FR2514354A1 - Nouveaux derives de 5-aminoisoxazole et procedes de leur preparation - Google Patents
Nouveaux derives de 5-aminoisoxazole et procedes de leur preparation Download PDFInfo
- Publication number
- FR2514354A1 FR2514354A1 FR8216914A FR8216914A FR2514354A1 FR 2514354 A1 FR2514354 A1 FR 2514354A1 FR 8216914 A FR8216914 A FR 8216914A FR 8216914 A FR8216914 A FR 8216914A FR 2514354 A1 FR2514354 A1 FR 2514354A1
- Authority
- FR
- France
- Prior art keywords
- group
- methyl
- lower alkyl
- alkyl group
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/14—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP56161206A JPS5862169A (ja) | 1981-10-09 | 1981-10-09 | 新規な5−アミノイソオキサゾ−ル誘導体 |
Publications (1)
Publication Number | Publication Date |
---|---|
FR2514354A1 true FR2514354A1 (fr) | 1983-04-15 |
Family
ID=15730608
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR8216914A Withdrawn FR2514354A1 (fr) | 1981-10-09 | 1982-10-08 | Nouveaux derives de 5-aminoisoxazole et procedes de leur preparation |
Country Status (7)
Country | Link |
---|---|
JP (1) | JPS5862169A (es) |
DE (1) | DE3237149A1 (es) |
ES (2) | ES516787A0 (es) |
FR (1) | FR2514354A1 (es) |
GB (1) | GB2107710A (es) |
IT (1) | IT8223685A0 (es) |
SE (1) | SE8205583L (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5338857A (en) * | 1989-08-04 | 1994-08-16 | Mitsui Toatsu Chemicals Incorporated | Aminoketone derivatives of 1,2-oxazole and use thereof |
JPH0625178B2 (ja) * | 1989-08-04 | 1994-04-06 | 三井東圧化学株式会社 | アミノケトン誘導体及びその用途 |
JPH04368375A (ja) * | 1991-06-17 | 1992-12-21 | Otsuka Pharmaceut Factory Inc | イソオキサゾール誘導体 |
US6544982B1 (en) * | 1999-10-29 | 2003-04-08 | Merck & Co., Inc. | Thrombin receptor antagonists |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2068418A1 (en) * | 1969-10-27 | 1971-08-27 | Innothera Lab Sa | 2-substd-5-amino isoxazole derivs |
-
1981
- 1981-10-09 JP JP56161206A patent/JPS5862169A/ja active Pending
-
1982
- 1982-09-30 SE SE8205583A patent/SE8205583L/xx not_active Application Discontinuation
- 1982-10-07 DE DE19823237149 patent/DE3237149A1/de not_active Withdrawn
- 1982-10-08 FR FR8216914A patent/FR2514354A1/fr not_active Withdrawn
- 1982-10-08 GB GB08228896A patent/GB2107710A/en not_active Withdrawn
- 1982-10-08 ES ES516787A patent/ES516787A0/es active Granted
- 1982-10-08 IT IT8223685A patent/IT8223685A0/it unknown
-
1983
- 1983-10-31 ES ES526914A patent/ES8504156A1/es not_active Expired
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2068418A1 (en) * | 1969-10-27 | 1971-08-27 | Innothera Lab Sa | 2-substd-5-amino isoxazole derivs |
Non-Patent Citations (1)
Title |
---|
CHEMICAL ABSTRACTS, vol. 90, no. 25, 18 juin 1979, pages 611-612, abrégé 203924k, Columbus, Ohio, US; J.P. TRIVEDI et al.: "Synthesis and pharmacology of 5-(N,N-(di-alkylamino)-acetamido)-3,4-dimethyl isoxazoles and N-(di-alkylamino)-acetyl-11-H-dibenz(b,e)azepine", & Indian J. Pharm. Sci. 1979, 41(1), 28-31 * |
Also Published As
Publication number | Publication date |
---|---|
SE8205583L (sv) | 1983-04-10 |
ES8402278A1 (es) | 1984-02-01 |
DE3237149A1 (de) | 1983-04-21 |
ES526914A0 (es) | 1985-04-01 |
ES516787A0 (es) | 1984-02-01 |
JPS5862169A (ja) | 1983-04-13 |
SE8205583D0 (sv) | 1982-09-30 |
ES8504156A1 (es) | 1985-04-01 |
GB2107710A (en) | 1983-05-05 |
IT8223685A0 (it) | 1982-10-08 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |