DK128247B - 2,4-Diamino-5-(4'-hydroxybenzyl)-pyrimidiner til anvendelse som udgangsmaterialer ved fremstilling af tilsvarende forbindelser, hvori hydroxygruppens hydrogenatom er substitueret. - Google Patents

2,4-Diamino-5-(4'-hydroxybenzyl)-pyrimidiner til anvendelse som udgangsmaterialer ved fremstilling af tilsvarende forbindelser, hvori hydroxygruppens hydrogenatom er substitueret.

Info

Publication number
DK128247B
DK128247B DK59371A DK59371A DK128247B DK 128247 B DK128247 B DK 128247B DK 59371 A DK59371 A DK 59371A DK 59371 A DK59371 A DK 59371A DK 128247 B DK128247 B DK 128247B
Authority
DK
Denmark
Prior art keywords
hydroxybenzyl
pyrimidines
diamino
substituted
preparation
Prior art date
Application number
DK59371A
Other languages
English (en)
Inventor
B Roth
J Strelitz
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of DK128247B publication Critical patent/DK128247B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50Three nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52Two oxygen atoms
    • C07D239/54Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Lubricants (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Liquid Crystal Substances (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK59371A 1966-02-19 1971-02-10 2,4-Diamino-5-(4'-hydroxybenzyl)-pyrimidiner til anvendelse som udgangsmaterialer ved fremstilling af tilsvarende forbindelser, hvori hydroxygruppens hydrogenatom er substitueret. DK128247B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB737666A GB1128234A (en) 1966-02-19 1966-02-19 5-benzylpyrimidine derivatives and process for the preparation thereof

Publications (1)

Publication Number Publication Date
DK128247B true DK128247B (da) 1974-03-25

Family

ID=9831956

Family Applications (2)

Application Number Title Priority Date Filing Date
DK91167A DK120344B (da) 1966-02-19 1967-02-20 Fremgangsmåde til fremstilling af 5-benzyl-pyrimidiner.
DK59371A DK128247B (da) 1966-02-19 1971-02-10 2,4-Diamino-5-(4'-hydroxybenzyl)-pyrimidiner til anvendelse som udgangsmaterialer ved fremstilling af tilsvarende forbindelser, hvori hydroxygruppens hydrogenatom er substitueret.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK91167A DK120344B (da) 1966-02-19 1967-02-20 Fremgangsmåde til fremstilling af 5-benzyl-pyrimidiner.

Country Status (16)

Country Link
AT (2) AT275534B (da)
BE (1) BE694244A (da)
CA (1) CA977754A (da)
CH (2) CH513179A (da)
DE (2) DE1795635C3 (da)
DK (2) DK120344B (da)
ES (1) ES336945A1 (da)
FI (1) FI49714C (da)
FR (1) FR6595M (da)
GB (1) GB1128234A (da)
GR (1) GR33641B (da)
IL (1) IL27424A (da)
MY (1) MY7100226A (da)
NL (1) NL146811B (da)
NO (1) NO124601B (da)
SE (2) SE338998B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE789904A (fr) * 1971-10-12 1973-04-10 Wellcome Found Procedes de synthese organique
NO791699L (no) * 1978-05-24 1979-11-27 Wellcome Found Benzylpyrimidinforbindelser og fremgangsmaate til deres fremstilling
DE2944145A1 (de) 1979-11-02 1981-05-14 Dynamit Nobel Ag, 5210 Troisdorf Verfahren zur herstellung von 2,4-diaminopyrimidin

Also Published As

Publication number Publication date
SE338998B (da) 1971-09-27
DE1720012A1 (de) 1972-04-06
NL6702397A (da) 1967-08-21
DE1795635C3 (de) 1978-05-11
FI49714B (da) 1975-06-02
GB1128234A (en) 1968-09-25
MY7100226A (en) 1971-12-31
CA977754A (en) 1975-11-11
NO124601B (da) 1972-05-08
FR6595M (da) 1969-01-06
IL27424A (en) 1971-02-25
GR33641B (el) 1968-01-03
DK120344B (da) 1971-05-17
DE1795635A1 (de) 1972-10-19
CH513179A (de) 1971-09-30
DE1720012B2 (de) 1977-06-08
AT275534B (de) 1969-10-27
NL146811B (nl) 1975-08-15
SE390412B (sv) 1976-12-20
BE694244A (da) 1967-08-17
FI49714C (fi) 1975-09-10
AT270653B (de) 1969-05-12
CH511239A (de) 1971-08-15
ES336945A1 (es) 1968-01-16
DE1795635B2 (de) 1977-09-22

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