FR2873585B1 - Nouvelles formulations galeniques de principes actifs - Google Patents

Nouvelles formulations galeniques de principes actifs

Info

Publication number
FR2873585B1
FR2873585B1 FR0408269A FR0408269A FR2873585B1 FR 2873585 B1 FR2873585 B1 FR 2873585B1 FR 0408269 A FR0408269 A FR 0408269A FR 0408269 A FR0408269 A FR 0408269A FR 2873585 B1 FR2873585 B1 FR 2873585B1
Authority
FR
France
Prior art keywords
active principles
galenic formulations
new galenic
new
formulations
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0408269A
Other languages
English (en)
Other versions
FR2873585A1 (fr
Inventor
Jean Pachot
Chicq Serge Segot
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharma SA
Original Assignee
Aventis Pharma SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR0408269A priority Critical patent/FR2873585B1/fr
Application filed by Aventis Pharma SA filed Critical Aventis Pharma SA
Priority to JP2007521988A priority patent/JP2008508191A/ja
Priority to US11/572,402 priority patent/US20080193519A1/en
Priority to CA002579449A priority patent/CA2579449A1/fr
Priority to PCT/FR2005/001853 priority patent/WO2006018501A1/fr
Priority to BRPI0513622-9A priority patent/BRPI0513622A/pt
Priority to EP05790808A priority patent/EP1771154A1/fr
Priority to NZ552715A priority patent/NZ552715A/en
Priority to AU2005273839A priority patent/AU2005273839A1/en
Priority to CNA2005800268156A priority patent/CN101001608A/zh
Priority to KR1020077001445A priority patent/KR20070046819A/ko
Priority to RU2007107199/15A priority patent/RU2381789C2/ru
Priority to MX2007001141A priority patent/MX2007001141A/es
Priority to TW094125195A priority patent/TW200616640A/zh
Publication of FR2873585A1 publication Critical patent/FR2873585A1/fr
Publication of FR2873585B1 publication Critical patent/FR2873585B1/fr
Application granted granted Critical
Priority to IL180714A priority patent/IL180714A0/en
Priority to ZA200700553A priority patent/ZA200700553B/en
Priority to NO20070354A priority patent/NO20070354L/no
Priority to MA29627A priority patent/MA28748B1/fr
Priority to US12/870,250 priority patent/US20110104268A1/en
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FR0408269A 2004-07-20 2004-07-27 Nouvelles formulations galeniques de principes actifs Expired - Fee Related FR2873585B1 (fr)

Priority Applications (19)

Application Number Priority Date Filing Date Title
FR0408269A FR2873585B1 (fr) 2004-07-27 2004-07-27 Nouvelles formulations galeniques de principes actifs
CA002579449A CA2579449A1 (fr) 2004-07-27 2005-07-20 Applications galeniques de melanges auto-emulsionnants d'excipients lipidiques
RU2007107199/15A RU2381789C2 (ru) 2004-07-27 2005-07-20 Применение самоэмульгирующихся смесей липидных эксципиентов в галеновых препаратах
PCT/FR2005/001853 WO2006018501A1 (fr) 2004-07-27 2005-07-20 Applications galeniques de melanges auto-emulsionnants d'excipients lipidiques
BRPI0513622-9A BRPI0513622A (pt) 2004-07-27 2005-07-20 aplicação de combinações auto-emulsificantes (seeds) de excipientes lipìdicos, de surfactantes; composição farmacêutica contendo um princìpio ativo e uma combinação auto-emulsificante (seeds) de excipientes lipìdicos, de surfactantes; e processo para a preparação de combinações auto-emulsificantes (seeds) de excipientes lipìdios, de surfactantes
EP05790808A EP1771154A1 (fr) 2004-07-27 2005-07-20 Applications galeniques de melanges auto-emulsionnants d'excipients lipidiques
NZ552715A NZ552715A (en) 2004-07-27 2005-07-20 Galenic applications of self-emulsifying mixtures of lipidic excipients
AU2005273839A AU2005273839A1 (en) 2004-07-27 2005-07-20 Galenic applications of self-emulsifying mixtures of lipidic excipients
CNA2005800268156A CN101001608A (zh) 2004-07-27 2005-07-20 脂类赋形剂的自乳化混合物的药物应用
KR1020077001445A KR20070046819A (ko) 2004-07-27 2005-07-20 지질 부형제의 자가 유화 혼합물의 갈레노스 용도
JP2007521988A JP2008508191A (ja) 2004-07-27 2005-07-20 脂質賦形剤の自己乳化混合物のガレノス式適用
MX2007001141A MX2007001141A (es) 2004-07-27 2005-07-20 Aplicaciones galenicas de mezclas auto-emulsionantes de excipientes lipidicos.
US11/572,402 US20080193519A1 (en) 2004-07-20 2005-07-20 Galenic Applications of Self-Emulsifying Mixtures of Lipidic Excipients
TW094125195A TW200616640A (en) 2004-07-27 2005-07-26 Novel pharmaceutical formulations of active principles
IL180714A IL180714A0 (en) 2004-07-27 2007-01-15 Galenic applications of self-emulsifying mixtures of lipidic excipients
NO20070354A NO20070354L (no) 2004-07-27 2007-01-19 Galeniske anvendelser om selvemulgerende blandinger av lipideksipienter
ZA200700553A ZA200700553B (en) 2004-07-27 2007-01-19 Galenic applications of self-emulsifying mixtures of lipidic excipients
MA29627A MA28748B1 (fr) 2004-07-27 2007-01-23 Applications galeniques de melanges auto-emulsionnants d'excipients lipidiques
US12/870,250 US20110104268A1 (en) 2004-07-27 2010-08-27 Galenic applications of self-emulsifying mixtures of lipidic excipients

