HK1179606A1 - 酰胺基-托烷衍生物 - Google Patents
酰胺基-托烷衍生物Info
- Publication number
- HK1179606A1 HK1179606A1 HK13106598.8A HK13106598A HK1179606A1 HK 1179606 A1 HK1179606 A1 HK 1179606A1 HK 13106598 A HK13106598 A HK 13106598A HK 1179606 A1 HK1179606 A1 HK 1179606A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- amido
- tropane derivatives
- tropane
- derivatives
- amido tropane
- Prior art date
Links
- -1 Amido tropane derivatives Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10166757 | 2010-06-22 | ||
PCT/EP2011/060073 WO2011161006A1 (en) | 2010-06-22 | 2011-06-17 | Amido-tropane derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1179606A1 true HK1179606A1 (zh) | 2013-10-04 |
Family
ID=44310862
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK13106598.8A HK1179606A1 (zh) | 2010-06-22 | 2013-06-05 | 酰胺基-托烷衍生物 |
Country Status (24)
Country | Link |
---|---|
US (1) | US8153653B2 (zh) |
EP (1) | EP2585456B1 (zh) |
JP (1) | JP5546684B2 (zh) |
KR (1) | KR101445016B1 (zh) |
CN (1) | CN102947297B (zh) |
AR (1) | AR081961A1 (zh) |
AU (1) | AU2011269145A1 (zh) |
BR (1) | BR112012032576A2 (zh) |
CA (1) | CA2801458C (zh) |
CL (1) | CL2012003552A1 (zh) |
CO (1) | CO6630160A2 (zh) |
CR (1) | CR20120614A (zh) |
EA (1) | EA201291374A1 (zh) |
EC (1) | ECSP12012347A (zh) |
ES (1) | ES2550831T3 (zh) |
HK (1) | HK1179606A1 (zh) |
IL (1) | IL222998A0 (zh) |
MA (1) | MA34251B1 (zh) |
MX (1) | MX2012013820A (zh) |
PE (1) | PE20130317A1 (zh) |
SG (1) | SG186329A1 (zh) |
TW (1) | TWI417097B (zh) |
WO (1) | WO2011161006A1 (zh) |
ZA (1) | ZA201209248B (zh) |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PT885220E (pt) * | 1996-02-22 | 2001-11-30 | Neurosearch As | Derivados de tropano a sua preparacao e utilizacao |
US5834484A (en) * | 1997-03-12 | 1998-11-10 | Board Of Supervisors Of Louisiana State University And Agricultural And Mechanical College | Cocaine analogs |
JP4563386B2 (ja) * | 2003-09-09 | 2010-10-13 | エフ.ホフマン−ラ ロシュ アーゲー | 精神病の処置のためのグリシン取り込み阻害剤としての1−(2−アミノ−ベンゾール)−ピペラジン誘導体 |
FR2861076B1 (fr) | 2003-10-17 | 2006-01-06 | Sanofi Synthelabo | Derives de n-heterocyclymethylbenzamide, leur preparation et leur application en therapeutique |
EP1745018A1 (en) * | 2004-04-29 | 2007-01-24 | Merck & Co., Inc. | Azetidine glycine transporter inhibitors |
FR2873693B1 (fr) * | 2004-07-29 | 2006-09-15 | Sanofi Synthelabo | Derives d'amino-tropane, leur preparation et leur application en therapeutique |
GB0428231D0 (en) * | 2004-12-23 | 2005-01-26 | Glaxo Group Ltd | Compounds |
EP1836178A1 (en) * | 2005-01-06 | 2007-09-26 | F. Hoffmann-Roche AG | Sulfanyl substituted phenyl methanones as glycine transporter 1 (glyt-1) inhibitors for the treatment of neurological and neuropsychiatric disorders |
JP2010517959A (ja) * | 2007-02-01 | 2010-05-27 | グラクソ グループ リミテッド | GlyT1トランスポーター阻害薬および神経学的および神経精神病学的障害の治療におけるその使用 |
