FR3713M - Pyrimido [5,4-d] pyrimidines basiquement substituées. - Google Patents

Pyrimido [5,4-d] pyrimidines basiquement substituées.

Info

Publication number
FR3713M
FR3713M FR977447A FR977447A FR3713M FR 3713 M FR3713 M FR 3713M FR 977447 A FR977447 A FR 977447A FR 977447 A FR977447 A FR 977447A FR 3713 M FR3713 M FR 3713M
Authority
FR
France
Prior art keywords
pyrimidines
basically substituted
substituted pyrimido
pyrimido
basically
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR977447A
Other languages
English (en)
French (fr)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Dr Karl Thomae GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR966678A external-priority patent/FR1543161A/fr
Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH
Priority to FR977447A priority Critical patent/FR3713M/fr
Application granted granted Critical
Publication of FR3713M publication Critical patent/FR3713M/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
FR977447A 1963-03-09 1964-06-08 Pyrimido [5,4-d] pyrimidines basiquement substituées. Expired FR3713M (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR977447A FR3713M (fr) 1963-03-09 1964-06-08 Pyrimido [5,4-d] pyrimidines basiquement substituées.

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DET0023605 1963-03-09
FR966678A FR1543161A (fr) 1963-03-09 1964-03-09 Procédé de fabrication de pyrimido [5, 4-d]-pyrimidines basiquement substituées
FR977447A FR3713M (fr) 1963-03-09 1964-06-08 Pyrimido [5,4-d] pyrimidines basiquement substituées.

Publications (1)

Publication Number Publication Date
FR3713M true FR3713M (fr) 1965-11-29

Family

ID=7551073

Family Applications (1)

Application Number Title Priority Date Filing Date
FR977447A Expired FR3713M (fr) 1963-03-09 1964-06-08 Pyrimido [5,4-d] pyrimidines basiquement substituées.

Country Status (5)

Country Link
CH (1) CH438344A (enExample)
DE (1) DE1470341C3 (enExample)
FR (1) FR3713M (enExample)
GB (1) GB1051218A (enExample)
IT (1) IT7950418A0 (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12037346B2 (en) 2021-04-13 2024-07-16 Nuvalent, Inc. Amino-substituted heteroaryls for treating cancers with EGFR mutations

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2004201A1 (de) * 1970-01-30 1971-08-05 Thomae Gmbh Dr K Neue 2,6-Bis(dialkanolamino)-pyrimido-[5,4-d]pyrimidine und Verfahren zu ihrer Herstellung
DE3049207A1 (de) * 1980-12-27 1982-07-29 Dr. Karl Thomae Gmbh, 7950 Biberach Neue trisubstituierte pyrimido (5,4-d) pyrimidine, ihre herstellung und ihre verwendung als arzneimittel
US7772188B2 (en) 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
WO2004093881A2 (en) 2003-04-24 2004-11-04 Boehringer Ingelheim International Gmbh Use of dipyridamole or mopidamole for treatment and prevention of thrombo-embolic diseases and disorders caused by excessive formation of thrombin and/or by elevated expression of thrombin receptors
WO2008151257A2 (en) 2007-06-04 2008-12-11 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
ES2627848T3 (es) 2008-06-04 2017-07-31 Synergy Pharmaceuticals Inc. Agonistas de la guanilato ciclasa útiles para el tratamiento de trastornos gastrointestinales, inflamación, cáncer y otros trastornos
ES2624828T3 (es) 2008-07-16 2017-07-17 Synergy Pharmaceuticals Inc. Agonistas de la guanilato ciclasa útiles para el tratamiento de trastornos gastrointestinales, inflamación, cáncer y otros
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
MX357121B (es) 2011-03-01 2018-06-27 Synergy Pharmaceuticals Inc Star Proceso de preparacion de agonistas c de guanilato ciclasa.
EP2958577A2 (en) 2013-02-25 2015-12-30 Synergy Pharmaceuticals Inc. Guanylate cyclase receptor agonists for use in colonic cleansing
EP2968439A2 (en) 2013-03-15 2016-01-20 Synergy Pharmaceuticals Inc. Compositions useful for the treatment of gastrointestinal disorders
US9708367B2 (en) 2013-03-15 2017-07-18 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase and their uses
PL3004138T3 (pl) 2013-06-05 2024-07-29 Bausch Health Ireland Limited Ultra-oczyszczeni agoniści peptydowi cyklazy guanylanowej C, sposób ich uzyskiwania i ich zastosowanie
CA2920856C (en) 2013-08-09 2026-03-03 Ardelyx, Inc. Ph modulating compounds for inhibiting gastrointestinal phosphate uptake
JP2022533251A (ja) 2019-05-21 2022-07-21 アルデリックス, インコーポレイテッド 患者において血清リン酸塩を低下させるための組み合わせ

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12037346B2 (en) 2021-04-13 2024-07-16 Nuvalent, Inc. Amino-substituted heteroaryls for treating cancers with EGFR mutations

Also Published As

Publication number Publication date
CH438344A (de) 1967-06-30
IT7950418A0 (it) 1979-10-01
DE1470341C3 (de) 1974-07-04
DE1470341A1 (de) 1969-07-03
GB1051218A (enExample)
DE1470341B2 (de) 1973-12-06

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