BR112015012877A2 - composto de fórmula, composição farmacêutica, uso do composto e método para o tratamento do câncer - Google Patents

composto de fórmula, composição farmacêutica, uso do composto e método para o tratamento do câncer

Info

Publication number
BR112015012877A2
BR112015012877A2 BR112015012877A BR112015012877A BR112015012877A2 BR 112015012877 A2 BR112015012877 A2 BR 112015012877A2 BR 112015012877 A BR112015012877 A BR 112015012877A BR 112015012877 A BR112015012877 A BR 112015012877A BR 112015012877 A2 BR112015012877 A2 BR 112015012877A2
Authority
BR
Brazil
Prior art keywords
compound
pharmaceutical composition
cancer treatment
formula
formula compound
Prior art date
Application number
BR112015012877A
Other languages
English (en)
Inventor
Mertz Eric
Derryberry Johnmark
Gillespie Paul
David Erickson Shawn
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of BR112015012877A2 publication Critical patent/BR112015012877A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/14Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Epidemiology (AREA)
BR112015012877A 2012-12-03 2013-11-29 composto de fórmula, composição farmacêutica, uso do composto e método para o tratamento do câncer BR112015012877A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261732463P 2012-12-03 2012-12-03
PCT/EP2013/075035 WO2014086667A1 (en) 2012-12-03 2013-11-29 Substituted isoxazole amine compounds as inhibitors of scd1

Publications (1)

Publication Number Publication Date
BR112015012877A2 true BR112015012877A2 (pt) 2018-04-24

Family

ID=49709654

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015012877A BR112015012877A2 (pt) 2012-12-03 2013-11-29 composto de fórmula, composição farmacêutica, uso do composto e método para o tratamento do câncer

Country Status (11)

Country Link
US (1) US9290465B2 (pt)
EP (1) EP2925408A1 (pt)
JP (1) JP2016501210A (pt)
KR (1) KR20150091071A (pt)
CN (1) CN104822420A (pt)
BR (1) BR112015012877A2 (pt)
CA (1) CA2890300A1 (pt)
HK (1) HK1211863A1 (pt)
MX (1) MX2015006930A (pt)
RU (1) RU2015123276A (pt)
WO (1) WO2014086667A1 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3529245A4 (en) 2016-10-24 2020-12-23 Yumanity Therapeutics, Inc. COMPOUNDS AND USES OF THE LATEST
IL304017A (en) 2017-01-06 2023-08-01 Yumanity Therapeutics Inc Methods for treating neurological disorders
CA3083000A1 (en) 2017-10-24 2019-05-02 Yumanity Therapeutics, Inc. Compounds and uses thereof
CN112724157B (zh) * 2021-01-23 2022-04-19 中国科学院新疆理化技术研究所 二氢噁唑并[5,4-d]吡咯并[1,2-a]嘧啶-9(5H)-酮类衍生物及用途

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7919496B2 (en) * 2004-09-20 2011-04-05 Xenon Pharmaceuticals Inc. Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-CoA desaturase enzymes
EP2148878A4 (en) * 2007-04-20 2011-08-10 Merck Canada Inc NEW HETEROAROMATIC COMPOUNDS AS INHIBITORS OF STEAROYL-COENZYME-A-DELTA-9-DESATURASE
WO2009073973A1 (en) * 2007-12-11 2009-06-18 Merck Frosst Canada Ltd. Novel heteroaromatic compounds as inhibitors of stearoyl-coenzyme a delta-9 desaturase

Also Published As

Publication number Publication date
US20150315160A1 (en) 2015-11-05
WO2014086667A1 (en) 2014-06-12
CN104822420A (zh) 2015-08-05
JP2016501210A (ja) 2016-01-18
KR20150091071A (ko) 2015-08-07
MX2015006930A (es) 2015-09-08
CA2890300A1 (en) 2014-06-12
HK1211863A1 (en) 2016-06-03
US9290465B2 (en) 2016-03-22
RU2015123276A (ru) 2017-01-13
EP2925408A1 (en) 2015-10-07

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired
B350 Update of information on the portal [chapter 15.35 patent gazette]