GT200100113AA - Nuevo procedimiento para la preparacion de pirazolopirimidinonas . - Google Patents
Nuevo procedimiento para la preparacion de pirazolopirimidinonas .Info
- Publication number
- GT200100113AA GT200100113AA GT200100113AK GT200100113K GT200100113AA GT 200100113A A GT200100113A A GT 200100113AA GT 200100113A K GT200100113A K GT 200100113AK GT 200100113 K GT200100113 K GT 200100113K GT 200100113A A GT200100113A A GT 200100113AA
- Authority
- GT
- Guatemala
- Prior art keywords
- new procedure
- pirazolopirimidinonas
- preparation
- alquilpiperazinil
- pirimidin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
- C07D295/26—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/70—Sulfur atoms
- C07D213/71—Sulfur atoms to which a second hetero atom is attached
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Reproductive Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
ESTA INVENCION SE REFIERE A UN NUEVO PROCEDIMIENTO PARA LA PRODUCCIÓN DE DERIVADOS DE 4-ALQUILPIPERAZINIL-SULFONILFENIL- Y 4-ALQUILPIPERAZINIL-SULFONIL-PIRIDINIL-DIHIDROPIRAZOLO[4,3D]PIRIMIDIN-7-ONA Y EN PARTICULAR EL FARMACO ANTIIMPOTENCIA SILDENAFILO Y SUS ANÁLOGOS. EL SIDENAFILO (5-[2-ETOXI-5-(4-METILPIPERAZIN-1-ILSULFONIL)FENIL]-1-METIL-3-N-PROPIL-1,6-DIHIDRO-7H-PIRAZOLO[4,3-D]PIRIMIDIN-7-ONA) QUE ES EL INGREDIENTE ACTIVO EN EL VIAGRA.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0015462A GB0015462D0 (en) | 2000-06-22 | 2000-06-22 | Novel process for the preparation of pyrazolopyrimidinones |
GB0105878A GB0105878D0 (en) | 2001-03-09 | 2001-03-09 | Novel process for the preparation of pyrazoloprimidinones |
Publications (1)
Publication Number | Publication Date |
---|---|
GT200100113AA true GT200100113AA (es) | 2006-04-10 |
Family
ID=26244537
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT200100113AK GT200100113AA (es) | 2000-06-22 | 2001-06-14 | Nuevo procedimiento para la preparacion de pirazolopirimidinonas . |
GT200100113A GT200100113A (es) | 2000-06-22 | 2001-06-14 | Nuevo procedimiento para la preparacion de pirazolopirimidinonas |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GT200100113A GT200100113A (es) | 2000-06-22 | 2001-06-14 | Nuevo procedimiento para la preparacion de pirazolopirimidinonas |
Country Status (26)
Country | Link |
---|---|
EP (1) | EP1296983B1 (es) |
JP (1) | JP2004501154A (es) |
KR (1) | KR100525699B1 (es) |
AP (1) | AP2001002195A0 (es) |
AR (1) | AR028729A1 (es) |
AT (1) | ATE282619T1 (es) |
AU (2) | AU6259201A (es) |
BR (1) | BR0111864A (es) |
CA (1) | CA2411957C (es) |
CZ (1) | CZ20024130A3 (es) |
DE (1) | DE60107248T2 (es) |
ES (1) | ES2231498T3 (es) |
GT (2) | GT200100113AA (es) |
HK (1) | HK1079198A1 (es) |
HU (1) | HUP0301207A3 (es) |
IL (1) | IL152983A0 (es) |
MX (1) | MXPA02012887A (es) |
MY (1) | MY127737A (es) |
PA (1) | PA8520001A1 (es) |
PE (1) | PE20020091A1 (es) |
PL (1) | PL360299A1 (es) |
PT (1) | PT1296983E (es) |
SV (1) | SV2002000502A (es) |
TN (1) | TNSN01092A1 (es) |
WO (1) | WO2001098303A1 (es) |
YU (1) | YU84702A (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2310144B1 (es) | 2007-06-15 | 2010-01-12 | Galenicum Health, S.L. | Intermedios para la preparacion de un inhibidor de la fosfodiesterasa tipo 5. |
TW201221505A (en) | 2010-07-05 | 2012-06-01 | Sanofi Sa | Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9013750D0 (en) * | 1990-06-20 | 1990-08-08 | Pfizer Ltd | Therapeutic agents |
GB9612514D0 (en) * | 1996-06-14 | 1996-08-14 | Pfizer Ltd | Novel process |
