FR2894965B1 - Nouveaux derives d'oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent - Google Patents

Nouveaux derives d'oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Info

Publication number
FR2894965B1
FR2894965B1 FR0512924A FR0512924A FR2894965B1 FR 2894965 B1 FR2894965 B1 FR 2894965B1 FR 0512924 A FR0512924 A FR 0512924A FR 0512924 A FR0512924 A FR 0512924A FR 2894965 B1 FR2894965 B1 FR 2894965B1
Authority
FR
France
Prior art keywords
preparing
pharmaceutical compositions
compositions containing
containing same
novel heterocyclic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0512924A
Other languages
English (en)
Other versions
FR2894965A1 (fr
Inventor
Franck Suzenet
Gerald Guillaumet
Christelle Pillard
Carine Bassene
Catherine Dacquet
Alain Ktorza
Daniel Henri Caignard
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Laboratoires Servier SAS
Original Assignee
Laboratoires Servier SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR0512924A priority Critical patent/FR2894965B1/fr
Application filed by Laboratoires Servier SAS filed Critical Laboratoires Servier SAS
Priority to BRPI0620190-3A priority patent/BRPI0620190A2/pt
Priority to KR1020087017808A priority patent/KR20080077030A/ko
Priority to AU2006334310A priority patent/AU2006334310A1/en
Priority to US12/086,785 priority patent/US20090274674A1/en
Priority to JP2008546513A priority patent/JP2009520007A/ja
Priority to EP06847063A priority patent/EP1966204A1/fr
Priority to PCT/FR2006/002778 priority patent/WO2007077313A1/fr
Priority to EA200801566A priority patent/EA014317B1/ru
Priority to CNA200680052931XA priority patent/CN101374837A/zh
Priority to CA002634320A priority patent/CA2634320A1/fr
Priority to ZA200805976A priority patent/ZA200805976B/xx
Priority to ARP060105638A priority patent/AR058573A1/es
Publication of FR2894965A1 publication Critical patent/FR2894965A1/fr
Application granted granted Critical
Publication of FR2894965B1 publication Critical patent/FR2894965B1/fr
Priority to MA31052A priority patent/MA30068B1/fr
Priority to NO20082821A priority patent/NO20082821L/no
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Neurology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurosurgery (AREA)
  • Vascular Medicine (AREA)
  • Dermatology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Psychiatry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR0512924A 2005-12-20 2005-12-20 Nouveaux derives d'oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent Expired - Fee Related FR2894965B1 (fr)

Priority Applications (15)

Application Number Priority Date Filing Date Title
FR0512924A FR2894965B1 (fr) 2005-12-20 2005-12-20 Nouveaux derives d'oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
CA002634320A CA2634320A1 (fr) 2005-12-20 2006-12-19 Nouveaux derives d'oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
AU2006334310A AU2006334310A1 (en) 2005-12-20 2006-12-19 Novel heterocyclic oxime derivatives, process for the preparation thereof and pharmaceutical compositions containing them
US12/086,785 US20090274674A1 (en) 2005-12-20 2006-12-19 Heterocyclic Oxime Compounds, Process for Their Preparation and Pharmaceutical Compositions Containing Them
JP2008546513A JP2009520007A (ja) 2005-12-20 2006-12-19 新規な複素環オキシム誘導体、その製造方法及びこれらを含む薬剤組成物
EP06847063A EP1966204A1 (fr) 2005-12-20 2006-12-19 Nouveaux derives d oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
PCT/FR2006/002778 WO2007077313A1 (fr) 2005-12-20 2006-12-19 Nouveaux derives d’oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
EA200801566A EA014317B1 (ru) 2005-12-20 2006-12-19 Новые гетероциклические соединения оксима, способ их получения и фармацевтические композиции, которые их содержат
BRPI0620190-3A BRPI0620190A2 (pt) 2005-12-20 2006-12-19 derivados de oximas heterocìclicas, respectivo processo de preparação e composições farmacêuticas que os contêm
KR1020087017808A KR20080077030A (ko) 2005-12-20 2006-12-19 헤테로시클릭 옥심 유도체, 이의 제조방법, 및 이를함유하는 약제학적 조성물
ZA200805976A ZA200805976B (en) 2005-12-20 2006-12-19 Novel heterocyclic oxime derivatives, process for the preparation thereof and pharmaceutical compositions containing them
CNA200680052931XA CN101374837A (zh) 2005-12-20 2006-12-19 新的杂环肟衍生物、其制备方法和包含它们的药物组合物
ARP060105638A AR058573A1 (es) 2005-12-20 2006-12-20 Derivados de oximas heterociclicas procedimiento para su preparacion y composiciones farmaceuticas que los contienen
MA31052A MA30068B1 (fr) 2005-12-20 2008-06-19 Nouveaux derives d'oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
NO20082821A NO20082821L (no) 2005-12-20 2008-06-25 Nye heterocykliske oksim-derivater, fremgangsmaten for fremstilling derav samt farmasoytiske sammensetninger inneholdende slike

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0512924A FR2894965B1 (fr) 2005-12-20 2005-12-20 Nouveaux derives d'oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number Publication Date
FR2894965A1 FR2894965A1 (fr) 2007-06-22
FR2894965B1 true FR2894965B1 (fr) 2008-01-25

Family

ID=37055975

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0512924A Expired - Fee Related FR2894965B1 (fr) 2005-12-20 2005-12-20 Nouveaux derives d'oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Country Status (15)

Country Link
US (1) US20090274674A1 (fr)
EP (1) EP1966204A1 (fr)
JP (1) JP2009520007A (fr)
KR (1) KR20080077030A (fr)
CN (1) CN101374837A (fr)
AR (1) AR058573A1 (fr)
AU (1) AU2006334310A1 (fr)
BR (1) BRPI0620190A2 (fr)
CA (1) CA2634320A1 (fr)
EA (1) EA014317B1 (fr)
FR (1) FR2894965B1 (fr)
MA (1) MA30068B1 (fr)
NO (1) NO20082821L (fr)
WO (1) WO2007077313A1 (fr)
ZA (1) ZA200805976B (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010026771A1 (fr) * 2008-09-08 2010-03-11 日本曹達株式会社 Composé hétérocyclique azoté et son sel, et agent bactéricide pour des applications en agriculture ou horticulture

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2804431A1 (fr) * 2000-02-02 2001-08-03 Adir Nouveaux derives heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2858321B1 (fr) * 2003-07-28 2006-01-20 Servier Lab Nouveaux derives d'oximes heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2868313B1 (fr) * 2004-03-31 2008-08-15 Servier Lab Nouvelle association entre un compose heterocyclique et un agent antioxydant et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
AR058573A1 (es) 2008-02-13
KR20080077030A (ko) 2008-08-20
JP2009520007A (ja) 2009-05-21
EP1966204A1 (fr) 2008-09-10
EA200801566A1 (ru) 2008-12-30
FR2894965A1 (fr) 2007-06-22
BRPI0620190A2 (pt) 2011-11-01
CA2634320A1 (fr) 2007-07-12
AU2006334310A1 (en) 2007-07-12
CN101374837A (zh) 2009-02-25
EA014317B1 (ru) 2010-10-29
MA30068B1 (fr) 2008-12-01
WO2007077313A1 (fr) 2007-07-12
US20090274674A1 (en) 2009-11-05
NO20082821L (no) 2008-08-26
ZA200805976B (en) 2009-11-25

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Effective date: 20120831