HK1211863A1 - Substituted isoxazole amine compounds as inhibitors of scd1 scd1 - Google Patents
Substituted isoxazole amine compounds as inhibitors of scd1 scd1Info
- Publication number
- HK1211863A1 HK1211863A1 HK15112883.8A HK15112883A HK1211863A1 HK 1211863 A1 HK1211863 A1 HK 1211863A1 HK 15112883 A HK15112883 A HK 15112883A HK 1211863 A1 HK1211863 A1 HK 1211863A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- scd1
- inhibitors
- amine compounds
- substituted isoxazole
- isoxazole amine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/14—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Epidemiology (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261732463P | 2012-12-03 | 2012-12-03 | |
| PCT/EP2013/075035 WO2014086667A1 (en) | 2012-12-03 | 2013-11-29 | Substituted isoxazole amine compounds as inhibitors of scd1 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HK1211863A1 true HK1211863A1 (en) | 2016-06-03 |
Family
ID=49709654
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HK15112883.8A HK1211863A1 (en) | 2012-12-03 | 2015-12-31 | Substituted isoxazole amine compounds as inhibitors of scd1 scd1 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US9290465B2 (pt) |
| EP (1) | EP2925408A1 (pt) |
| JP (1) | JP2016501210A (pt) |
| KR (1) | KR20150091071A (pt) |
| CN (1) | CN104822420A (pt) |
| BR (1) | BR112015012877A2 (pt) |
| CA (1) | CA2890300A1 (pt) |
| HK (1) | HK1211863A1 (pt) |
| MX (1) | MX2015006930A (pt) |
| RU (1) | RU2015123276A (pt) |
| WO (1) | WO2014086667A1 (pt) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MA46589A (fr) | 2016-10-24 | 2019-08-28 | Yumanity Therapeutics Inc | Composés et utilisations de ces derniers |
| CN110392833A (zh) | 2017-01-06 | 2019-10-29 | 优曼尼蒂治疗公司 | 治疗神经病症的方法 |
| US11873298B2 (en) | 2017-10-24 | 2024-01-16 | Janssen Pharmaceutica Nv | Compounds and uses thereof |
| EP3914593A4 (en) | 2019-01-24 | 2022-11-02 | Yumanity Therapeutics, Inc. | COMPOUNDS AND THEIR USES |
| CN112724157B (zh) * | 2021-01-23 | 2022-04-19 | 中国科学院新疆理化技术研究所 | 二氢噁唑并[5,4-d]吡咯并[1,2-a]嘧啶-9(5H)-酮类衍生物及用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BRPI0515483A (pt) * | 2004-09-20 | 2008-07-22 | Xenon Pharmaceuticals Inc | derivados heterocìclicos para o tratamento de doenças mediadas por enzimas estearoil-coa desaturase |
| AU2008241313A1 (en) * | 2007-04-20 | 2008-10-30 | Merck Frosst Canada Ltd. | Novel heteroaromatic compounds as inhibitors of stearoyl-coenzyme a delta-9 desaturase |
| US20100249192A1 (en) * | 2007-12-11 | 2010-09-30 | Merck Frosst Canada Ltd. | Novel heteroaromatic compounds as inhibitors of stearoyl-coenzyme a delta-9 desaturase |
-
2013
- 2013-11-29 MX MX2015006930A patent/MX2015006930A/es unknown
- 2013-11-29 EP EP13799270.7A patent/EP2925408A1/en not_active Withdrawn
- 2013-11-29 KR KR1020157014612A patent/KR20150091071A/ko not_active Application Discontinuation
- 2013-11-29 CN CN201380063224.0A patent/CN104822420A/zh active Pending
- 2013-11-29 JP JP2015544468A patent/JP2016501210A/ja active Pending
- 2013-11-29 US US14/443,849 patent/US9290465B2/en not_active Expired - Fee Related
- 2013-11-29 CA CA2890300A patent/CA2890300A1/en not_active Abandoned
- 2013-11-29 WO PCT/EP2013/075035 patent/WO2014086667A1/en active Application Filing
- 2013-11-29 BR BR112015012877A patent/BR112015012877A2/pt not_active Application Discontinuation
- 2013-11-29 RU RU2015123276A patent/RU2015123276A/ru unknown
-
2015
- 2015-12-31 HK HK15112883.8A patent/HK1211863A1/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US9290465B2 (en) | 2016-03-22 |
| CN104822420A (zh) | 2015-08-05 |
| WO2014086667A1 (en) | 2014-06-12 |
| MX2015006930A (es) | 2015-09-08 |
| RU2015123276A (ru) | 2017-01-13 |
| CA2890300A1 (en) | 2014-06-12 |
| BR112015012877A2 (pt) | 2018-04-24 |
| JP2016501210A (ja) | 2016-01-18 |
| KR20150091071A (ko) | 2015-08-07 |
| EP2925408A1 (en) | 2015-10-07 |
| US20150315160A1 (en) | 2015-11-05 |
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