FR2452486A1 - Nouveaux derives d'a-(3,4-dichlorophenyl)-imidazoline ou pyrimidine-2-methane utiles notamment comme agents antisecretoires et leur procede de preparation - Google Patents

Nouveaux derives d'a-(3,4-dichlorophenyl)-imidazoline ou pyrimidine-2-methane utiles notamment comme agents antisecretoires et leur procede de preparation

Info

Publication number
FR2452486A1
FR2452486A1 FR8006391A FR8006391A FR2452486A1 FR 2452486 A1 FR2452486 A1 FR 2452486A1 FR 8006391 A FR8006391 A FR 8006391A FR 8006391 A FR8006391 A FR 8006391A FR 2452486 A1 FR2452486 A1 FR 2452486A1
Authority
FR
France
Prior art keywords
imidazoline
dichlorophenyl
pyrimidine
novel
preparation process
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR8006391A
Other languages
English (en)
Other versions
FR2452486B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Richardson Vicks Inc
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of FR2452486A1 publication Critical patent/FR2452486A1/fr
Application granted granted Critical
Publication of FR2452486B1 publication Critical patent/FR2452486B1/fr
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D233/22—Radicals substituted by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

L'INVENTION CONCERNE DE NOUVEAUX DERIVES D'A-(3,4-DICHLOROPHENYL)-IMIDAZOLINE OU PYRIMIDINE-2-METHANOLS REPONDANT A LA FORMULE GENERALE: (CF DESSIN DANS BOPI) DANS LAQUELLE R EST UN GROUPE (CF DESSIN DANS BOPI) ET LEURS SELS D'ADDITION D'ACIDES ACCEPTABLES EN PHARMACIE. ON PEUT LES ADMINISTRER PAR VOIE ORALE, PARENTERALE OU LOCALE A DES DOSES JOURNALIERES DE 1-50MGKG DE POIDS CORPOREL POUR LUTTER CONTRE L'EXCES DE SECRETION ACIDE GASTRIQUE.
FR8006391A 1979-03-26 1980-03-21 Nouveaux derives d'a-(3,4-dichlorophenyl)-imidazoline ou pyrimidine-2-methane utiles notamment comme agents antisecretoires et leur procede de preparation Granted FR2452486A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/023,920 US4260626A (en) 1979-03-26 1979-03-26 Tetrahydro and imidazoline antisecretory compounds

Publications (2)

Publication Number Publication Date
FR2452486A1 true FR2452486A1 (fr) 1980-10-24
FR2452486B1 FR2452486B1 (fr) 1983-09-16

Family

ID=21817931

Family Applications (1)

Application Number Title Priority Date Filing Date
FR8006391A Granted FR2452486A1 (fr) 1979-03-26 1980-03-21 Nouveaux derives d'a-(3,4-dichlorophenyl)-imidazoline ou pyrimidine-2-methane utiles notamment comme agents antisecretoires et leur procede de preparation

Country Status (21)

Country Link
US (1) US4260626A (fr)
JP (1) JPS55130963A (fr)
AT (1) AT374186B (fr)
AU (1) AU528325B2 (fr)
BE (1) BE882420A (fr)
CA (1) CA1111038A (fr)
CH (1) CH644107A5 (fr)
DE (1) DE3004439A1 (fr)
DK (1) DK155324C (fr)
ES (1) ES487629A0 (fr)
FR (1) FR2452486A1 (fr)
GB (1) GB2045240B (fr)
IE (1) IE49231B1 (fr)
IL (1) IL58934A (fr)
IT (1) IT1143009B (fr)
NL (1) NL7909348A (fr)
NO (1) NO152090C (fr)
NZ (1) NZ192405A (fr)
PH (1) PH15349A (fr)
SE (1) SE446983B (fr)
ZA (1) ZA796743B (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2069481B (en) * 1980-02-13 1983-07-27 Farmos Oy Substituted imidazole derivatives
US6099850A (en) * 1981-10-26 2000-08-08 Battelle Memorial Institute Termite and boring insect barrier for the protection of wooden structures
US6060076A (en) * 1981-10-26 2000-05-09 Battelle Memorial Institute Method and apparatus for providing long term protection from intrusion by insects and other cold blooded animals
US6331308B1 (en) 1981-10-26 2001-12-18 Battelle Memorial Institute Method and apparatus for providing long term protection from intrusion by insects and other cold blooded animals
US5925368A (en) * 1981-10-26 1999-07-20 Battelle Memorial Institute Protection of wooden objects in direct contact with soil from pest invasion
US5272167A (en) * 1986-12-10 1993-12-21 Schering Corporation Pharmaceutically active compounds
US6319511B1 (en) 1989-09-01 2001-11-20 Battelle Memorial Institute Termite and boring insect barrier for the protection of wooden structures
US6572872B2 (en) 1989-09-01 2003-06-03 Battelle Memorial Institute Method and apparatus for providing long term protection from intrusion by insects and other cold blooded animals
US6852328B1 (en) 1989-09-01 2005-02-08 Battelle Memorial Institute K1-53 Method and device for protection of wooden objects proximate soil from pest invasion
US5134154A (en) * 1989-10-20 1992-07-28 Merrell Dow Pharmaceuticals Inc. Phenoxy-heterocyclic compounds
CA2027530C (fr) * 1989-10-20 2001-05-08 Jules Freedman Composes w-phenoxy-heterocycliques
US5985304A (en) * 1998-02-25 1999-11-16 Battelle Memorial Institute Barrier preventing wood pest access to wooden structures
US20020192259A1 (en) * 1998-02-25 2002-12-19 Voris Peter Van Barrier preventing wood pest access to wooden structures
US20060201053A1 (en) * 2000-12-03 2006-09-14 Voris Peter V Barrier preventing wood pest access to wooden structures
US8075910B2 (en) * 2004-05-20 2011-12-13 Pbm Pharmaceuticals, Inc. Oral compositions comprising edible oils and vitamins and/or minerals and methods for making oral compositions

