GB1447329A - Preparation of sulphonyl-benzamide derivatives - Google Patents

Preparation of sulphonyl-benzamide derivatives

Info

Publication number
GB1447329A
GB1447329A GB4131474A GB4131474A GB1447329A GB 1447329 A GB1447329 A GB 1447329A GB 4131474 A GB4131474 A GB 4131474A GB 4131474 A GB4131474 A GB 4131474A GB 1447329 A GB1447329 A GB 1447329A
Authority
GB
United Kingdom
Prior art keywords
radical
alkyl
formula
preparation
monoalkylamino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB4131474A
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
DETEUDES SCINTIFIQUES ET IND D
Original Assignee
DETEUDES SCINTIFIQUES ET IND D
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by DETEUDES SCINTIFIQUES ET IND D filed Critical DETEUDES SCINTIFIQUES ET IND D
Publication of GB1447329A publication Critical patent/GB1447329A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical

Abstract

1447329 Preparation of sulphonyl benzamide derivatives SOC D'ETUDES SCIENTIFIQUES ET INDUSTRIELLES DE L'ILE - DEFRANCE 23 Sept 1974 [28 Sept 1973] 41314/74 Heading C2C A method of preparing 2,5-disubstituted benzamides having the general formula in which A is a C 1 to C 5 monoalkylamino or di- (C 1 to C 5 alkyl) amino radical, a nitrogen attached saturated heterocyclic ring optionally containing an oxygen, sulphur or second nitrogen atom, the second nitrogen atom optionally having a C 1 to C 5 alkyl substituent attached to it, or a heterocyclic radical having the formula in which R is a C 1 to C 5 alkyl radical or an alkenyl radical and m is 1, 2, 3 or 4, B is a C 1 to C 5 alkyl radical or an alkenyl radical; n is 1 or 2 and X is an amino, monoalkylamino, dialkylamino, alkyl or alkenyl radical, comprises heating a 2,5-disubstituted benzoic acid having the formula in which B and X are as above with an amine having the formula H 2 N(CH 2 ) n A in which A and n are as above, in the presence of phosphoric anhydride. The benzamides so prepared may be converted into an acid-addition salt.
GB4131474A 1973-09-28 1974-09-23 Preparation of sulphonyl-benzamide derivatives Expired GB1447329A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7335095A FR2245628B1 (en) 1973-09-28 1973-09-28

Publications (1)

Publication Number Publication Date
GB1447329A true GB1447329A (en) 1976-08-25

Family

ID=9125782

Family Applications (1)

Application Number Title Priority Date Filing Date
GB4131474A Expired GB1447329A (en) 1973-09-28 1974-09-23 Preparation of sulphonyl-benzamide derivatives

Country Status (11)

Country Link
JP (1) JPS5715752B2 (en)
AR (1) AR205172A1 (en)
AT (1) AT338235B (en)
CA (1) CA1055502A (en)
CY (1) CY974A (en)
DE (1) DE2444587A1 (en)
ES (1) ES430341A1 (en)
FI (1) FI59087C (en)
FR (1) FR2245628B1 (en)
GB (1) GB1447329A (en)
IE (1) IE40402B1 (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003055857A1 (en) * 2001-12-28 2003-07-10 Farmaceutsko-Hemijska Industrija 'zdravlje' A process for synthesis of heterocyclic aminoalkyl benzamides

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2418225A1 (en) * 1978-02-27 1979-09-21 Synthelabo N-1-Cycloalkyl-2-pyrrolidinyl-methyl 2-methoxy-benzamide derivs. - for treating psychoses and depressive states, prepd. by reaction of 1-cycloalkyl-2-aminomethyl-pyrrolidine with methoxy-benzoic acid deriv.
FR2418226A1 (en) * 1978-02-27 1979-09-21 Synthelabo METHOXY-2 ALKYLTHIO-5 BENZAMIDES AND THEIR THERAPEUTIC APPLICATION
FR2447910A2 (en) * 1979-02-05 1980-08-29 Synthelabo Neuroleptics used to treat psychoses and depression - are N 1-cycloalkyl-alkyl-2-pyrrolidinyl-methyl 2-methoxy 5-alkylthio-benzamide derivs.
FR2478093A1 (en) * 1980-03-12 1981-09-18 Ile De France Prepn. of N-pyrrolidinyl methyl-2-methoxy-5-sulphamoyl benzamide cpds. - from 2-methoxy-5- chlorosulphonyl-benzoic acid cpds.

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003055857A1 (en) * 2001-12-28 2003-07-10 Farmaceutsko-Hemijska Industrija 'zdravlje' A process for synthesis of heterocyclic aminoalkyl benzamides

Also Published As

Publication number Publication date
FR2245628B1 (en) 1977-03-11
JPS5059350A (en) 1975-05-22
AT338235B (en) 1977-08-10
AR205172A1 (en) 1976-04-12
DE2444587A1 (en) 1975-04-03
FI59087B (en) 1981-02-27
ES430341A1 (en) 1977-05-01
CY974A (en) 1978-12-22
JPS5715752B2 (en) 1982-04-01
IE40402L (en) 1975-03-28
CA1055502A (en) 1979-05-29
FI59087C (en) 1981-06-10
IE40402B1 (en) 1979-05-23
FI276274A (en) 1975-03-29
ATA770474A (en) 1976-12-15
FR2245628A1 (en) 1975-04-25

Similar Documents

Publication Publication Date Title
GB1466646A (en) Substituted benzamides
GB1369248A (en) Amides the preparation thereof and their use in pharmacjeutical compositions
GB1461185A (en) Preparation of sulphonyl-benzamide derivatives
IL72166A (en) Beta-carboline dicarboxylic acid derivatives and pharmaceutical compositions containing the same
GB1447329A (en) Preparation of sulphonyl-benzamide derivatives
SE7606424L (en) SUBSTITUTED BENZAMIDS
GB1455595A (en) Preparation of 2,5-disubstituted benzamides
GB1394563A (en) Process for preparing benzamides
GB1466822A (en) Substituted benzamides
IE39925L (en) Preparation of sulphonyl and sulphamyl-benzamide derivatives
GB1474039A (en) Preparation of 2-alkoxy-5-sulphamoylbenzoic acids
GB1419733A (en) Benzamide derivative
GB1184047A (en) Process for Preparing Derivatives of N-substituted Benzamides
IE38948L (en) Preparation of 2, 5-disubstituted benzamides
IE38930L (en) Sulphonylbenzamide derivatives
GB1383269A (en) Preparation of n-tertiary aminoalkyl-2-alkoxy benzamides and benzoic anhydride derivatives produced during it
GB1146333A (en) 4-amino-5-halo-2-substituted benzamide derivatives
IE38928L (en) Sulphonylbenzamide derivatives
IE38925L (en) Sulphonylbenzamide derivatives
GB1455522A (en) Benzopyrano-3,4-c pyridines
GB1415421A (en) Preparation of benzamides
ES344072A1 (en) Basically substituted 2-imidazolidone derivatives and their production
GB1492236A (en) Di-hydroethanoanthracene derivatives
GB1420897A (en) Preparation of 2,5-disubstituted benzamides
GB1501771A (en) Preparation of benzenesulphonamides

Legal Events

Date Code Title Description
PS Patent sealed
PCNP Patent ceased through non-payment of renewal fee

Effective date: 19920923