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0408269A FR2873585B1 (fr) 2004-07-27 2004-07-27 Nouvelles formulations galeniques de principes actifs

Publications (2)

Publication Number Publication Date
FR2873585A1 FR2873585A1 (fr) 2006-02-03
FR2873585B1 true FR2873585B1 (fr) 2006-11-17

Family

ID=34951660

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0408269A Expired - Fee Related FR2873585B1 (fr) 2004-07-20 2004-07-27 Nouvelles formulations galeniques de principes actifs

Country Status (18)

Country Link
US (2) US20080193519A1 (fr)
EP (1) EP1771154A1 (fr)
JP (1) JP2008508191A (fr)
KR (1) KR20070046819A (fr)
CN (1) CN101001608A (fr)
AU (1) AU2005273839A1 (fr)
BR (1) BRPI0513622A (fr)
CA (1) CA2579449A1 (fr)
FR (1) FR2873585B1 (fr)
IL (1) IL180714A0 (fr)
MA (1) MA28748B1 (fr)
MX (1) MX2007001141A (fr)
NO (1) NO20070354L (fr)
NZ (1) NZ552715A (fr)
RU (1) RU2381789C2 (fr)
TW (1) TW200616640A (fr)
WO (1) WO2006018501A1 (fr)
ZA (1) ZA200700553B (fr)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1867323A1 (fr) * 2006-06-13 2007-12-19 Farmatron Ltd. Formulations pharmaceutiques avec pénétration améliorée à travers des barrières biologiques
MX2010001730A (es) * 2007-08-21 2010-03-10 Basilea Pharmaceutica Ag Composicion antimicotica.
JP5951489B2 (ja) 2009-10-16 2016-07-13 グラクソスミスクライン・リミテッド・ライアビリティ・カンパニーGlaxoSmithKline LLC 組成物
JP2013209294A (ja) * 2010-07-30 2013-10-10 Meiji Seikaファルマ株式会社 液状医薬組成物
BR112014012444B1 (pt) 2011-11-23 2021-12-14 Therapeuticsmd, Inc Composição farmacêutica compreendendo estradiol solubilizado, progesterona e um agente de solubilização, bem como usos desta para tratar um sintoma relacionado à menopausa em uma mulher
US9301920B2 (en) 2012-06-18 2016-04-05 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US20150196640A1 (en) 2012-06-18 2015-07-16 Therapeuticsmd, Inc. Progesterone formulations having a desirable pk profile
US10806740B2 (en) 2012-06-18 2020-10-20 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US20130338122A1 (en) 2012-06-18 2013-12-19 Therapeuticsmd, Inc. Transdermal hormone replacement therapies
US10806697B2 (en) 2012-12-21 2020-10-20 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US11266661B2 (en) 2012-12-21 2022-03-08 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US9180091B2 (en) 2012-12-21 2015-11-10 Therapeuticsmd, Inc. Soluble estradiol capsule for vaginal insertion
US11246875B2 (en) 2012-12-21 2022-02-15 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10537581B2 (en) 2012-12-21 2020-01-21 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10471072B2 (en) 2012-12-21 2019-11-12 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10568891B2 (en) 2012-12-21 2020-02-25 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
JP2017516768A (ja) 2014-05-22 2017-06-22 セラピューティックスエムディー インコーポレーテッドTherapeuticsmd, Inc. 天然の併用ホルモン補充療法剤及び療法
KR101542364B1 (ko) * 2014-10-31 2015-08-07 대화제약 주식회사 탁산을 포함하는 경구 투여용 약학 조성물
US10328087B2 (en) 2015-07-23 2019-06-25 Therapeuticsmd, Inc. Formulations for solubilizing hormones
