HK1202117A1 - Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an so2-containing group as vanilloid receptor ligands - Google Patents

Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an so2-containing group as vanilloid receptor ligands Download PDF

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Publication number
HK1202117A1
HK1202117A1 HK15102581.4A HK15102581A HK1202117A1 HK 1202117 A1 HK1202117 A1 HK 1202117A1 HK 15102581 A HK15102581 A HK 15102581A HK 1202117 A1 HK1202117 A1 HK 1202117A1
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HK
Hong Kong
Prior art keywords
substituted
containing group
receptor ligands
phenyl moiety
urea derivatives
Prior art date
Application number
HK15102581.4A
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English (en)
Chinese (zh)
Inventor
Robert Frank-Foltyn
Thomas Christoph
Nils Damann
Bernhard Lesch
Gregor Bahrenberg
Derek John Saunders
Hannelore Stockhausen
Yong-Soo Kim
Myeong-Seop Kim
Jeewoo Lee
Original Assignee
Grünenthal GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Grünenthal GmbH filed Critical Grünenthal GmbH
Publication of HK1202117A1 publication Critical patent/HK1202117A1/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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HK15102581.4A 2011-11-09 2012-11-08 Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an so2-containing group as vanilloid receptor ligands HK1202117A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11008927 2011-11-09
EP11008927.3 2011-11-09
PCT/EP2012/072143 WO2013068464A1 (en) 2011-11-09 2012-11-08 Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an so2-containing group as vanilloid receptor ligands

Publications (1)

Publication Number Publication Date
HK1202117A1 true HK1202117A1 (en) 2015-09-18

Family

ID=47143914

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Application Number Title Priority Date Filing Date
HK15102581.4A HK1202117A1 (en) 2011-11-09 2012-11-08 Substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with an so2-containing group as vanilloid receptor ligands

Country Status (13)

Country Link
EP (1) EP2776401A1 (enrdf_load_html_response)
JP (1) JP2014532744A (enrdf_load_html_response)
KR (1) KR20140091041A (enrdf_load_html_response)
CN (1) CN104066720A (enrdf_load_html_response)
AR (1) AR088799A1 (enrdf_load_html_response)
AU (1) AU2012334068A1 (enrdf_load_html_response)
BR (1) BR112014011108A2 (enrdf_load_html_response)
CA (1) CA2854424A1 (enrdf_load_html_response)
HK (1) HK1202117A1 (enrdf_load_html_response)
IN (1) IN2014KN00865A (enrdf_load_html_response)
MX (1) MX2014005233A (enrdf_load_html_response)
TW (1) TW201326135A (enrdf_load_html_response)
WO (1) WO2013068464A1 (enrdf_load_html_response)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2836373T3 (es) 2014-03-07 2021-06-24 Biocryst Pharm Inc Pirazoles sustituidos con trifluorometilo como inhibidores de calicreína del plasma humano
KR101909092B1 (ko) 2014-11-24 2018-10-17 (주) 메디프론디비티 바닐로이드 수용체 리간드 ii로서의 치환된 옥사졸계 및 싸이아졸계 카복스아미드 및 우레아 유도체
CN114920697A (zh) * 2022-05-16 2022-08-19 河南应用技术职业学院 杂环基取代的茚满丙酰胺类化合物及其应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR076752A1 (es) 2009-05-07 2011-07-06 Gruenenthal Chemie Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloides.
TWI504589B (zh) 2009-05-07 2015-10-21 作為香草類化合物受體之配體之經取代芳香族羧醯胺及尿素衍生物

Also Published As

Publication number Publication date
TW201326135A (zh) 2013-07-01
WO2013068464A1 (en) 2013-05-16
AR088799A1 (es) 2014-07-10
BR112014011108A2 (pt) 2017-05-16
MX2014005233A (es) 2014-08-22
AU2012334068A1 (en) 2014-05-22
IN2014KN00865A (enrdf_load_html_response) 2015-10-02
EP2776401A1 (en) 2014-09-17
JP2014532744A (ja) 2014-12-08
CN104066720A (zh) 2014-09-24
KR20140091041A (ko) 2014-07-18
CA2854424A1 (en) 2013-05-16

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