GB1416872A - 4-aminoquinoline derivatives - Google Patents

4-aminoquinoline derivatives

Info

Publication number
GB1416872A
GB1416872A GB553173A GB553173A GB1416872A GB 1416872 A GB1416872 A GB 1416872A GB 553173 A GB553173 A GB 553173A GB 553173 A GB553173 A GB 553173A GB 1416872 A GB1416872 A GB 1416872A
Authority
GB
United Kingdom
Prior art keywords
alkyl
benzyl
compounds
derivatives
iiia
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB553173A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
John Wyeth and Brother Ltd
Original Assignee
John Wyeth and Brother Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by John Wyeth and Brother Ltd filed Critical John Wyeth and Brother Ltd
Priority to GB553173A priority Critical patent/GB1416872A/en
Priority to AU52421/73A priority patent/AU467944B2/en
Priority to CH270476A priority patent/CH576964A5/xx
Priority to CH343873A priority patent/CH577476A5/xx
Priority to DE2311570A priority patent/DE2311570C2/de
Priority to JP48027544A priority patent/JPS604187B2/ja
Priority to FR7308625A priority patent/FR2181807B1/fr
Priority to US05/543,217 priority patent/US3971787A/en
Priority to US05/543,218 priority patent/US3971789A/en
Publication of GB1416872A publication Critical patent/GB1416872A/en
Priority to BE178465A priority patent/BE855713Q/xx
Priority to KE2916A priority patent/KE2916A/xx
Priority to HK102/79A priority patent/HK10279A/xx
Priority to MY1979137A priority patent/MY7900137A/xx
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4
    • C07D215/44—Nitrogen atoms attached in position 4 with aryl radicals attached to said nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Transplantation (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
GB553173A 1972-03-10 1973-02-05 4-aminoquinoline derivatives Expired GB1416872A (en)

Priority Applications (13)

Application Number Priority Date Filing Date Title
GB553173A GB1416872A (en) 1972-03-10 1973-02-05 4-aminoquinoline derivatives
AU52421/73A AU467944B2 (en) 1972-03-10 1973-02-21 4-aminoquinoline derivatives
CH270476A CH576964A5 (enrdf_load_stackoverflow) 1972-03-10 1973-03-08
CH343873A CH577476A5 (enrdf_load_stackoverflow) 1972-03-10 1973-03-08
DE2311570A DE2311570C2 (de) 1972-03-10 1973-03-08 4-Aminochinoline, Verfahren zu ihrer Herstellung und sie enthaltende pharmazeutische Zubereitungen
JP48027544A JPS604187B2 (ja) 1972-03-10 1973-03-08 ４−アミノキノリン誘導体の製造方法
FR7308625A FR2181807B1 (enrdf_load_stackoverflow) 1972-03-10 1973-03-09
US05/543,217 US3971787A (en) 1973-02-05 1975-01-23 (4-Quinolylamino)benzamides
US05/543,218 US3971789A (en) 1972-10-21 1975-01-23 O-(4-Quinolylamino)benzamides
BE178465A BE855713Q (fr) 1972-03-10 1977-06-15 Nouveaux derives de 4-aminoquinoleine, leur procede de preparation et medicament les contenant
KE2916A KE2916A (en) 1972-03-10 1979-01-29 4-aminoquinoline derivatives
HK102/79A HK10279A (en) 1972-03-10 1979-03-01 4-aminoquinoline derivatives
MY1979137A MY7900137A (en) 1972-03-10 1979-12-31 4-aminoquinoline derivatives

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB1125172 1972-03-10
GB3063572 1972-06-30
GB4859372 1972-10-21
GB553173A GB1416872A (en) 1972-03-10 1973-02-05 4-aminoquinoline derivatives

Publications (1)

Publication Number Publication Date
GB1416872A true GB1416872A (en) 1975-12-10

Family

ID=27447454

Family Applications (1)

Application Number Title Priority Date Filing Date
GB553173A Expired GB1416872A (en) 1972-03-10 1973-02-05 4-aminoquinoline derivatives

Country Status (10)

Country Link
JP (1) JPS604187B2 (enrdf_load_stackoverflow)
AU (1) AU467944B2 (enrdf_load_stackoverflow)
BE (1) BE855713Q (enrdf_load_stackoverflow)
CH (2) CH576964A5 (enrdf_load_stackoverflow)
DE (1) DE2311570C2 (enrdf_load_stackoverflow)
FR (1) FR2181807B1 (enrdf_load_stackoverflow)
GB (1) GB1416872A (enrdf_load_stackoverflow)
HK (1) HK10279A (enrdf_load_stackoverflow)
KE (1) KE2916A (enrdf_load_stackoverflow)
MY (1) MY7900137A (enrdf_load_stackoverflow)

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0001175A1 (en) * 1977-09-14 1979-03-21 JOHN WYETH & BROTHER LIMITED 4-Aminoquinoline derivatives, a process for their preparation and pharmaceutical compositions containing them
US4735952A (en) * 1985-02-11 1988-04-05 Fujisawa Pharmaceutical Co., Ltd. Arylthio piperidinamide of (4-quinolinylamino)benzoic acid and S-oxidized derivatives
WO2001060821A1 (en) * 2000-02-18 2001-08-23 Astrazeneca Ab Novel biarylcarboxamides
US7803825B2 (en) 2007-07-16 2010-09-28 Wyeth Llc Aminoalkylazole derivatives as histamine-3 antagonists
US7820825B2 (en) 2006-03-15 2010-10-26 Wyeth Llc N-substituted-azacyclylamines as histamine-3 antagonists
US7935719B2 (en) 2006-10-06 2011-05-03 Wyeth Llc N-substituted-azacyclylamines as histamine-3 antagonists
EP2050735A4 (en) * 2006-07-28 2011-12-21 Kaneka Corp METHOD FOR PRODUCING AN OPTICALLY ACTIVE 3-AMINO-NITROGENATED COMPOUND
US8430132B2 (en) 2007-02-01 2013-04-30 Hobart Brothers Company Air hose delivery assemblies

