018-11-30

Family

ID=54063149

Family Applications (1)

Application Number Title Priority Date Filing Date
HK18109572.7A HK1250138A1 (zh) 2015-08-03 2018-07-24 毒蕈碱激動劑

Country Status (11)

Country Link
US (3) US10738029B2 (zh)
EP (1) EP3331529B1 (zh)
JP (1) JP6843114B2 (zh)
CN (1) CN108025004B (zh)
AU (1) AU2016304387B2 (zh)
CA (1) CA2994203C (zh)
DK (1) DK3331529T3 (zh)
ES (1) ES2894637T3 (zh)
GB (1) GB201513743D0 (zh)
HK (1) HK1250138A1 (zh)
WO (1) WO2017021729A1 (zh)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN106831541B (zh) 2011-11-18 2019-09-06 赫普泰雅治疗有限公司 毒蕈碱性m1受体激动剂
GB201513743D0 (en) 2015-08-03 2015-09-16 Heptares Therapeutics Ltd Muscarinic agonists
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AU2018352828A1 (en) 2017-10-17 2020-04-23 Vanderbilt University Antagonists of the muscarinic acetylcholine receptor M4
CA3094366A1 (en) * 2018-03-23 2019-09-26 Pfizer Inc. Piperazine azaspiro derivatives
GB201810245D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201810239D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds
CR20220153A (es) * 2019-10-09 2022-05-03 Novartis Ag Derivados de 2–azaespiro [3.4] octano como agonistas de m4
CA3156320A1 (en) * 2019-10-09 2021-04-15 Novartis Ag 2-AZASPIRO[3,4] OCTANE DERIVATIVES USED AS M4 AGONISTS

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GB201810239D0 (en) 2018-06-22 2018-08-08 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819961D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB201819960D0 (en) 2018-12-07 2019-01-23 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202020191D0 (en) 2020-12-18 2021-02-03 Heptares Therapeutics Ltd Pharmaceutical compounds
GB202103211D0 (en) 2021-03-08 2021-04-21 Heptares Therapeutics Ltd Pharmaceutical compounds for use in therapy

Also Published As

Publication number Publication date
JP6843114B2 (ja) 2021-03-17
US12024499B2 (en) 2024-07-02
US20230002354A1 (en) 2023-01-05
WO2017021729A1 (en) 2017-02-09
AU2016304387A1 (en) 2018-02-22
CA2994203A1 (en) 2017-02-09
AU2016304387B2 (en) 2020-10-22
US20200354339A1 (en) 2020-11-12
US20180222885A1 (en) 2018-08-09
EP3331529B1 (en) 2021-09-29
JP2018522033A (ja) 2018-08-09
EP3331529A1 (en) 2018-06-13
CN108025004A (zh) 2018-05-11
GB201513743D0 (en) 2015-09-16
US10738029B2 (en) 2020-08-11
CA2994203C (en) 2023-11-28
US11254656B2 (en) 2022-02-22
ES2894637T3 (es) 2022-02-15
CN108025004B (zh) 2021-07-09
DK3331529T3 (da) 2021-10-18

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