US6087368A (en) * | 1998-06-08 | 2000-07-11 | Bristol-Myers Squibb Company | Quinazolinone inhibitors of cGMP phosphodiesterase |
DE69911448T2 (de) * | 1998-10-23 | 2004-04-08 | Pfizer Inc. | Pyrazolopyrimidinone, cgmp pde5 inhibitoren, zur behandlung von sexuellen funktionsstörungen |
-
2001
- 2001-06-07 PL PL36029901A patent/PL360299A1/xx not_active Application Discontinuation
- 2001-06-07 DE DE60107248T patent/DE60107248T2/de not_active Expired - Fee Related
- 2001-06-07 CZ CZ20024130A patent/CZ20024130A3/cs unknown
- 2001-06-07 EP EP01936729A patent/EP1296983B1/en not_active Expired - Lifetime
- 2001-06-07 BR BR0111864-1A patent/BR0111864A/pt not_active IP Right Cessation
- 2001-06-07 HU HU0301207A patent/HUP0301207A3/hu unknown
- 2001-06-07 CA CA002411957A patent/CA2411957C/en not_active Expired - Fee Related
- 2001-06-07 KR KR10-2002-7017475A patent/KR100525699B1/ko not_active IP Right Cessation
- 2001-06-07 YU YU84702A patent/YU84702A/sh unknown
- 2001-06-07 AU AU6259201A patent/AU6259201A/xx active Pending
- 2001-06-07 JP JP2002504259A patent/JP2004501154A/ja not_active Ceased
- 2001-06-07 IL IL15298301A patent/IL152983A0/xx unknown
- 2001-06-07 WO PCT/IB2001/001038 patent/WO2001098303A1/en not_active Application Discontinuation
- 2001-06-07 ES ES01936729T patent/ES2231498T3/es not_active Expired - Lifetime
- 2001-06-07 AP APAP/P/2001/002195A patent/AP2001002195A0/en unknown
- 2001-06-07 PT PT01936729T patent/PT1296983E/pt unknown
- 2001-06-07 AT AT01936729T patent/ATE282619T1/de not_active IP Right Cessation
- 2001-06-07 AU AU2001262592A patent/AU2001262592B2/en not_active Ceased
- 2001-06-07 MX MXPA02012887A patent/MXPA02012887A/es active IP Right Grant
- 2001-06-14 GT GT200100113AK patent/GT200100113AA/es unknown
- 2001-06-14 GT GT200100113A patent/GT200100113A/es unknown
- 2001-06-15 AR ARP010102878A patent/AR028729A1/es unknown
- 2001-06-18 PE PE2001000586A patent/PE20020091A1/es not_active Application Discontinuation
- 2001-06-19 MY MYPI20012890A patent/MY127737A/en unknown
- 2001-06-19 PA PA20018520001A patent/PA8520001A1/es unknown
- 2001-06-21 SV SV2001000502A patent/SV2002000502A/es not_active Application Discontinuation
- 2001-06-21 TN TNTNSN01092A patent/TNSN01092A1/fr unknown
-
2005
- 2005-12-06 HK HK05111131A patent/HK1079198A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
JP2004501154A (ja) | 2004-01-15 |
KR100525699B1 (ko) | 2005-11-03 |
GT200100113A (es) | 2002-06-04 |
YU84702A (sh) | 2005-09-19 |
TNSN01092A1 (fr) | 2005-11-10 |
AU6259201A (en) | 2002-01-02 |
PA8520001A1 (es) | 2003-09-05 |
CA2411957A1 (en) | 2001-12-27 |
KR20030017556A (ko) | 2003-03-03 |
IL152983A0 (en) | 2003-06-24 |
DE60107248T2 (de) | 2005-12-01 |
CA2411957C (en) | 2007-09-18 |
DE60107248D1 (de) | 2004-12-23 |
PL360299A1 (en) | 2004-09-06 |
ATE282619T1 (de) | 2004-12-15 |
PT1296983E (pt) | 2005-02-28 |
SV2002000502A (es) | 2002-07-03 |
EP1296983A1 (en) | 2003-04-02 |
PE20020091A1 (es) | 2002-02-21 |
ES2231498T3 (es) | 2005-05-16 |
CZ20024130A3 (cs) | 2004-01-14 |
MY127737A (en) | 2006-12-29 |
EP1296983B1 (en) | 2004-11-17 |
AP2001002195A0 (en) | 2002-12-21 |
HK1079198A1 (en) | 2006-03-31 |
MXPA02012887A (es) | 2003-05-14 |
AU2001262592B2 (en) | 2006-07-06 |
WO2001098303A1 (en) | 2001-12-27 |
BR0111864A (pt) | 2003-07-01 |
HUP0301207A3 (en) | 2006-02-28 |
HUP0301207A2 (hu) | 2003-08-28 |
AR028729A1 (es) | 2003-05-21 |
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