FR2475554A1 - 7-((2-amino-4-thiazolyl)(carboxy(alkylthio)alcoxyimino)-acetamido)cephalospori-nes a action anti-bacterienne - Google Patents

7-((2-amino-4-thiazolyl)(carboxy(alkylthio)alcoxyimino)-acetamido)cephalospori-nes a action anti-bacterienne Download PDF

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Publication number
FR2475554A1
FR2475554A1 FR8102612A FR8102612A FR2475554A1 FR 2475554 A1 FR2475554 A1 FR 2475554A1 FR 8102612 A FR8102612 A FR 8102612A FR 8102612 A FR8102612 A FR 8102612A FR 2475554 A1 FR2475554 A1 FR 2475554A1
Authority
FR
France
Prior art keywords
amino
methyl
oxo
thia
thiazolyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR8102612A
Other languages
English (en)
French (fr)
Other versions
FR2475554B1 (enrdf_load_stackoverflow
Inventor
Hermann Breuer
Uwe Treuner
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
ER Squibb and Sons LLC
Original Assignee
ER Squibb and Sons LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ER Squibb and Sons LLC filed Critical ER Squibb and Sons LLC
Publication of FR2475554A1 publication Critical patent/FR2475554A1/fr
Application granted granted Critical
Publication of FR2475554B1 publication Critical patent/FR2475554B1/fr
Granted legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
FR8102612A 1980-02-11 1981-02-10 7-((2-amino-4-thiazolyl)(carboxy(alkylthio)alcoxyimino)-acetamido)cephalospori-nes a action anti-bacterienne Granted FR2475554A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12017580A 1980-02-11 1980-02-11

Publications (2)

Publication Number Publication Date
FR2475554A1 true FR2475554A1 (fr) 1981-08-14
FR2475554B1 FR2475554B1 (enrdf_load_stackoverflow) 1983-07-18

Family

ID=22388685

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8102612A Granted FR2475554A1 (fr) 1980-02-11 1981-02-10 7-((2-amino-4-thiazolyl)(carboxy(alkylthio)alcoxyimino)-acetamido)cephalospori-nes a action anti-bacterienne

Country Status (5)

Country Link
JP (1) JPS56127389A (enrdf_load_stackoverflow)
DE (1) DE3104696A1 (enrdf_load_stackoverflow)
FR (1) FR2475554A1 (enrdf_load_stackoverflow)
GB (1) GB2068958B (enrdf_load_stackoverflow)
IT (1) IT1167706B (enrdf_load_stackoverflow)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4868173A (en) * 1984-11-20 1989-09-19 Ici Pharma Cephalosporin derivatives
EP0187456A1 (en) * 1984-11-29 1986-07-16 Ici Pharma Cephalosporin derivatives
GB8626245D0 (en) * 1985-11-27 1986-12-03 Ici Pharma Cephalosporin compounds
TW209223B (enrdf_load_stackoverflow) * 1989-09-26 1993-07-11 Yamanouchi Pharma Co Ltd

Also Published As

Publication number Publication date
FR2475554B1 (enrdf_load_stackoverflow) 1983-07-18
JPS56127389A (en) 1981-10-06
IT1167706B (it) 1987-05-13
IT8119672A0 (it) 1981-02-11
IT8119672A1 (it) 1982-08-11
GB2068958A (en) 1981-08-19
GB2068958B (en) 1984-02-29
DE3104696A1 (de) 1981-11-26

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