WO2010020548A1 (en) * | 2008-08-20 | 2010-02-25 | F. Hoffmann-La Roche Ag | Glyt1 receptor antagonists |
-
2011
- 2011-06-15 US US13/160,559 patent/US8153653B2/en not_active Expired - Fee Related
- 2011-06-17 ES ES11728224.4T patent/ES2550831T3/es active Active
- 2011-06-17 BR BR112012032576A patent/BR112012032576A2/pt active Search and Examination
- 2011-06-17 JP JP2013515816A patent/JP5546684B2/ja not_active Expired - Fee Related
- 2011-06-17 KR KR1020127033182A patent/KR101445016B1/ko active IP Right Grant
- 2011-06-17 CN CN201180030703.3A patent/CN102947297B/zh not_active Expired - Fee Related
- 2011-06-17 WO PCT/EP2011/060073 patent/WO2011161006A1/en active Application Filing
- 2011-06-17 SG SG2012091708A patent/SG186329A1/en unknown
- 2011-06-17 PE PE2012002444A patent/PE20130317A1/es not_active Application Discontinuation
- 2011-06-17 MA MA35398A patent/MA34251B1/fr unknown
- 2011-06-17 CA CA2801458A patent/CA2801458C/en not_active Expired - Fee Related
- 2011-06-17 AU AU2011269145A patent/AU2011269145A1/en not_active Abandoned
- 2011-06-17 EP EP11728224.4A patent/EP2585456B1/en active Active
- 2011-06-17 MX MX2012013820A patent/MX2012013820A/es active IP Right Grant
- 2011-06-17 EA EA201291374A patent/EA201291374A1/ru unknown
- 2011-06-20 TW TW100121503A patent/TWI417097B/zh not_active IP Right Cessation
- 2011-06-21 AR ARP110102138A patent/AR081961A1/es unknown
-
2012
- 2012-10-26 CO CO12192372A patent/CO6630160A2/es active IP Right Grant
- 2012-11-12 IL IL222998A patent/IL222998A0/en unknown
- 2012-12-05 CR CR20120614A patent/CR20120614A/es unknown
- 2012-12-06 ZA ZA2012/09248A patent/ZA201209248B/en unknown
- 2012-12-17 CL CL2012003552A patent/CL2012003552A1/es unknown
- 2012-12-20 EC ECSP12012347 patent/ECSP12012347A/es unknown
-
2013
- 2013-06-05 HK HK13106598.8A patent/HK1179606A1/zh not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
EP2585456B1 (en) | 2015-09-16 |
CR20120614A (es) | 2013-01-11 |
WO2011161006A1 (en) | 2011-12-29 |
IL222998A0 (en) | 2013-02-03 |
US20110312993A1 (en) | 2011-12-22 |
SG186329A1 (en) | 2013-01-30 |
ZA201209248B (en) | 2013-08-28 |
KR101445016B1 (ko) | 2014-09-26 |
MA34251B1 (fr) | 2013-05-02 |
US8153653B2 (en) | 2012-04-10 |
PE20130317A1 (es) | 2013-03-11 |
AU2011269145A1 (en) | 2012-11-08 |
AR081961A1 (es) | 2012-10-31 |
EP2585456A1 (en) | 2013-05-01 |
JP2013529607A (ja) | 2013-07-22 |
CA2801458C (en) | 2018-10-30 |
CL2012003552A1 (es) | 2013-04-12 |
KR20130029414A (ko) | 2013-03-22 |
ECSP12012347A (es) | 2013-01-31 |
JP5546684B2 (ja) | 2014-07-09 |
CA2801458A1 (en) | 2011-12-29 |
CN102947297B (zh) | 2015-12-16 |
TWI417097B (zh) | 2013-12-01 |
MX2012013820A (es) | 2013-01-28 |
EA201291374A1 (ru) | 2013-06-28 |
ES2550831T3 (es) | 2015-11-12 |
CN102947297A (zh) | 2013-02-27 |
TW201206438A (en) | 2012-02-16 |
BR112012032576A2 (pt) | 2016-11-22 |
CO6630160A2 (es) | 2013-03-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20230615 |