US10286077B2 (en) 2016-04-01 2019-05-14 Therapeuticsmd, Inc. Steroid hormone compositions in medium chain oils
EP3435977A4 (fr) 2016-04-01 2019-10-16 Therapeuticsmd, Inc. Composition pharmaceutique d'hormone stéroïde
WO2020123551A1 (fr) * 2018-12-10 2020-06-18 Halo Science LLC Formulations stables d'anesthésiques et formes galéniques associées
CZ309587B6 (cs) * 2021-01-22 2023-05-03 Oncora S.R.O. Mikroemulzní prekoncentrát s obsahem kladribinu a způsob jeho přípravy
CN114246827B (zh) * 2022-01-04 2023-04-11 中山大学 一种鱼油微乳制剂及其制备方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8916901D0 (en) * 1989-07-24 1989-09-06 Sandoz Ltd Improvements in or relating to organic compounds
FR2710535B1 (fr) * 1993-09-30 1995-11-24 Gattefosse Ets Sa Composition à usage pharmaceutique ou cosmétique apte à former une microémulsion.
US6054136A (en) * 1993-09-30 2000-04-25 Gattefosse S.A. Orally administrable composition capable of providing enhanced bioavailability when ingested
EP0933367A1 (fr) * 1997-12-19 1999-08-04 Hoechst Marion Roussel Deutschland GmbH Dérivés d'acylguanidine comme inhibiteurs de résorbtion osseuse et comme antagonistes de récepteur vitronectine
WO1999037621A1 (fr) * 1998-01-23 1999-07-29 Aventis Pharma Deutschland Gmbh Nouveaux derives de sulfamide comme inhibiteurs de la resorption osseuse et comme inhibiteurs de l'adherence cellulaire
AU756752B2 (en) * 1998-04-01 2003-01-23 Skyepharma Canada Inc. Anticancer compositions
CA2302735A1 (fr) * 1998-07-14 2000-01-27 Em Industries, Inc. Systemes d'apport de medicaments par microdispersion
GB0003685D0 (en) * 2000-02-17 2000-04-05 Univ Cardiff Sensitisation of cellular material
FR2818905A1 (fr) * 2000-12-28 2002-07-05 Cll Pharma Compositions pharmaceutiques colloidales micellaires renfermant un principe actif lipophile
FR2827770B1 (fr) * 2001-07-27 2005-08-19 Gattefosse Ets Sa Composition pharmaceutique a usage oral comprenant un principe actif susceptible de subir un important effet de premier passage intestinal
AU2002357012A1 (en) * 2001-11-27 2003-06-10 Transform Pharmaceuticals, Inc. Oral pharmaceutical formulations comprising paclitaxel, derivatives and methods of administration thereof
JP4464814B2 (ja) * 2002-05-14 2010-05-19 アバーント・ファーマシューティカルズ・(インディア)・リミテッド アントラニル酸誘導体の水和物の製造方法

Also Published As

Publication number Publication date
ZA200700553B (en) 2008-05-28
CA2579449A1 (fr) 2006-02-23
NZ552715A (en) 2010-12-24
AU2005273839A1 (en) 2006-02-23
NO20070354L (no) 2007-04-17
RU2007107199A (ru) 2008-09-10
WO2006018501A1 (fr) 2006-02-23
WO2006018501A8 (fr) 2007-03-01
RU2381789C2 (ru) 2010-02-20
EP1771154A1 (fr) 2007-04-11
JP2008508191A (ja) 2008-03-21
US20110104268A1 (en) 2011-05-05
FR2873585A1 (fr) 2006-02-03
MA28748B1 (fr) 2007-07-02
CN101001608A (zh) 2007-07-18
KR20070046819A (ko) 2007-05-03
IL180714A0 (en) 2007-06-03
US20080193519A1 (en) 2008-08-14
BRPI0513622A (pt) 2008-05-13
MX2007001141A (es) 2007-04-19
TW200616640A (en) 2006-06-01

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Legal Events

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ST Notification of lapse

Effective date: 20130329