GB1260465A - 11beta-CHLORO-19-NOR-STEROIDS - Google Patents
11beta-CHLORO-19-NOR-STEROIDSInfo
- Publication number
- GB1260465A GB1260465A GB4570/68A GB457068A GB1260465A GB 1260465 A GB1260465 A GB 1260465A GB 4570/68 A GB4570/68 A GB 4570/68A GB 457068 A GB457068 A GB 457068A GB 1260465 A GB1260465 A GB 1260465A
- Authority
- GB
- United Kingdom
- Prior art keywords
- pyrazolino
- steroids
- chloro
- activity
- methylene
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 239000000203 mixture Substances 0.000 abstract 3
- 230000003054 hormonal effect Effects 0.000 abstract 2
- -1 16, 17-methylene Chemical group 0.000 abstract 1
- 239000004593 Epoxy Substances 0.000 abstract 1
- BFPYWIDHMRZLRN-SLHNCBLASA-N Ethinyl estradiol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 BFPYWIDHMRZLRN-SLHNCBLASA-N 0.000 abstract 1
- 125000004423 acyloxy group Chemical group 0.000 abstract 1
- 230000002280 anti-androgenic effect Effects 0.000 abstract 1
- 230000001833 anti-estrogenic effect Effects 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 239000011203 carbon fibre reinforced carbon Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229940124558 contraceptive agent Drugs 0.000 abstract 1
- 239000003433 contraceptive agent Substances 0.000 abstract 1
- 125000003700 epoxy group Chemical group 0.000 abstract 1
- 229940011871 estrogen Drugs 0.000 abstract 1
- 239000000262 estrogen Substances 0.000 abstract 1
- 229960002568 ethinylestradiol Drugs 0.000 abstract 1
- 125000001570 methylene group Chemical group [H]C([H])([*:1])[*:2] 0.000 abstract 1
- 239000007935 oral tablet Substances 0.000 abstract 1
- 230000001072 progestational effect Effects 0.000 abstract 1
- 150000003431 steroids Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
- C07J7/0005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21
- C07J7/001—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group
- C07J7/0015—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group not substituted in position 17 alfa
- C07J7/0025—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group not substituted in position 17 alfa substituted in position 16
- C07J7/0035—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group not substituted in position 17 alfa substituted in position 16 by a hydroxy group free esterified or etherified
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
- C07J13/005—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 16 (17)
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
- C07J53/002—Carbocyclic rings fused
- C07J53/004—3 membered carbocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
- C07J7/0005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21
- C07J7/001—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group
- C07J7/004—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa
- C07J7/005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa substituted in position 16
- C07J7/0055—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0036—Nitrogen-containing hetero ring
- C07J71/0057—Nitrogen and oxygen
- C07J71/0068—Nitrogen and oxygen at position 16(17)
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
- C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
- C07J73/003—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by oxygen as hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (19)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB4570/68A GB1260465A (en) | 1968-01-29 | 1968-01-29 | 11beta-CHLORO-19-NOR-STEROIDS |
| IE105/69A IE33924B1 (en) | 1968-01-29 | 1969-01-27 | 11beta -chloro-19-nor-steroids |
| NL6901342A NL6901342A (enrdf_load_stackoverflow) | 1968-01-29 | 1969-01-28 | |
| BR205985/69A BR6905985D0 (pt) | 1968-01-29 | 1969-01-29 | Novo u-beta-cloro-esteroides e processo de sua preparacao |
| DK46569AA DK128715B (da) | 1968-01-29 | 1969-01-29 | 9α-Usubstituerede 11β-klor-19-norpregnaner til anvendelse til svangerskabsforebyggelse. |
| FR6901753A FR2000924A1 (enrdf_load_stackoverflow) | 1968-01-29 | 1969-01-29 | |
| AT91269A AT309703B (de) | 1968-01-29 | 1969-01-29 | Verfahren zur Herstellung von neuen 9α-unsubstituierten 11β-Chlor-19-norsteroiden |
| DE1904325A DE1904325C3 (de) | 1968-01-29 | 1969-01-29 | 9alpha-unsubstituierte 1 lbeta-Chlor-19-norsteroide, Verfahren zu deren Herstellung und diese enthaltende pharmazeutische Zusammensetzungen |
