FR2411181A1 - Derives d'imidazole utiles comme intermediaires de preparation du (r)-3-(2-desoxy-ss-d-erythropentofurannosyl)-3,6,7,8-tetrahydro-imidazol-(4,5-d) (1,3)-diazepin-8-ol - Google Patents
Derives d'imidazole utiles comme intermediaires de preparation du (r)-3-(2-desoxy-ss-d-erythropentofurannosyl)-3,6,7,8-tetrahydro-imidazol-(4,5-d) (1,3)-diazepin-8-olInfo
- Publication number
- FR2411181A1 FR2411181A1 FR7906590A FR7906590A FR2411181A1 FR 2411181 A1 FR2411181 A1 FR 2411181A1 FR 7906590 A FR7906590 A FR 7906590A FR 7906590 A FR7906590 A FR 7906590A FR 2411181 A1 FR2411181 A1 FR 2411181A1
- Authority
- FR
- France
- Prior art keywords
- preparation
- erythropentofurannosyl
- desoxy
- diazepin
- intermediaries
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/052—Imidazole radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/88—Nitrogen atoms, e.g. allantoin
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/91—Nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/91—Nitro radicals
- C07D233/92—Nitro radicals attached in position 4 or 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Saccharide Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
LA PRESENTE INVENTION CONCERNE DE NOUVEAUX DERIVES D'IMIDAZOLE ET UN PROCEDE POUR LEUR PREPARATION. CES NOUVEAUX DERIVES SONT LA 2-AMINO-1-(5-AMINO-1H-IMIDAZOL-4-YL)-ETHANONE DE FORMULE: (CF DESSIN DANS BOPI) ET SES SELS D'ADDITION ACIDE. CES DERIVES SONT UTILES COMME INTERMEDIAIRES DE PREPARATION DU (R)-3-(2-DESOXY-SS-D-ERYTHROPENTOFURANNOSYL)-3,6,7,8-TETRAHYDRO-IMIDAZO-4,5-D 1,3-DIAZEPIN-8-OL.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/841,098 US4117229A (en) | 1977-10-11 | 1977-10-11 | 2-amino-1-(5-amino-1h-imidazol-4-yl)ethanone and method of preparation |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2411181A1 true FR2411181A1 (fr) | 1979-07-06 |
FR2411181B1 FR2411181B1 (fr) | 1981-10-23 |
Family
ID=25284009
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7823597A Granted FR2411207A1 (fr) | 1977-10-11 | 1978-08-10 | Derives d'imidazole, procedes pour leur preparation et transformation de ces derives en (r)-3-(2-desoxy-b-d-erythropentofurannosyl)-3,6,7,8-tetrahydro-imidazol-(4,5-d)-(1,3) diazepin-8-ol |
FR7906591A Granted FR2411191A1 (fr) | 1977-10-11 | 1979-03-15 | Derives d'imidazole-diazepine utiles comme intermediaires de preparation du (r)-3-(2-desoxy-ss-d-erythropentofurannosyl)-2,6,7,8, - tetrahydro - imidazol - /,5-d)(1,3) - diazepin-8-ol |
FR7906590A Granted FR2411181A1 (fr) | 1977-10-11 | 1979-03-15 | Derives d'imidazole utiles comme intermediaires de preparation du (r)-3-(2-desoxy-ss-d-erythropentofurannosyl)-3,6,7,8-tetrahydro-imidazol-(4,5-d) (1,3)-diazepin-8-ol |
Family Applications Before (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7823597A Granted FR2411207A1 (fr) | 1977-10-11 | 1978-08-10 | Derives d'imidazole, procedes pour leur preparation et transformation de ces derives en (r)-3-(2-desoxy-b-d-erythropentofurannosyl)-3,6,7,8-tetrahydro-imidazol-(4,5-d)-(1,3) diazepin-8-ol |
FR7906591A Granted FR2411191A1 (fr) | 1977-10-11 | 1979-03-15 | Derives d'imidazole-diazepine utiles comme intermediaires de preparation du (r)-3-(2-desoxy-ss-d-erythropentofurannosyl)-2,6,7,8, - tetrahydro - imidazol - /,5-d)(1,3) - diazepin-8-ol |
Country Status (11)
Country | Link |
---|---|
US (1) | US4117229A (fr) |
JP (1) | JPS5461177A (fr) |
AU (1) | AU520742B2 (fr) |
CA (1) | CA1109465A (fr) |
DE (1) | DE2835144A1 (fr) |
ES (3) | ES472478A1 (fr) |
FR (3) | FR2411207A1 (fr) |
GB (2) | GB2005661B (fr) |
IT (1) | IT1107776B (fr) |
MY (1) | MY8500742A (fr) |
NL (1) | NL7808365A (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3321023A1 (de) * | 1983-06-10 | 1984-12-13 | Basf Ag, 6700 Ludwigshafen | Triazolylalkohole, verfahren zu ihrer herstellung und ihre verwendung als fungizide |
JPH01250380A (ja) * | 1987-12-26 | 1989-10-05 | Tokyo Tanabe Co Ltd | 光学活性ベンゾキノリジン誘導体、その製造方法およびそれを有効成分とする抗菌剤 |
JPH09241294A (ja) * | 1996-03-07 | 1997-09-16 | Microbial Chem Res Found | 2′−デオキシ−2′−ハロコホルマイシン又はその立体異性体の製造法 |
ES2567152T3 (es) * | 2003-09-15 | 2016-04-20 | Hospira UK Limited | Síntesis y fabricación de pentostatina y sus precursores, análogos y derivados |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3670007A (en) * | 1967-11-21 | 1972-06-13 | Salk Inst For Biological Studi | Aminomalonitrile and method of preparation thereof |
US3923785A (en) * | 1974-04-22 | 1975-12-02 | Parke Davis & Co | (R)-3-(2-deoxy-{62 -D-erythro-pentofuranosyl)-3,6,7,8-tetrahydroimidazo{8 4,5-d{9 {8 1,3{9 diazepin-8-ol |
-
1977
- 1977-10-11 US US05/841,098 patent/US4117229A/en not_active Expired - Lifetime
-
1978
- 1978-08-10 GB GB7832981A patent/GB2005661B/en not_active Expired
- 1978-08-10 FR FR7823597A patent/FR2411207A1/fr active Granted
- 1978-08-10 ES ES472478A patent/ES472478A1/es not_active Expired
- 1978-08-10 JP JP9674878A patent/JPS5461177A/ja active Pending
- 1978-08-10 GB GB7907717A patent/GB2013680B/en not_active Expired
- 1978-08-10 AU AU38816/78A patent/AU520742B2/en not_active Expired
- 1978-08-10 IT IT50697/78A patent/IT1107776B/it active
- 1978-08-10 CA CA309,121A patent/CA1109465A/fr not_active Expired
- 1978-08-10 NL NL7808365A patent/NL7808365A/xx not_active Application Discontinuation
- 1978-08-10 DE DE19782835144 patent/DE2835144A1/de not_active Withdrawn
-
1979
- 1979-03-15 FR FR7906591A patent/FR2411191A1/fr active Granted
- 1979-03-15 FR FR7906590A patent/FR2411181A1/fr active Granted
- 1979-04-16 ES ES479618A patent/ES479618A1/es not_active Expired
- 1979-04-16 ES ES479619A patent/ES479619A0/es active Granted
-
1985
- 1985-12-30 MY MY742/85A patent/MY8500742A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
GB2005661B (en) | 1982-03-10 |
AU520742B2 (en) | 1982-02-25 |
ES8104992A1 (es) | 1981-05-16 |
ES479619A0 (es) | 1981-05-16 |
IT7850697A0 (it) | 1978-08-10 |
NL7808365A (nl) | 1979-04-17 |
ES472478A1 (es) | 1979-10-16 |
ES479618A1 (es) | 1979-08-01 |
DE2835144A1 (de) | 1979-04-12 |
GB2013680A (en) | 1979-08-15 |
CA1109465A (fr) | 1981-09-22 |
FR2411181B1 (fr) | 1981-10-23 |
MY8500742A (en) | 1985-12-31 |
US4117229A (en) | 1978-09-26 |
FR2411191A1 (fr) | 1979-07-06 |
FR2411207A1 (fr) | 1979-07-06 |
FR2411207B1 (fr) | 1982-07-02 |
GB2013680B (en) | 1982-03-31 |
FR2411191B1 (fr) | 1982-02-12 |
JPS5461177A (en) | 1979-05-17 |
GB2005661A (en) | 1979-04-25 |
IT1107776B (it) | 1985-11-25 |
AU3881678A (en) | 1980-02-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |