GB201218864D0 - Bicyclic heterocycle compounds and their uses in therapy - Google Patents

Bicyclic heterocycle compounds and their uses in therapy

Info

Publication number
GB201218864D0
GB201218864D0 GBGB1218864.5A GB201218864A GB201218864D0 GB 201218864 D0 GB201218864 D0 GB 201218864D0 GB 201218864 A GB201218864 A GB 201218864A GB 201218864 D0 GB201218864 D0 GB 201218864D0
Authority
GB
United Kingdom
Prior art keywords
therapy
bicyclic heterocycle
heterocycle compounds
compounds
bicyclic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
GBGB1218864.5A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Astex Therapeutics Ltd
Original Assignee
Astex Therapeutics Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astex Therapeutics Ltd filed Critical Astex Therapeutics Ltd
Priority to GBGB1218864.5A priority Critical patent/GB201218864D0/en
Publication of GB201218864D0 publication Critical patent/GB201218864D0/en
Priority to CA2888112A priority patent/CA2888112C/en
Priority to US14/436,364 priority patent/US9663512B2/en
Priority to KR1020157012697A priority patent/KR102299832B1/ko
Priority to PCT/GB2013/052721 priority patent/WO2014060768A1/en
Priority to CN201380066425.6A priority patent/CN104870440B/zh
Priority to JP2015537355A priority patent/JP6324976B2/ja
Priority to DK13780388.8T priority patent/DK2909197T3/da
Priority to ES13780388T priority patent/ES2794009T3/es
Priority to EP13780388.8A priority patent/EP2909197B1/en
Priority to US15/411,463 priority patent/US9980973B2/en
Ceased legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epidemiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
GBGB1218864.5A 2012-10-19 2012-10-19 Bicyclic heterocycle compounds and their uses in therapy Ceased GB201218864D0 (en)

Priority Applications (11)

Application Number Priority Date Filing Date Title
GBGB1218864.5A GB201218864D0 (en) 2012-10-19 2012-10-19 Bicyclic heterocycle compounds and their uses in therapy
EP13780388.8A EP2909197B1 (en) 2012-10-19 2013-10-18 Bicyclic heterocycle compounds and their uses in therapy
PCT/GB2013/052721 WO2014060768A1 (en) 2012-10-19 2013-10-18 Bicyclic heterocycle compounds and their uses in therapy
US14/436,364 US9663512B2 (en) 2012-10-19 2013-10-18 Bicyclic heterocycle compounds and their uses in therapy
KR1020157012697A KR102299832B1 (ko) 2012-10-19 2013-10-18 바이사이클릭 헤테로사이클 화합물 및 치료에서의 그것의 용도
CA2888112A CA2888112C (en) 2012-10-19 2013-10-18 Bicyclic heterocycle compounds and their uses in therapy
CN201380066425.6A CN104870440B (zh) 2012-10-19 2013-10-18 双环杂环化合物及其治疗用途
JP2015537355A JP6324976B2 (ja) 2012-10-19 2013-10-18 二環式複素環化合物およびそれらの治療での使用
DK13780388.8T DK2909197T3 (da) 2012-10-19 2013-10-18 Bicykliske heterocykliske forbindelser og anvendelser deraf ved terapi
ES13780388T ES2794009T3 (es) 2012-10-19 2013-10-18 Compuestos heterocíclicos bicíclicos y sus usos en terapia
US15/411,463 US9980973B2 (en) 2012-10-19 2017-01-20 Bicyclic heterocycle compounds and their uses in therapy

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB1218864.5A GB201218864D0 (en) 2012-10-19 2012-10-19 Bicyclic heterocycle compounds and their uses in therapy

Publications (1)

Publication Number Publication Date
GB201218864D0 true GB201218864D0 (en) 2012-12-05

Family

ID=47359191

Family Applications (1)

Application Number Title Priority Date Filing Date
GBGB1218864.5A Ceased GB201218864D0 (en) 2012-10-19 2012-10-19 Bicyclic heterocycle compounds and their uses in therapy

Country Status (10)

Country Link
US (1) US9663512B2 (https=)
EP (1) EP2909197B1 (https=)
JP (1) JP6324976B2 (https=)
KR (1) KR102299832B1 (https=)
CN (1) CN104870440B (https=)
CA (1) CA2888112C (https=)
DK (1) DK2909197T3 (https=)
ES (1) ES2794009T3 (https=)
GB (1) GB201218864D0 (https=)
WO (1) WO2014060768A1 (https=)

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GB201106817D0 (en) 2011-04-21 2011-06-01 Astex Therapeutics Ltd New compound
GB201106814D0 (en) 2011-04-21 2011-06-01 Astex Therapeutics Ltd New compounds
US9980973B2 (en) 2012-10-19 2018-05-29 Astex Therapeutics Limited Bicyclic heterocycle compounds and their uses in therapy
GB201218862D0 (en) 2012-10-19 2012-12-05 Astex Therapeutics Ltd Bicyclic heterocycle compounds and their uses in therapy
GB201218850D0 (en) 2012-10-19 2012-12-05 Astex Therapeutics Ltd Bicyclic heterocycle compounds and their uses in therapy
GB201218864D0 (en) 2012-10-19 2012-12-05 Astex Therapeutics Ltd Bicyclic heterocycle compounds and their uses in therapy
BR122022015241B1 (pt) 2013-12-20 2023-09-26 Astex Therapeutics Limited Compostos heterocíclicos bicíclicos intermediários para a preparação de um composto de fórmula (i)
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EP3999182A1 (en) 2019-07-17 2022-05-25 Arvinas Operations, Inc. Tau-protein targeting compounds and associated methods of use
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WO2024240858A1 (en) 2023-05-23 2024-11-28 Valerio Therapeutics Protac molecules directed against dna damage repair system and uses thereof

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GB201218850D0 (en) 2012-10-19 2012-12-05 Astex Therapeutics Ltd Bicyclic heterocycle compounds and their uses in therapy
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Also Published As

Publication number Publication date
JP2015534975A (ja) 2015-12-07
US20150266873A1 (en) 2015-09-24
US9663512B2 (en) 2017-05-30
CA2888112A1 (en) 2014-04-24
EP2909197A1 (en) 2015-08-26
ES2794009T3 (es) 2020-11-17
DK2909197T3 (da) 2020-05-25
CN104870440A (zh) 2015-08-26
JP6324976B2 (ja) 2018-05-16
CA2888112C (en) 2021-03-30
WO2014060768A1 (en) 2014-04-24
EP2909197B1 (en) 2020-03-04
KR20150072436A (ko) 2015-06-29
CN104870440B (zh) 2018-10-19
KR102299832B1 (ko) 2021-09-07

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Legal Events

Date Code Title Description
AT Applications terminated before publication under section 16(1)