| JP44006062A JPS4828907B1 (enrdf_load_stackoverflow) | 1968-01-29 | 1969-01-29 | |
| CH138669A CH578017A5 (enrdf_load_stackoverflow) | 1968-01-29 | 1969-01-29 | |
| ES363068A ES363068A1 (es) | 1968-01-29 | 1969-01-29 | Un procedimiento para la preparacion de 11-beta-cloro-este-roides. |
| CH45972A CH592688A5 (enrdf_load_stackoverflow) | 1968-01-29 | 1969-01-29 | |
| BE727578D BE727578A (enrdf_load_stackoverflow) | 1968-01-29 | 1969-01-29 | |
| SE01193/69A SE364267B (enrdf_load_stackoverflow) | 1968-01-29 | 1969-01-29 | |
| SE7208742A SE386903B (sv) | 1968-01-29 | 1969-01-29 | Forfarande for framstellning av beta-11-klorsubstituerade steroider tillhorande pregnanserien |
| IL31515A IL31515A0 (en) | 1968-01-29 | 1969-01-30 | New 11beta-cloro-steroids |
| DK218671A DK129042B (da) | 1968-01-29 | 1971-05-06 | Analogifremgangsmåde til fremstilling af 9α-usubstituerede 11β-klor-16-metylen-19-norpregn-4-en-3,20-dioner eller 3-enolætere eller -estere deraf. |
| JP46079507A JPS4830051B1 (enrdf_load_stackoverflow) | 1968-01-29 | 1971-10-11 | |
| AT1109871A AT341117B (de) | 1968-01-29 | 1971-12-23 | Verfahren zur herstellung von neuen 11beta-chlorsteroiden der pregnanreihe |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB4570/68A GB1260465A (en) | 1968-01-29 | 1968-01-29 | 11beta-CHLORO-19-NOR-STEROIDS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1260465A true GB1260465A (en) | 1972-01-19 |
Family
ID=9779640
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB4570/68A Expired GB1260465A (en) | 1968-01-29 | 1968-01-29 | 11beta-CHLORO-19-NOR-STEROIDS |
Country Status (14)
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0866798A4 (en) * | 1995-10-13 | 1998-12-02 | Population Council Inc | PRESENTATION OF ESTER DERIVATIVES OF STEROIDS |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS52119945U (enrdf_load_stackoverflow) * | 1976-03-08 | 1977-09-12 |
-
1968
- 1968-01-29 GB GB4570/68A patent/GB1260465A/en not_active Expired
-
1969
- 1969-01-27 IE IE105/69A patent/IE33924B1/xx unknown
- 1969-01-28 NL NL6901342A patent/NL6901342A/xx not_active Application Discontinuation
- 1969-01-29 CH CH138669A patent/CH578017A5/xx not_active IP Right Cessation
- 1969-01-29 CH CH45972A patent/CH592688A5/xx not_active IP Right Cessation
- 1969-01-29 FR FR6901753A patent/FR2000924A1/fr not_active Withdrawn
- 1969-01-29 BR BR205985/69A patent/BR6905985D0/pt unknown
- 1969-01-29 SE SE7208742A patent/SE386903B/xx unknown
- 1969-01-29 AT AT91269A patent/AT309703B/de not_active IP Right Cessation
- 1969-01-29 DE DE1904325A patent/DE1904325C3/de not_active Expired
- 1969-01-29 JP JP44006062A patent/JPS4828907B1/ja active Pending
- 1969-01-29 DK DK46569AA patent/DK128715B/da unknown
- 1969-01-29 BE BE727578D patent/BE727578A/xx unknown
- 1969-01-29 ES ES363068A patent/ES363068A1/es not_active Expired
- 1969-01-29 SE SE01193/69A patent/SE364267B/xx unknown
- 1969-01-30 IL IL31515A patent/IL31515A0/xx unknown
-
1971
- 1971-10-11 JP JP46079507A patent/JPS4830051B1/ja active Pending
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0866798A4 (en) * | 1995-10-13 | 1998-12-02 | Population Council Inc | PRESENTATION OF ESTER DERIVATIVES OF STEROIDS |
Also Published As
| Publication number | Publication date |
|---|---|
| SE364267B (enrdf_load_stackoverflow) | 1974-02-18 |
| DE1904325A1 (de) | 1969-09-04 |
| DK128715B (da) | 1974-06-24 |
| DE1904325C3 (de) | 1978-10-26 |
| AT309703B (de) | 1973-08-27 |
| IE33924L (en) | 1969-07-29 |
| BR6905985D0 (pt) | 1973-04-19 |
| FR2000924A1 (enrdf_load_stackoverflow) | 1969-09-19 |
| JPS4830051B1 (enrdf_load_stackoverflow) | 1973-09-17 |
| DE1904325B2 (de) | 1978-02-16 |
| SE386903B (sv) | 1976-08-23 |
| IL31515A0 (en) | 1969-03-27 |
| CH592688A5 (enrdf_load_stackoverflow) | 1977-11-15 |
| BE727578A (enrdf_load_stackoverflow) | 1969-07-29 |
| JPS4828907B1 (enrdf_load_stackoverflow) | 1973-09-05 |
| NL6901342A (enrdf_load_stackoverflow) | 1969-07-31 |
| ES363068A1 (es) | 1971-06-16 |
| CH578017A5 (enrdf_load_stackoverflow) | 1976-07-30 |
| IE33924B1 (en) | 1974-12-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PS | Patent sealed [section 19, patents act 1949] | ||
| 426 | Order made revoking patent and granting patent of addition in lieu thereof (sect. 26(2)/1949) | ||
| SP | Amendment (slips) printed | ||
| PCNP | Patent ceased through non-payment of renewal fee |