FR2577925B1 - Aminoalcanoylureido amino et imino acides et esters a substituant ester, a proprietes therapeutiques - Google Patents

Aminoalcanoylureido amino et imino acides et esters a substituant ester, a proprietes therapeutiques

Info

Publication number
FR2577925B1
FR2577925B1 FR8602835A FR8602835A FR2577925B1 FR 2577925 B1 FR2577925 B1 FR 2577925B1 FR 8602835 A FR8602835 A FR 8602835A FR 8602835 A FR8602835 A FR 8602835A FR 2577925 B1 FR2577925 B1 FR 2577925B1
Authority
FR
France
Prior art keywords
aminoalcanoylureido
esters
amino
therapeutic properties
substituted ester
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
FR8602835A
Other languages
English (en)
Other versions
FR2577925A1 (fr
Inventor
Harold N Weller Iii
Eric M Gordon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of FR2577925A1 publication Critical patent/FR2577925A1/fr
Application granted granted Critical
Publication of FR2577925B1 publication Critical patent/FR2577925B1/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Indole Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FR8602835A 1985-02-28 1986-02-28 Aminoalcanoylureido amino et imino acides et esters a substituant ester, a proprietes therapeutiques Expired FR2577925B1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/707,123 US4638010A (en) 1985-02-28 1985-02-28 Ester substituted aminoalkanoylureido amino and imino acid and ester compounds

Publications (2)

Publication Number Publication Date
FR2577925A1 FR2577925A1 (fr) 1986-08-29
FR2577925B1 true FR2577925B1 (fr) 1987-11-27

Family

ID=24840442

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8602835A Expired FR2577925B1 (fr) 1985-02-28 1986-02-28 Aminoalcanoylureido amino et imino acides et esters a substituant ester, a proprietes therapeutiques

Country Status (7)

Country Link
US (1) US4638010A (fr)
JP (1) JPS61227558A (fr)
CA (1) CA1261332A (fr)
DE (1) DE3606448A1 (fr)
FR (1) FR2577925B1 (fr)
GB (1) GB2171698B (fr)
IT (1) IT1188556B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0190852A3 (fr) * 1985-01-31 1988-11-02 Ajinomoto Co., Inc. Dérivés dipeptides et les médicaments antihypertensifs les contenant
US5013861A (en) * 1985-02-28 1991-05-07 E. R. Squibb & Sons, Inc. Ester substituted aminoalkanoylureido amino and imino acid and ester compounds
US5151513A (en) * 1988-04-29 1992-09-29 E. R. Squibb & Sons, Inc. N-heterocyclic alcohol derivatives
CA1340588C (fr) * 1988-06-13 1999-06-08 Balraj Krishan Handa Derive d'aminoacides
US6586466B2 (en) 1995-10-30 2003-07-01 Smithkline Beecham Corporation Carbohydrazide-protease inhibitors
KR19990067184A (ko) 1995-10-30 1999-08-16 스튜어트 알. 수터, 스티븐 베네티아너, 피터 존 기딩스 프로테아제 억제제
EP0915093B1 (fr) * 1996-06-06 2002-11-27 Otsuka Pharmaceutical Factory, Inc. Derives d'amides
BR9815469A (pt) * 1997-05-08 2001-03-06 Smithkline Beecham Corp Inibidores de protease
US20030144175A1 (en) * 1998-12-23 2003-07-31 Smithkline Beecham Corporation Protease inhibitors
US20030044399A1 (en) * 1998-12-23 2003-03-06 Smithkline Beecham Corporation Method of treatment
WO2001034599A1 (fr) 1999-11-10 2001-05-17 Smithkline Beecham Corporation Inhibiteurs de protease
US6534498B1 (en) 1999-11-10 2003-03-18 Smithkline Beecham Corporation Protease inhibitors
WO2001034600A1 (fr) 1999-11-10 2001-05-17 Smithkline Beecham Corporation Inhibiteurs de protease
AU2001243441B2 (en) * 2000-03-21 2004-11-25 Smithkline Beecham Corporation Protease inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4329473A (en) * 1979-06-01 1982-05-11 Almquist Ronald G Oxoalkanoic acid derivatives as inhibitors of angiotensin converting enzyme
US4402969A (en) * 1981-03-23 1983-09-06 Merck & Co., Inc. Antihypertensive proline derivatives
JPS58170752A (ja) * 1982-03-30 1983-10-07 Kureha Chem Ind Co Ltd Ｎ−カルバモイルアミノ酸誘導体
IT8222367V0 (it) * 1982-07-09 1982-07-09 Cavalli Alfredo Trafila per pasta sfoglia, particolarmente per macchine per la pasta di uso domestico.
US4623729A (en) * 1982-07-22 1986-11-18 E. R. Squibb & Sons, Inc. Acylalkylaminocarbonyl substituted amino and imino acid compounds

Also Published As

Publication number Publication date
FR2577925A1 (fr) 1986-08-29
CA1261332A (fr) 1989-09-26
GB2171698A (en) 1986-09-03
IT1188556B (it) 1988-01-20
IT8619593A0 (it) 1986-02-28
US4638010A (en) 1987-01-20
DE3606448A1 (de) 1986-08-28
JPS61227558A (ja) 1986-10-09
IT8619593A1 (it) 1987-08-28
GB8603626D0 (en) 1986-03-19
GB2171698B (en) 1989-02-01

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Legal Events

Date Code Title Description
ST Notification of lapse