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2207706A1 (fr) * 1972-11-24 1974-06-21 Souchard Maddy

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2919274A (en) * 1957-09-17 1959-12-29 Sahyun Melville Amidines
US3657229A (en) * 1968-05-02 1972-04-18 Sterling Drug Inc 1 3-diaza-2 3-cycloalkene derivatives
US3897431A (en) * 1969-04-24 1975-07-29 Sterling Drug Inc 2-{8 {60 -Alkoxy-arylmethyl{9 -2-imidazolines and -1,4,5,6-tetrahydropyrimidines
US3926994A (en) * 1971-01-11 1975-12-16 Wyeth John & Brother Ltd Heterocyclic compounds
US3996207A (en) * 1971-01-11 1976-12-07 John Wyeth & Brother Limited Derivatives of tetrahydro-1H-1,3-diazepine and hexahydro-1,3-diazocine
CA1010448A (en) 1971-01-11 1977-05-17 John Wyeth And Brother Limited Tetrahydropyrimidine, imidazoline and tetrahydro-1,3-diazepine derivatives
US3965112A (en) * 1971-01-11 1976-06-22 John Wyeth & Brother Limited Imidazoline derivatives
ZA718536B (en) * 1971-01-11 1972-09-27 Wyeth John & Brother Ltd Heterocyclic compounds
US3998842A (en) * 1971-01-11 1976-12-21 John Wyeth & Brother Limited Diazepino[1,2-α]indoles
ZA727999B (en) * 1971-12-06 1973-08-29 Wyeth John & Brother Ltd Derivatives of tetrahydropyrimidine,imidazoline and tetrahydro-1,3-diazepine
GB1538097A (en) * 1976-01-26 1979-01-10 Lafon Labor Substituted phenyl-amidines

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2207706A1 (fr) * 1972-11-24 1974-06-21 Souchard Maddy

Also Published As

Publication number Publication date
DK155324B (da) 1989-03-28
NO800857L (no) 1980-09-29
AT374186B (de) 1984-03-26
DE3004439A1 (de) 1980-12-11
IE49231B1 (en) 1985-09-04
CH644107A5 (de) 1984-07-13
GB2045240B (en) 1982-12-22
SE446983B (sv) 1986-10-20
DK155324C (da) 1989-09-11
BE882420A (fr) 1980-07-16
CA1111038A (fr) 1981-10-20
DE3004439C2 (fr) 1989-05-24
DK101980A (da) 1980-09-27
IE792387L (en) 1980-09-26
NO152090B (no) 1985-04-22
IT8047680A0 (it) 1980-01-23
AU5472880A (en) 1980-10-02
US4260626A (en) 1981-04-07
FR2452486B1 (fr) 1983-09-16
IT1143009B (it) 1986-10-22
ES8100273A1 (es) 1980-11-01
ZA796743B (en) 1980-11-26
AU528325B2 (en) 1983-04-21
ATA144780A (de) 1983-08-15
NO152090C (no) 1985-07-31
NL7909348A (nl) 1980-09-30
GB2045240A (en) 1980-10-29
NZ192405A (en) 1984-07-06
JPH0212949B2 (fr) 1990-03-30
JPS55130963A (en) 1980-10-11
PH15349A (en) 1982-12-02
ES487629A0 (es) 1980-11-01
SE8002293L (sv) 1980-09-27
IL58934A (en) 1984-05-31

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