GB1128234A - 5-benzylpyrimidine derivatives and process for the preparation thereof - Google Patents
5-benzylpyrimidine derivatives and process for the preparation thereofInfo
- Publication number
- GB1128234A GB1128234A GB737666A GB737666A GB1128234A GB 1128234 A GB1128234 A GB 1128234A GB 737666 A GB737666 A GB 737666A GB 737666 A GB737666 A GB 737666A GB 1128234 A GB1128234 A GB 1128234A
- Authority
- GB
- United Kingdom
- Prior art keywords
- group
- benzyl
- hydrogen
- halogen
- hydrogen atom
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
- C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/50—Three nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Lubricants (AREA)
- Liquid Crystal Substances (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Priority Applications (27)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB737666A GB1128234A (en) | 1966-02-19 | 1966-02-19 | 5-benzylpyrimidine derivatives and process for the preparation thereof |
| IL2742467A IL27424A (en) | 1966-02-19 | 1967-02-13 | Method of preparing 5-benzylpyrimidines and novel 5-benzylpyrimidines |
| GR670133641A GR33641B (el) | 1966-02-19 | 1967-02-13 | Χημικαι συνθεσεις και μεθοδος. |
| CA983,015A CA977754A (en) | 1966-02-19 | 1967-02-15 | 2-(3',4',5'-trisubstituted-benzyl) pyrimidine compounds |
| AT153867A AT270653B (de) | 1966-02-19 | 1967-02-16 | Verfahren zur Herstellung von neuen 5-Benzylpyrimidinen |
| NO16687667A NO124601B (US06346242-20020212-C00066.png) | 1966-02-19 | 1967-02-16 | |
| AT409368A AT275534B (de) | 1966-02-19 | 1967-02-16 | Verfahren zur Herstellung von 5-Benzylpyrimidinen |
| DE19671795635 DE1795635C3 (de) | 1966-02-19 | 1967-02-17 | 2,4-Diamino-5-benzyIpyrimidine |
| CH237967A CH511239A (de) | 1966-02-19 | 1967-02-17 | Verfahren zur Herstellung von 5-Benzylpyrimidinen |
| CH191468A CH513179A (de) | 1966-02-19 | 1967-02-17 | Verfahren zur Herstellung von 5-Benzylpyrimidinen |
| BE694244D BE694244A (US06346242-20020212-C00066.png) | 1966-02-19 | 1967-02-17 | |
| NL6702397A NL146811B (nl) | 1966-02-19 | 1967-02-17 | Werkwijze ter bereiding van 5-benzylpyrimidinederivaten. |
| FI48067A FI49714C (fi) | 1966-02-19 | 1967-02-17 | Menetelmä 5-bentsyylipyrimidiinien valmistamiseksi. |
| DE1967W0043385 DE1720012B2 (de) | 1966-02-19 | 1967-02-17 | Verfahren zur herstellung von 2,4-diamino-5-(3,4,5-trimethoxybenzyl)- pyrimidin |
| ES336945A ES336945A1 (es) | 1966-02-19 | 1967-02-17 | Un metodo de preparar 5-bencil-pirimidinas. |
| SE796270A SE390412B (sv) | 1966-02-19 | 1967-02-20 | 2,4-diamino-5-(4'-hydroxybensyl)pyrimidiner till anvendning, som utgangsmaterial for framstellning av 2,4-diamino-5-(3',4',5'-trialikocibensyl)pyrimidiner |
| FR95595A FR1536204A (fr) | 1966-02-19 | 1967-02-20 | Procédé de préparation de dérivés de la pyrimidine |
| SE227867A SE338998B (US06346242-20020212-C00066.png) | 1966-02-19 | 1967-02-20 | |
| DK91167A DK120344B (da) | 1966-02-19 | 1967-02-20 | Fremgangsmåde til fremstilling af 5-benzyl-pyrimidiner. |
| FR106573A FR6595M (US06346242-20020212-C00066.png) | 1966-02-19 | 1967-05-16 | |
| DE19681720031 DE1720031A1 (de) | 1966-02-19 | 1968-02-02 | Biologisch wirksame 5-Benzylpyrimidin-Derivate und Verfahren zu ihrer Herstellung |
| FI26868A FI55031C (fi) | 1966-02-19 | 1968-02-02 | Foerfarande foer framstaellning av antibakteriella 5-bensylpyrimidiner |
| FR138498A FR94837E (fr) | 1966-02-19 | 1968-02-02 | Procédé de préparation de dérivés de la pyrimidine. |
| DK59371A DK128247B (da) | 1966-02-19 | 1971-02-10 | 2,4-Diamino-5-(4'-hydroxybenzyl)-pyrimidiner til anvendelse som udgangsmaterialer ved fremstilling af tilsvarende forbindelser, hvori hydroxygruppens hydrogenatom er substitueret. |
| FI250271A FI55032C (fi) | 1966-02-19 | 1971-09-07 | Som utgaongsmaterial vid framstaellning av antibakteriella 2,4-diamino-5-(3',4',5'-trialkoxibensyl)-pyrimidiner anvaendbara 2,4-diamino-5-(4'-hydroxibensyl)-pyrimidiner |
| NO377771A NO133550C (US06346242-20020212-C00066.png) | 1966-02-19 | 1971-10-13 | |
