GB1081757A - Derivatives of rifamycin o and s - Google Patents

Derivatives of rifamycin o and s

Info

Publication number
GB1081757A
GB1081757A GB41587/64A GB4158764A GB1081757A GB 1081757 A GB1081757 A GB 1081757A GB 41587/64 A GB41587/64 A GB 41587/64A GB 4158764 A GB4158764 A GB 4158764A GB 1081757 A GB1081757 A GB 1081757A
Authority
GB
United Kingdom
Prior art keywords
rifamycin
derivative
formula
tetrahydro
produced
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
GB41587/64A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF Schweiz AG
Gruppo Lepetit SpA
Original Assignee
Ciba AG
Lepetit SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba AG, Lepetit SpA filed Critical Ciba AG
Publication of GB1081757A publication Critical patent/GB1081757A/en
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/20—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/20—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/22—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/20—Spiro-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
GB41587/64A 1963-10-11 1964-10-12 Derivatives of rifamycin o and s Expired GB1081757A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH1254063A CH478139A (de) 1963-10-11 1963-10-11 Verfahren zur Herstellung neuer antibiotisch wirksamer Kondensationsprodukte von Rifamycin O
CH1004564A CH504457A (de) 1963-10-11 1964-07-31 Verfahren zur Herstellung neuer antibiotisch wirksamer Kondensationsprodukte von Rifamycin S
CH1179764 1964-09-10

Publications (1)

Publication Number Publication Date
GB1081757A true GB1081757A (en) 1967-08-31

Family

ID=27176360

Family Applications (1)

Application Number Title Priority Date Filing Date
GB41587/64A Expired GB1081757A (en) 1963-10-11 1964-10-12 Derivatives of rifamycin o and s

Country Status (14)

Country Link
US (1) US3338888A (enExample)
AT (1) AT261805B (enExample)
BE (1) BE654209A (enExample)
BR (1) BR6463319D0 (enExample)
CH (2) CH478139A (enExample)
DE (1) DE1445634A1 (enExample)
ES (1) ES304831A1 (enExample)
FI (1) FI41029C (enExample)
FR (4) FR4122M (enExample)
GB (1) GB1081757A (enExample)
IL (1) IL22215A (enExample)
NL (2) NL6411794A (enExample)
OA (1) OA01187A (enExample)
SE (2) SE327501B (enExample)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0190709A1 (en) * 1985-02-05 1986-08-13 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Benzoxazinorifamycin derivative, process for preparing the same and anti-bacterial agent containing the same
US4859661A (en) * 1986-07-14 1989-08-22 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Alkyl-substituted benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
US4983602A (en) * 1988-11-01 1991-01-08 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha 3'-hydroxybenzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
EP0333176A3 (en) * 1988-03-18 1991-03-20 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Substituted benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
EP0787494A4 (en) * 1995-09-01 2000-04-26 Kaneka Corp MEDICINE FOR DISEASES CAUSED BY INFECTIONS WITH HELICOBACTER

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH536851A (de) * 1966-10-25 1973-05-15 Ciba Geigy Ag Verfahren zur Herstellung neuer antibiotisch wirksamer Verbindungen der Rifamycinreihen
GB1165179A (en) * 1966-10-25 1969-09-24 Lepetit Spa Derivatives of Rifamycin SV
GB1159267A (en) * 1966-11-03 1969-07-23 Lepetit Spa Rifamycin Derivatives
IT1056271B (it) * 1975-05-20 1982-01-30 Archifar Ind Chim Trentino Prodotti derivati dalle amine aromatiche
IT1056272B (it) * 1975-06-13 1982-01-30 Archifar Ind Chim Trentino Prodotti derivati dalle amine aromatiche
US4690919A (en) * 1984-01-04 1987-09-01 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
GB8608080D0 (en) * 1986-04-02 1986-05-08 Fujisawa Pharmaceutical Co Solid dispersion composition
US7122525B2 (en) * 2001-11-21 2006-10-17 Activbiotics, Inc. Targeted therapeutics and uses thereof
US7078399B2 (en) * 2001-12-13 2006-07-18 Activbiotics, Inc. Sulfhydryl rifamycins and uses thereof
JP2007503439A (ja) * 2003-08-22 2007-02-22 アクティブバイオティクス インコーポレイティッド リファマイシンアナログおよびそれらの使用法
US7820652B2 (en) * 2003-09-24 2010-10-26 Activbiotics Pharma, Llc Regimen for the administration of rifamycin-class antibiotics
EP1697382A4 (en) * 2003-12-10 2008-11-05 Activbiotics Inc ANALOGUES OF RIFAMYCIN AND USES THEREOF
AU2004308399A1 (en) * 2003-12-23 2005-07-14 Activbiotics, Inc. Rifamycin analogs and uses thereof

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0190709A1 (en) * 1985-02-05 1986-08-13 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Benzoxazinorifamycin derivative, process for preparing the same and anti-bacterial agent containing the same
US4859661A (en) * 1986-07-14 1989-08-22 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Alkyl-substituted benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
EP0333176A3 (en) * 1988-03-18 1991-03-20 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Substituted benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
US4983602A (en) * 1988-11-01 1991-01-08 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha 3'-hydroxybenzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
EP0366914A3 (en) * 1988-11-01 1991-07-17 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha 3'-hydroxybenzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
EP0787494A4 (en) * 1995-09-01 2000-04-26 Kaneka Corp MEDICINE FOR DISEASES CAUSED BY INFECTIONS WITH HELICOBACTER

Also Published As

Publication number Publication date
CH504457A (de) 1971-03-15
US3338888A (en) 1967-08-29
BR6463319D0 (pt) 1973-07-17
DE1445634A1 (de) 1968-12-05
FI41029C (fi) 1969-08-11
FR4133M (enExample) 1966-05-02
SE327501B (enExample) 1970-08-24
ES304831A1 (es) 1965-04-01
FR4122M (enExample) 1966-04-25
AT261805B (de) 1968-05-10
NL130099C (enExample)
BE654209A (enExample) 1965-04-09
FI41029B (enExample) 1969-04-30
CH478139A (de) 1969-09-15
FR4152M (enExample) 1966-05-09
SE342458B (enExample) 1972-02-07
NL6411794A (enExample) 1965-04-12
IL22215A (en) 1968-06-20
OA01187A (fr) 1969-01-25
FR4134M (enExample) 1966-05-02

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