FR2458540A1 - Nouveaux derives de l'encephaline, procede de preparation de ces derives et medicaments les contenant - Google Patents
Nouveaux derives de l'encephaline, procede de preparation de ces derives et medicaments les contenant Download PDFInfo
- Publication number
- FR2458540A1 FR2458540A1 FR8012496A FR8012496A FR2458540A1 FR 2458540 A1 FR2458540 A1 FR 2458540A1 FR 8012496 A FR8012496 A FR 8012496A FR 8012496 A FR8012496 A FR 8012496A FR 2458540 A1 FR2458540 A1 FR 2458540A1
- Authority
- FR
- France
- Prior art keywords
- amide
- group
- enkephalin
- derivatives
- salts
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/70—Enkephalins
- C07K14/702—Enkephalins with at least 1 amino acid in D-form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Zoology (AREA)
- Toxicology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Gastroenterology & Hepatology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU79GO1448A HU178004B (en) | 1979-06-12 | 1979-06-12 | Process for preparing new encephaline derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2458540A1 true FR2458540A1 (fr) | 1981-01-02 |
FR2458540B1 FR2458540B1 (de) | 1984-04-27 |
Family
ID=10996895
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR8012496A Granted FR2458540A1 (fr) | 1979-06-12 | 1980-06-05 | Nouveaux derives de l'encephaline, procede de preparation de ces derives et medicaments les contenant |
Country Status (8)
Country | Link |
---|---|
JP (1) | JPS56115752A (de) |
BE (1) | BE883641A (de) |
CH (1) | CH645093A5 (de) |
DE (1) | DE3022098A1 (de) |
FR (1) | FR2458540A1 (de) |
GB (1) | GB2053925B (de) |
HU (1) | HU178004B (de) |
NL (1) | NL8003423A (de) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1248299A (en) * | 1982-02-05 | 1989-01-03 | Lawrence A. Lowe | Pharmaceutical compounds, preparation, use and intermediates therefor and their preparation |
-
1979
- 1979-06-12 HU HU79GO1448A patent/HU178004B/hu unknown
-
1980
- 1980-06-05 FR FR8012496A patent/FR2458540A1/fr active Granted
- 1980-06-05 BE BE1/9839A patent/BE883641A/fr not_active IP Right Cessation
- 1980-06-09 GB GB8018785A patent/GB2053925B/en not_active Expired
- 1980-06-11 CH CH448180A patent/CH645093A5/de not_active IP Right Cessation
- 1980-06-12 NL NL8003423A patent/NL8003423A/nl not_active Application Discontinuation
- 1980-06-12 DE DE19803022098 patent/DE3022098A1/de not_active Withdrawn
- 1980-06-12 JP JP7844680A patent/JPS56115752A/ja active Pending
Non-Patent Citations (3)
Title |
---|
Chemical Abstracts vol. 83, no. 13, 29 septembre 1975, Columbus, Ohio, USA G. WEITZEL et al. "Structure and activity of insulin. XIII. Specificity of the arginine-guanidino group in biologically active tetrapeptides of the insulin sequence B 22-25 (Arg-Gly-Phe-Phe) * |
Chemical Abstracts vol. 84, no. 11, 15 mars 1976 Columbus, Ohio, USA K. EISELE et al. "Synthesis of homoarginine and a homoarginyl tetrapeptide amide" page 488, colonne 2, abrégé no. 74606h, en combi naison avec C.A. Chemical subject index 1972-76, p * |
Chemical Abstracts vol. 92, no. 17, 28 avril 1980 Columbus, Ohio, USA S. BAJUSZ et al. "Further enhancement of analgesic activity: enkephalin analogs with terminal guanidino group" page 71, colonne 1, abrégé no. 140894u * |
Also Published As
Publication number | Publication date |
---|---|
GB2053925A (en) | 1981-02-11 |
GB2053925B (en) | 1983-04-07 |
JPS56115752A (en) | 1981-09-11 |
FR2458540B1 (de) | 1984-04-27 |
HU178004B (en) | 1982-02-28 |
BE883641A (fr) | 1980-12-05 |
CH645093A5 (de) | 1984-09-14 |
NL8003423A (nl) | 1980-12-16 |
DE3022098A1 (de) | 1980-12-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |