GT200500320A - Metabolitos glucuronidos de tigeciclina y epimeros de los mismos - Google Patents

Metabolitos glucuronidos de tigeciclina y epimeros de los mismos

Info

Publication number
GT200500320A
GT200500320A GT200500320A GT200500320A GT200500320A GT 200500320 A GT200500320 A GT 200500320A GT 200500320 A GT200500320 A GT 200500320A GT 200500320 A GT200500320 A GT 200500320A GT 200500320 A GT200500320 A GT 200500320A
Authority
GT
Guatemala
Prior art keywords
tigecicline
glucuronid
metabolites
same
glucurònids
Prior art date
Application number
GT200500320A
Other languages
English (en)
Inventor
Ronald A Jordan
William Demaio
Matthew Hoffmann
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT200500320A publication Critical patent/GT200500320A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Peptides Or Proteins (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Investigating Or Analysing Materials By Optical Means (AREA)
  • Other Investigation Or Analysis Of Materials By Electrical Means (AREA)

Abstract

LA PRESENTE INVENCIÒN SE REFIERE A GLUCURÒNIDOS, MÀS PARTICULARMENTE A GLUCURÒNIDOS DERIVADOS DE TIGECICLINA. LA TIGECICLINA ES UN ANTIBIÒTICO DE GLICILCICLINA Y UN ANÀLOGO DE LA TETRACICLINA SEMISINTÈTICA, MINOCICLINA QUE SON ACTIVOS CONTRA MUCHAS BACTERIAS PATOGÈNICAS GRAMPOSITIVAS RESISTENTES A ANTIBIÒTICOS.
GT200500320A 2004-11-05 2005-11-04 Metabolitos glucuronidos de tigeciclina y epimeros de los mismos GT200500320A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US62512104P 2004-11-05 2004-11-05

Publications (1)

Publication Number Publication Date
GT200500320A true GT200500320A (es) 2006-06-02

Family

ID=36337018

Family Applications (1)

Application Number Title Priority Date Filing Date
GT200500320A GT200500320A (es) 2004-11-05 2005-11-04 Metabolitos glucuronidos de tigeciclina y epimeros de los mismos

Country Status (22)

Country Link
US (1) US7534766B2 (es)
EP (1) EP1807441A2 (es)
JP (1) JP2008519038A (es)
KR (1) KR20070085761A (es)
CN (1) CN101132799A (es)
AR (1) AR051236A1 (es)
AU (1) AU2005304957A1 (es)
BR (1) BRPI0517715A (es)
CA (1) CA2586245A1 (es)
CR (1) CR9111A (es)
GT (1) GT200500320A (es)
HN (1) HN2005030775A (es)
IL (1) IL182640A0 (es)
MX (1) MX2007005105A (es)
NO (1) NO20072226L (es)
PA (1) PA8652001A1 (es)
PE (1) PE20061048A1 (es)
RU (1) RU2007116800A (es)
SV (1) SV2006002294A (es)
TW (1) TW200628485A (es)
WO (1) WO2006052717A2 (es)
ZA (1) ZA200703624B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2695259C (en) * 2007-07-31 2016-05-24 Gilead Colorado, Inc. Metabolites and derivatives of ambrisentan
US8766177B2 (en) 2010-10-11 2014-07-01 University Of North Texas Nanomanipulation coupled nanospray mass spectrometry (NMS)
JP6134191B2 (ja) 2013-04-07 2017-05-24 村川 惠美 回転型セミバッチａｌｄ装置

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG52361A1 (en) 1991-10-04 1998-09-28 American Cyanamid Co Novel 7-substituted-9-substituted amino-6-demethyl-6-deoxytetracyclines
US5494903A (en) 1991-10-04 1996-02-27 American Cyanamid Company 7-substituted-9-substituted amino-6-demethyl-6-deoxytetracyclines
US5284963A (en) 1992-08-13 1994-02-08 American Cyanamid Company Method of producing 7-(substituted)-9-[(substituted glycyl)-amidol]-6-demethyl-6-deoxytetra-cyclines
US5328902A (en) 1992-08-13 1994-07-12 American Cyanamid Co. 7-(substituted)-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
SG47520A1 (en) 1992-08-13 1998-04-17 American Cyanamid Co New method for the production of 9-amino-6-demethyl-6-deoxytetracycline
US5420272A (en) 1992-08-13 1995-05-30 American Cyanamid Company 7-(substituted)-8-(substituted)-9-](substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
EP2319829A1 (en) 2003-07-09 2011-05-11 Paratek Pharmaceuticals, Inc. 9-substituted tetracycline compounds
US20050137174A1 (en) 2003-07-09 2005-06-23 Paratek Pharmaceuticals, Inc. Prodrugs of 9-aminomethyl tetracycline compounds
US20050148553A1 (en) 2003-09-05 2005-07-07 Testa Raymond T. Use of tigecycline, alone, or in combination with rifampin to treat osteomyelitis and/or septic arthritis