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA743270B (en) * 1973-06-15 1975-05-28 Upjohn Co Anti-hypertensive compounds
GB1474296A (en) * 1975-01-23 1977-05-18 Wyeth John & Brother Ltd 4-aminoquinoline derivatives
JPS5717907Y2 (enrdf_load_stackoverflow) * 1977-09-05 1982-04-14
JPS6055170A (ja) * 1983-09-05 1985-03-30 株式会社多川工業 鉄骨切断装置
FI95572C (fi) 1987-06-22 1996-02-26 Eisai Co Ltd Menetelmä lääkeaineena käyttökelpoisen piperidiinijohdannaisten tai sen farmaseuttisen suolan valmistamiseksi
AU674207B2 (en) * 1993-04-07 1996-12-12 Otsuka Pharmaceutical Co., Ltd. N-acylated 4-amino piperidine derivatives
US5567718A (en) * 1994-08-11 1996-10-22 Hoechst Marion Roussel Inc. 2,3-dihydro-1h-isoindole derivatives and their use as serotonin reuptake inhibitors
AUPP818099A0 (en) * 1999-01-14 1999-02-11 Fujisawa Pharmaceutical Co., Ltd. New n-containing heterocyclic compounds
MY142362A (en) 2004-01-29 2010-11-30 Otsuka Pharma Co Ltd Pharmaceutical composition for promoting angiogenesis
PE20080371A1 (es) * 2006-05-19 2008-04-09 Wyeth Corp N-benzoil-y-n-bencilpirrolidin-3-ilaminas como antagonistas de histamina-3

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA731646A (en) * 1962-05-08 1966-04-05 Roussel-Uclaf 4-(2'(.beta.-MORPHOLYLETHOXYCARBONYL) PHENYLAMINE) 7-CHLORO QUINOLEINE ET SES SELS, AINSI QUE LEUR PROCEDE DE PREPARATION
BE754587A (fr) * 1969-08-08 1971-02-08 Upjohn Co Nouveaux p-(trihalomethylquinolylamino) benzamides et leur procede de preparation
BE754586A (fr) * 1969-08-08 1971-02-08 Upjohn Co Preparations pharmaceutiques a base de p-(4-quinolylamino) benzamide etleur utilisation

Cited By (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0001175A1 (en) * 1977-09-14 1979-03-21 JOHN WYETH & BROTHER LIMITED 4-Aminoquinoline derivatives, a process for their preparation and pharmaceutical compositions containing them
US4735952A (en) * 1985-02-11 1988-04-05 Fujisawa Pharmaceutical Co., Ltd. Arylthio piperidinamide of (4-quinolinylamino)benzoic acid and S-oxidized derivatives
WO2001060821A1 (en) * 2000-02-18 2001-08-23 Astrazeneca Ab Novel biarylcarboxamides
US7001914B2 (en) 2000-02-18 2006-02-21 Astrazeneca Ab Compounds
US7214688B2 (en) 2000-02-18 2007-05-08 Astrazeneca Ab Compounds
US7491734B2 (en) 2000-02-18 2009-02-17 Astrazeneca Ab 2-(pyridine-4-yl)-N-(quinuclidin-2-yl)thiazole-4-carboxide nicotinic acetylcholine receptor ligands
US7820825B2 (en) 2006-03-15 2010-10-26 Wyeth Llc N-substituted-azacyclylamines as histamine-3 antagonists
EP2050735A4 (en) * 2006-07-28 2011-12-21 Kaneka Corp METHOD FOR PRODUCING AN OPTICALLY ACTIVE 3-AMINO-NITROGENATED COMPOUND
US7935719B2 (en) 2006-10-06 2011-05-03 Wyeth Llc N-substituted-azacyclylamines as histamine-3 antagonists
US8430132B2 (en) 2007-02-01 2013-04-30 Hobart Brothers Company Air hose delivery assemblies
US7803825B2 (en) 2007-07-16 2010-09-28 Wyeth Llc Aminoalkylazole derivatives as histamine-3 antagonists

Also Published As

Publication number Publication date
KE2916A (en) 1979-03-30
DE2311570C2 (de) 1986-03-13
DE2311570A1 (de) 1973-09-13
HK10279A (en) 1979-03-09
FR2181807A1 (enrdf_load_stackoverflow) 1973-12-07
CH576964A5 (enrdf_load_stackoverflow) 1976-06-30
FR2181807B1 (enrdf_load_stackoverflow) 1976-10-22
AU5242173A (en) 1974-10-17
JPS49273A (enrdf_load_stackoverflow) 1974-01-05
AU467944B2 (en) 1975-12-18
MY7900137A (en) 1979-12-31
BE855713Q (fr) 1977-10-03
CH577476A5 (enrdf_load_stackoverflow) 1976-07-15
JPS604187B2 (ja) 1985-02-01

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Legal Events

Date Code Title Description
PS Patent sealed
PCNP Patent ceased through non-payment of renewal fee