HK1084394A1 - Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use for preparing neurokinin antagonists - Google Patents

Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use for preparing neurokinin antagonists

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Publication number
HK1084394A1
HK1084394A1 HK06104676.7A HK06104676A HK1084394A1 HK 1084394 A1 HK1084394 A1 HK 1084394A1 HK 06104676 A HK06104676 A HK 06104676A HK 1084394 A1 HK1084394 A1 HK 1084394A1
Authority
HK
Hong Kong
Prior art keywords
piperidin
substituted
preparing
piperazine derivatives
neurokinin antagonists
Prior art date
Application number
HK06104676.7A
Other languages
English (en)
Inventor
Frans Eduard Janssens
Francois Maria Sommen
Boeck Benoit Christian Albert Ghislain De
Joseph Elisabeth Leenaerts
Yves Emiel Maria Van Roosbroeck
Gaston Stanislas Marcella Diels
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/EP2002/014836 external-priority patent/WO2004056772A1/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of HK1084394A1 publication Critical patent/HK1084394A1/xx

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HK06104676.7A 2002-10-08 2006-04-19 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use for preparing neurokinin antagonists HK1084394A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP0211328 2002-10-08
PCT/EP2002/014836 WO2004056772A1 (en) 2002-12-23 2002-12-23 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as tachykinin antagonists
PCT/EP2003/050697 WO2004033428A1 (en) 2002-10-08 2003-10-07 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists

Publications (1)

Publication Number Publication Date
HK1084394A1 true HK1084394A1 (en) 2006-07-28

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JP2006510602A (ja) 2006-03-30
IL167885A (en) 2010-04-29
US20060167008A1 (en) 2006-07-27
EA200500616A1 (ru) 2005-10-27
ES2319642T3 (es) 2009-05-11
KR101049074B1 (ko) 2011-07-15
TW200413319A (en) 2004-08-01
EP1551804B1 (en) 2008-12-24
ATE418543T1 (de) 2009-01-15
CA2499903A1 (en) 2004-04-22
MY141736A (en) 2010-06-15
BR0315098A (pt) 2005-08-16
EA009217B1 (ru) 2007-12-28
EP1551804A1 (en) 2005-07-13
AU2003282115B2 (en) 2009-10-01
US7410970B2 (en) 2008-08-12
PA8584901A1 (es) 2005-10-28
JP4674086B2 (ja) 2011-04-20
AU2003282115A1 (en) 2004-05-04
CA2499903C (en) 2011-06-14
HRP20050309A2 (en) 2006-07-31
AR041545A1 (es) 2005-05-18
WO2004033428A1 (en) 2004-04-22
DE60325493D1 (de) 2009-02-05
TWI324995B (en) 2010-05-21

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