Also Published As

Publication number Publication date
US20060128950A1 (en) 2006-06-15
CN101132799A (zh) 2008-02-27
SV2006002294A (es) 2006-10-13
AR051236A1 (es) 2006-12-27
IL182640A0 (en) 2007-07-24
CR9111A (es) 2008-01-21
MX2007005105A (es) 2007-06-26
NO20072226L (no) 2007-06-04
KR20070085761A (ko) 2007-08-27
JP2008519038A (ja) 2008-06-05
TW200628485A (en) 2006-08-16
WO2006052717A2 (en) 2006-05-18
HN2005030775A (es) 2006-12-18
PE20061048A1 (es) 2006-11-15
BRPI0517715A (pt) 2008-10-21
WO2006052717A3 (en) 2007-11-15
PA8652001A1 (es) 2006-10-13
ZA200703624B (en) 2009-10-28
EP1807441A2 (en) 2007-07-18
AU2005304957A1 (en) 2006-05-18
CA2586245A1 (en) 2006-05-18
US7534766B2 (en) 2009-05-19
RU2007116800A (ru) 2008-12-10

Similar Documents

Publication Publication Date Title
DK1753440T3 (da) Oral administrationsform indeholdende probiotiske bakterier
TW200833465A (en) Retaining ring, flexible membrane for applying load to a retaining ring, and retaining ring assembly
MX2008007808A (es) Analogos de rifamicina y usos de ellos.
IL162318A0 (en) Transmission for a remote catheterization system
CO5570678A2 (es) N-alquilo-4-metileneamino-3-hidroxilo-2-piridonas como anti- microbianos
TW200738695A (en) Cis-4,5-biaryl-2-heterocyclic-imidazolines as MDM2 inhibitors
RS52183B (en) CRYSTAL SOLID RAZAGILINE BASE
FR2938439B1 (fr) Extrait de parties aeriennes d'avoine recoltees avant epiaison
CA112249S (en) Pet house carrier
ZA200709481B (en) Diaryl-purine, azapurines and -deazapurines as non-nucleoside reverse transcriptase inhibitors for treatment of HIV
GT200500187A (es) Moduladores de andrògenos
GB2450007A (en) Dynamic update adaptive idle timer
DE602004004808D1 (de) Acyloxymethylcarbamat-prodrugs von oxazolidinonen
CY1112877T1 (el) Μεταλλαγματα αυξητικου παραγoντα υψηλης δραστικοτητας
GT200600236A (es) PENEMES BICICLICOS DE 6-ALQUILIDENO COMO INHIBIDORES DE beta-LACTAMASAS CALSE D
GT200500320A (es) Metabolitos glucuronidos de tigeciclina y epimeros de los mismos
NZ586723A (en) Use of Biota orientalis for treating osteoarthritis
MX2023009146A (es) Anticuerpos y usos de estos.
FR2897780B1 (fr) Utilisation de la proteine a homeodomaine engrailed comme anxiolytique
EA201101113A1 (ru) Пестицидные комбинации
RU2008112962A (ru) ШТАММ БАЗИДИАЛЬНОГО ГРИБА Fomitopsis officinalis, ПРОЯВЛЯЮЩИЙ АНТИБАКТЕРИАЛЬНУЮ АКТИВНОСТЬ В ОТНОШЕНИИ БАКТЕРИЙ Yersinia pseudotuberculosis
GT200400259A (es) Derivados oxazol de tetraciclinas
RU2008145068A (ru) Слуховой аппарат с радиоканалом
AU2019902106A0 (en) ANTI MICROBIAL PLANT BASED CHEWING GUM. Our product is made from plant based gums from a variety of trees which exhibit antimicrobial activity. It is an environmentally friendly product that is biodegradable and offers health benefits. The said gum base is obtained from trunk exudates (gums) from various trees including the Dipterocarpaceae family of trees, mainly those of the genera Shorea, Balanocarpus or Hopea, and trees of the genus Pistachia. The trunk exudates of the aforementioned trees are mainly composed of triterpenes and triterpenoids with well-known antimicrobial activities.
RU2007123856A (ru) Средство, препятствующее развитию депрессии эритроидного ростка кроветворения при введении цитостатика