| MY7100226A MY7100226A (en) | 1966-02-19 | 1971-12-31 | 5-benzylpyrimidine derivatives and process for the preparation thereof |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB737666A GB1128234A (en) | 1966-02-19 | 1966-02-19 | 5-benzylpyrimidine derivatives and process for the preparation thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB1128234A true GB1128234A (en) | 1968-09-25 |
Family
ID=9831956
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB737666A Expired GB1128234A (en) | 1966-02-19 | 1966-02-19 | 5-benzylpyrimidine derivatives and process for the preparation thereof |
Country Status (16)
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2249532A1 (de) * | 1971-10-12 | 1973-04-26 | Wellcome Found | Verfahren zur herstellung von 2,4-diamino-5-benzylpyrimidinen |
| EP0006987A1 (en) * | 1978-05-24 | 1980-01-23 | The Wellcome Foundation Limited | 2,4-Diamino-5-benzylpyrimidines, especially for the treatment of microbial infections, pharmaceutical compositions containing these compounds and processes for preparing these compounds |
| DE2944145A1 (de) | 1979-11-02 | 1981-05-14 | Dynamit Nobel Ag, 5210 Troisdorf | Verfahren zur herstellung von 2,4-diaminopyrimidin |
-
1966
- 1966-02-19 GB GB737666A patent/GB1128234A/en not_active Expired
-
1967
- 1967-02-13 GR GR670133641A patent/GR33641B/el unknown
- 1967-02-13 IL IL2742467A patent/IL27424A/xx unknown
- 1967-02-15 CA CA983,015A patent/CA977754A/en not_active Expired
- 1967-02-16 NO NO16687667A patent/NO124601B/no unknown
- 1967-02-16 AT AT153867A patent/AT270653B/de active
- 1967-02-16 AT AT409368A patent/AT275534B/de active
- 1967-02-17 DE DE19671795635 patent/DE1795635C3/de not_active Expired
- 1967-02-17 CH CH237967A patent/CH511239A/de not_active IP Right Cessation
- 1967-02-17 ES ES336945A patent/ES336945A1/es not_active Expired
- 1967-02-17 NL NL6702397A patent/NL146811B/xx not_active IP Right Cessation
- 1967-02-17 BE BE694244D patent/BE694244A/xx not_active IP Right Cessation
- 1967-02-17 DE DE1967W0043385 patent/DE1720012B2/de active Granted
- 1967-02-17 FI FI48067A patent/FI49714C/fi active
- 1967-02-17 CH CH191468A patent/CH513179A/de not_active IP Right Cessation
- 1967-02-20 SE SE227867A patent/SE338998B/xx unknown
- 1967-02-20 DK DK91167A patent/DK120344B/da not_active IP Right Cessation
- 1967-02-20 SE SE796270A patent/SE390412B/xx unknown
- 1967-05-16 FR FR106573A patent/FR6595M/fr not_active Expired
-
1971
- 1971-02-10 DK DK59371A patent/DK128247B/da not_active IP Right Cessation
- 1971-12-31 MY MY7100226A patent/MY7100226A/xx unknown
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2249532A1 (de) * | 1971-10-12 | 1973-04-26 | Wellcome Found | Verfahren zur herstellung von 2,4-diamino-5-benzylpyrimidinen |
| EP0006987A1 (en) * | 1978-05-24 | 1980-01-23 | The Wellcome Foundation Limited | 2,4-Diamino-5-benzylpyrimidines, especially for the treatment of microbial infections, pharmaceutical compositions containing these compounds and processes for preparing these compounds |
| DE2944145A1 (de) | 1979-11-02 | 1981-05-14 | Dynamit Nobel Ag, 5210 Troisdorf | Verfahren zur herstellung von 2,4-diaminopyrimidin |
Also Published As
| Publication number | Publication date |
|---|---|
| AT270653B (de) | 1969-05-12 |
| DE1795635A1 (de) | 1972-10-19 |
| NL6702397A (US06346242-20020212-C00066.png) | 1967-08-21 |
| BE694244A (US06346242-20020212-C00066.png) | 1967-08-17 |
| SE390412B (sv) | 1976-12-20 |
| AT275534B (de) | 1969-10-27 |
| ES336945A1 (es) | 1968-01-16 |
| DE1795635C3 (de) | 1978-05-11 |
| CH513179A (de) | 1971-09-30 |
| FI49714C (fi) | 1975-09-10 |
| NL146811B (nl) | 1975-08-15 |
| MY7100226A (en) | 1971-12-31 |
| FR6595M (US06346242-20020212-C00066.png) | 1969-01-06 |
| DE1720012B2 (de) | 1977-06-08 |
| NO124601B (US06346242-20020212-C00066.png) | 1972-05-08 |
| GR33641B (el) | 1968-01-03 |
| DE1795635B2 (de) | 1977-09-22 |
| DK128247B (da) | 1974-03-25 |
| SE338998B (US06346242-20020212-C00066.png) | 1971-09-27 |
| DE1720012A1 (de) | 1972-04-06 |
| CH511239A (de) | 1971-08-15 |
| DK120344B (da) | 1971-05-17 |
| FI49714B (US06346242-20020212-C00066.png) | 1975-06-02 |
| IL27424A (en) | 1971-02-25 |
| CA977754A (en) | 1975-11-11 |
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